公开(公告)号：US20200231607A1

公开(公告)日：2020-07-23

申请号：US16610032

申请日：2018-05-02

Applicant: Bayer Aktiengesellschaft ,  Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Jeremy DUFOUR ,  Mathieu GOURGUES ,  Virginie LEMPEREUR ,  Dominique LOQUE ,  Sebastien NAUD ,  Valerie TOQUIN

IPC: C07F7/08 ,  A01N43/42

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to trisubstitutedsilylphenoxyheterocycles and analogues thereof, processes and, intermediates for their preparation as well as use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US20160316752A1

公开(公告)日：2016-11-03

申请号：US15100966

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07D231/16 ,  C07C47/546 ,  C07C47/55 ,  C07C25/18

CPC classification number: A01N43/56 ,  C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07C2601/02 ,  C07D231/16

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基}甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法

公开(公告)号：US20160262393A1

公开(公告)日：2016-09-15

申请号：US15029581

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Peter DAHMEN ,  Philippe DESBORDES ,  Tomoki TSUCHIYA ,  Ulrike WACHENDORFF-NEUMANN ,  Pierre-Yves COQUERON

IPC: A01N43/56 ,  A01N43/72 ,  A01N43/42 ,  A01N43/653

CPC classification number: A01N43/56 ,  A01N43/42 ,  A01N43/653 ,  A01N43/72

Abstract: The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a N-cyclopropyl-N-[substituted-benzyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide or thiocarboxamide derivative and a further fungicidally active compound (B). Moreover, the invention relates to a method for curatively or preventively or eradicatively controlling the phytopathogenic fungi of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.

Abstract translation: 本发明涉及活性化合物组合物，特别是杀真菌剂组合物，其包含（A）N-环丙基-N- [取代 - 苄基] -3-（二氟甲基）-5-氟-1-甲基-1H- 吡唑-4-甲酰胺或硫代羧酰胺衍生物和另外的杀真菌活性化合物（B）。 此外，本发明涉及一种方法，用于根据或预防或根除地控制植物或作物的植物病原真菌，根据本发明的组合用于种子的处理，用于保护种子的方法，至少不是至少 对待处理的种子。

公开(公告)号：US20200079801A1

公开(公告)日：2020-03-12

申请号：US16610093

申请日：2018-05-02

Applicant: Bayer Aktiengesellschaft ,  Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Jeremy DUFOUR ,  Mathieu GOURGUES ,  Virginie LEMPEREUR ,  Sebastien NAUD ,  Valérie TOQUIN

IPC: C07F7/08 ,  A01N55/00

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to trisubstitutedsilylbenzylbenzimidazoles and analogues thereof, processes and intermediates for their preparation as well as use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US20180139962A1

公开(公告)日：2018-05-24

申请号：US15575064

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

CPC classification number: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl derivatives of formula (I), their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20160326120A1

公开(公告)日：2016-11-10

申请号：US15101380

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: C07D231/12 ,  C07D249/06 ,  C07D307/38 ,  C07D263/32 ,  C07C211/27 ,  C07C217/48 ,  C07F7/08 ,  C07C255/46 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C22/04 ,  A01N43/56 ,  A01N43/647 ,  A01N43/10 ,  A01N43/76 ,  A01N33/04 ,  A01N55/00 ,  A01N37/34 ,  A01N35/04 ,  C07D307/54

CPC classification number: C07D231/12 ,  A01N33/04 ,  A01N35/04 ,  A01N37/34 ,  A01N43/10 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N55/00 ,  C07C22/04 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C211/27 ,  C07C217/48 ,  C07C255/46 ,  C07C2601/02 ,  C07D231/14 ,  C07D231/16 ,  C07D233/28 ,  C07D249/06 ,  C07D263/32 ,  C07D307/38 ,  C07D307/54 ,  C07F7/0803

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基]甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法。

公开(公告)号：US20190029255A1

公开(公告)日：2019-01-31

申请号：US16054744

申请日：2018-08-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07C47/55 ,  C07D231/16 ,  C07C25/18 ,  C07C47/546

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substituted cycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20200275656A1

公开(公告)日：2020-09-03

申请号：US16610038

申请日：2018-05-02

Applicant: Bayer Aktiengesellschaft ,  Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Jeremy DUFOUR ,  Mathieu GOURGUES ,  Virginie LEMPEREUR ,  Dominique LOQUE ,  Sebastien NAUD ,  Valérie TOQUIN ,  Andreas GOERTZ ,  Ruth MEISSNER

IPC: A01N43/42 ,  C07D215/20 ,  C07F7/08

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to trisubstitutedsllylmethylphenoxyquinolines and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US20190159452A1

公开(公告)日：2019-05-30

申请号：US15770897

申请日：2016-10-26

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre-Yves COQUERON ,  Pierre CRISTAU ,  Philippe DESBORDES ,  Thomas DRÖGE ,  Ruth MEISSNER

IPC: A01N43/56 ,  A01N43/54 ,  A01N43/653

Abstract: The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a N-cyclopropyl-N-[substituted-benzyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide or thiocarboxamide derivative and at least a further fungicidally active compound (B) consisting of 5-fluoro-4-imino-3-methyl-1-[(4-methylphenyl)sulfonyl]-3,4-dihydropyrimidin-2(1H)-one, 2-[4-(4-chlorophenoxy)-2-(trifluoromethyl)phenyl]-3-methyl-1-(1H-1,2,4-triazol-1-yl)butan-2-ol, (2E,3Z)-5-{[1-(4-chlorophenyl)-1H-pyrazol-3-yl]oxy}-2-(methoxyimino)-N,3-dimethylpent-3-enamide or (2E,3Z)-5-{[1-(4-chloro-2-fluorophenyl)-1H-pyrazol-3-yl]oxy}-2-(methoxyimino)-N,3-dimethylpent-3-enamide

公开(公告)号：US20180146670A1

公开(公告)日：2018-05-31

申请号：US15575292

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D409/12 ,  C07D401/12

CPC classification number: A01N43/56 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.