公开(公告)号：US10244757B2

公开(公告)日：2019-04-02

申请号：US16054744

申请日：2018-08-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan-Peter Schmidt ,  Tomoki Tsuchiya ,  Jean-Pierre Vors ,  Ulrike Wachendorff-Neumann

IPC: C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07D231/16 ,  A01N43/56

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10244756B2

公开(公告)日：2019-04-02

申请号：US15575292

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan Peter Schmidt ,  Tomoki Tsuchiya

IPC: A01N43/56 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.

公开(公告)号：US11213031B2

公开(公告)日：2022-01-04

申请号：US16762615

申请日：2018-11-08

Applicant: BAYER AKTIENGESELLSCHAFT ,  BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Alexander Sudau ,  Sebastian Hoffmann ,  Peter Dahmen ,  Robert Alan Webster ,  Ruth Meissner ,  Andreas Goertz ,  Ricarda Miller ,  Pierre-Yves Coqueron ,  David Bernier ,  Lionel Nicolas ,  Stephane Brunet ,  Philippe Kennel ,  Valerie Toquin ,  Mathieu Gourgues ,  Dominique Loque ,  Vincent Thomas

IPC: A01N43/713 ,  C07D257/04

Abstract: The present invention relates to tetrazolylpropyl derivatives of formula (I) wherein one of V1 and V2 represents CR3 and the other one of V1 and V2 represents N, Q represents a 6-membered aromatic cycle as defined in the specification, and R1, R2, R3, R4, and R5 are defined as disclosed in the specification, to compositions comprising such compounds, to the use of said compounds as fungicides, as well as to particular intermediates useful in the synthesis of said tetrazolylpropyl derivatives.

公开(公告)号：US10071967B2

公开(公告)日：2018-09-11

申请号：US15101380

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan-Peter Schmidt ,  Tomoki Tsuchiya ,  Jean-Pierre Vors ,  Ulrike Wachendorff-Neumann

IPC: C07D231/12 ,  A01N33/04 ,  C07D231/14 ,  C07D231/16 ,  C07D233/28 ,  A01N35/04 ,  A01N37/34 ,  A01N43/10 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N55/00 ,  C07C22/04 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C211/27 ,  C07C217/48 ,  C07C255/46 ,  C07D249/06 ,  C07D263/32 ,  C07D307/38 ,  C07D307/54 ,  C07F7/08

CPC classification number: C07D231/12 ,  A01N33/04 ,  A01N35/04 ,  A01N37/34 ,  A01N43/10 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N55/00 ,  C07C22/04 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C211/27 ,  C07C217/48 ,  C07C255/46 ,  C07C2601/02 ,  C07D231/14 ,  C07D231/16 ,  C07D233/28 ,  C07D249/06 ,  C07D263/32 ,  C07D307/38 ,  C07D307/54 ,  C07F7/0803

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10070645B2

公开(公告)日：2018-09-11

申请号：US15100966

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre Cristau ,  Philippe Desbordes ,  Julie Geist ,  Lionel Nicolas ,  Philippe Rinolfi ,  Jan-Peter Schmidt ,  Tomoki Tsuchiya ,  Jean-Pierre Vors ,  Ulrike Wachendorff-Neumann

IPC: A01N43/56 ,  C07D231/16 ,  C07C47/575 ,  C07C47/55 ,  C07C25/18 ,  C07C47/546

CPC classification number: A01N43/56 ,  C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07C2601/02 ,  C07D231/16

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US10076116B2

公开(公告)日：2018-09-18

申请号：US15029220

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe Desbordes ,  Philippe Rinolfi ,  Tomoki Tsuchiya ,  Julie Geist ,  Lionel Nicolas

IPC: A01N43/56 ,  C07D403/14 ,  C07D405/14 ,  C07D417/14 ,  A01N43/54 ,  A01N43/647 ,  A01N43/10 ,  A01N43/36 ,  C07D401/14 ,  C07D409/14 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38

CPC classification number: A01N43/56 ,  A01N43/10 ,  A01N43/36 ,  A01N43/54 ,  A01N43/647 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38 ,  C07D401/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylmethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.