公开(公告)号：US11219214B2

公开(公告)日：2022-01-11

申请号：US16913862

申请日：2020-06-26

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Philippe Desbordes ,  Christophe Dubost ,  Jeremy Dufour ,  Mathieu Gourgues ,  Philipp Holstein ,  Virginie Lempereur ,  Frederic Miege ,  Philippe Rinolfi ,  Vincent Rodeschini ,  Valerie Toquin ,  Francois Villalba ,  Ulrike Wachendorff-Neumann

IPC: A01N43/42 ,  A01N43/60 ,  C07D215/18 ,  C07D241/44 ,  A01N43/84 ,  A01N43/72 ,  C07D281/06 ,  C07D417/10

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to benzosultams and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US10349656B2

公开(公告)日：2019-07-16

申请号：US15320780

申请日：2015-06-22

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Christophe Dubost ,  Philipp Winter ,  Marco Brünjes ,  Mark James Ford ,  Ulrike Wachendorff-Neumann ,  Cyril Montagne ,  Jean-Pierre Vors ,  Stephane Brunet ,  Philippe Rinolfi

IPC: A01N43/40 ,  C07D213/82

Abstract: The present invention relates to novel difluoromethyl-nicotinic indanyl carboxamides, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials.

公开(公告)号：US10246420B2

公开(公告)日：2019-04-02

申请号：US15327531

申请日：2015-07-21

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Joachim Telser ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Pierre Cristau ,  Philippe Rinolfi

IPC: C07D231/38 ,  C07C331/28 ,  C07C217/76 ,  A01N43/56 ,  C07D401/04

Abstract: The present invention relates to novel pyrazole derivatives, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for controlling harmful microorganisms in crop protection and in the protection of materials. Further, the present invention also relates to certain intermediates useful for producing said novel pyrazole derivatives.

公开(公告)号：US10736321B2

公开(公告)日：2020-08-11

申请号：US16314641

申请日：2017-07-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Philippe Desbordes ,  Christophe Dubost ,  Jeremy Dufour ,  Mathieu Gourgues ,  Philipp Holstein ,  Virginie Lempereur ,  Frederic Miege ,  Philippe Rinolfi ,  Vincent Rodeschini ,  Valerie Toquin ,  Francois Villalba ,  Ulrike Wachendorff-Neumann

IPC: A01N43/42 ,  A01N43/80 ,  C07D417/04 ,  A01N43/84 ,  A01N43/72 ,  C07D281/06 ,  C07D417/10

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to benzosultams and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US10214510B2

公开(公告)日：2019-02-26

申请号：US15566159

申请日：2016-04-12

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Philippe Desbordes ,  Philippe Rinolfi

IPC: C07D401/04 ,  A01N43/46 ,  C07D409/14 ,  C07D405/14 ,  C07D471/04 ,  A01N43/90 ,  C07D401/14 ,  C07D417/14 ,  A01N43/56

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10076116B2

公开(公告)日：2018-09-18

申请号：US15029220

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe Desbordes ,  Philippe Rinolfi ,  Tomoki Tsuchiya ,  Julie Geist ,  Lionel Nicolas

IPC: A01N43/56 ,  C07D403/14 ,  C07D405/14 ,  C07D417/14 ,  A01N43/54 ,  A01N43/647 ,  A01N43/10 ,  A01N43/36 ,  C07D401/14 ,  C07D409/14 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38

CPC classification number: A01N43/56 ,  A01N43/10 ,  A01N43/36 ,  A01N43/54 ,  A01N43/647 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38 ,  C07D401/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylmethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10683311B2

公开(公告)日：2020-06-16

申请号：US15771846

申请日：2016-10-28

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Jérémy Dufour ,  Philippe Desbordes ,  Christophe Dubost ,  Mathieu Gourgues ,  Ruth Meissner ,  Andrew Pettinger ,  Philippe Rinolfi ,  Valérie Toquin ,  Ulrike Wachendorff-Neumann

IPC: C07D215/38 ,  C07F7/08 ,  C07D471/04 ,  C07D495/04 ,  C07D241/44 ,  C07D215/20 ,  C07D401/12 ,  C07D487/04 ,  C07D241/42 ,  A61P31/00 ,  C07D241/18 ,  C07D413/12 ,  C07F7/18

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to trisubstitutedsilylphenoxyhetero-cycles and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US09375010B2

公开(公告)日：2016-06-28

申请号：US14771667

申请日：2014-03-03

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Anne-Sophie Rebstock ,  Christophe Dubost ,  Pierre-Yves Coqueron ,  Simon Maechling ,  Helene Lachaise ,  Philippe Rinolfi ,  Ulrike Wachendorff-Neumann

IPC: C07D417/12 ,  A01N43/50 ,  A01N43/78 ,  A01N43/82 ,  C07D401/12 ,  C07D413/12

CPC classification number: A01N43/82 ,  A01N43/50 ,  A01N43/78 ,  C07D401/12 ,  C07D413/12 ,  C07D417/12

Abstract: The present invention provides 4-substituted-3-{phenyl[(heterocyclylmethoxy)imino]methyl}-1,2,4-oxadiazol-5(4H)-one derivatives of formula (I) Wherein A, X1 to X3, Y1 to Y5 represent various substituents.

Abstract translation: 本发明提供式（I）的4-取代-3- {苯基[（杂环基甲氧基）亚氨基]甲基} -1,2,4-恶二唑-5（4H） - 酮衍生物，其中A，X1至X3，Y1至 Y 5表示各种取代基。

公开(公告)号：US10244757B2

公开(公告)日：2019-04-02

申请号：US16054744

申请日：2018-08-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan-Peter Schmidt ,  Tomoki Tsuchiya ,  Jean-Pierre Vors ,  Ulrike Wachendorff-Neumann

IPC: C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07D231/16 ,  A01N43/56

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10244756B2

公开(公告)日：2019-04-02

申请号：US15575292

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan Peter Schmidt ,  Tomoki Tsuchiya

IPC: A01N43/56 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.