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1.发明授权公开(公告)号：US07208506B2
公开(公告)日：2007-04-24
申请号：US11477641
申请日：2006-06-29
申请人： Edward Boyd , Frederick Brookfield , Jonathan Gridley , Manfred Kubbies , Raymond Lau , Ulrike Reiff , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt , Timothy Woodcock
发明人： Edward Boyd , Frederick Brookfield , Jonathan Gridley , Manfred Kubbies , Raymond Lau , Ulrike Reiff , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt , Timothy Woodcock
IPC分类号： A61K31/38 , A61K31/42 , A61K31/425 , A61K31/44
CPC分类号： A61K31/38 , A61K31/381 , A61K31/44 , C07D213/59 , C07D333/24
摘要： The present invention relates to compounds of formula I wherein R1, R2 and R3 are defined herein, their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of the above compounds, medicaments containing them and their manufacture, as well as the use of the above compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明涉及式I化合物，其中R 1，R 2和R 3 3定义为其药学上可接受的盐，对映体形式 ，非对映异构体和外消旋物，上述化合物的制备，含有它们的药物及其制备，以及上述化合物在控制或预防诸如癌症等疾病中的用途。
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公开(公告)号：US20070010564A1
公开(公告)日：2007-01-11
申请号：US11477641
申请日：2006-06-29
申请人： Edward Boyd , Frederick Brookfield , Jonathan Gridley , Manfred Kubbies , Raymond Lau , Ulrike Reiff , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt , Timothy Woodcock
发明人： Edward Boyd , Frederick Brookfield , Jonathan Gridley , Manfred Kubbies , Raymond Lau , Ulrike Reiff , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt , Timothy Woodcock
IPC分类号： A61K31/44 , A61K31/381 , C07D333/22 , C07D213/56
CPC分类号： A61K31/38 , A61K31/381 , A61K31/44 , C07D213/59 , C07D333/24
摘要： The present invention relates to compounds of formula I wherein R1, R2 and R3 are defined herein, their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of the above compounds, medicaments containing them and their manufacture, as well as the use of the above compounds in the control or prevention of illnesses such as cancer.
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3.发明申请HETEROCYCLYL PYRIDYL SULFONAMIDE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS 失效间苯二酚吡啶酰胺衍生物及其制备和用作药物代理公开(公告)号：US20100292247A1
公开(公告)日：2010-11-18
申请号：US12377911
申请日：2007-10-24
申请人： Frederick Brookfield , Jonathan Gridley , Lothar Kling , Michael Prime , Ulrike Reiff , Wolfgang von der Saal , Thomas von Hirschheydt
发明人： Frederick Brookfield , Jonathan Gridley , Lothar Kling , Michael Prime , Ulrike Reiff , Wolfgang von der Saal , Thomas von Hirschheydt
IPC分类号： A61K31/496 , C07D401/14 , C07D401/04 , C07D491/113 , A61K31/438 , A61P35/00
CPC分类号： C07D295/04
摘要： Objects of the present invention are the compounds of formula I, their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of the above compounds, medicaments containing them and their manufacture, as well as the use of the above compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明的目的是式I化合物，其药学上可接受的盐，对映体形式，非对映异构体和外消旋体，上述化合物的制备，含有它们的药物及其制备，以及上述化合物在对照中的用途 或预防癌症等疾病。
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公开(公告)号：US20070123513A1
公开(公告)日：2007-05-31
申请号：US11594297
申请日：2006-11-08
申请人： Lothar Kling , Ulrike Reiff , Manfred Schwaiger , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt
发明人： Lothar Kling , Ulrike Reiff , Manfred Schwaiger , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt
IPC分类号： A61K31/55 , A61K31/4439 , A61K31/4412 , A61K31/4545 , C07D213/63
CPC分类号： C07D213/71
摘要： The present invention relates to the compounds of formula I: their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of such compounds, pharmaceutical compositions containing them and their manufacture, as well as the use of such compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明涉及式I化合物：其药学上可接受的盐，对映体形式，非对映异构体和外消旋体，这些化合物的制备，含有它们的药物组合物及其制备，以及这些化合物在控制或预防中的用途 的疾病，如癌症。
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公开(公告)号：US07625896B2
公开(公告)日：2009-12-01
申请号：US11594297
申请日：2006-11-08
申请人： Lothar Kling , Ulrike Reiff , Manfred Schwaiger , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt
发明人： Lothar Kling , Ulrike Reiff , Manfred Schwaiger , Georg Tiefenthaler , Wolfgang von der Saal , Thomas von Hirschheydt
IPC分类号： A61K31/535 , C07D413/00 , A61K31/445 , C07D211/68 , C07D401/00 , A61K31/44
CPC分类号： C07D213/71
摘要： The present invention relates to the compounds of formula I: their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of such compounds, pharmaceutical compositions containing them and their manufacture, as well as the use of such compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明涉及式I化合物：其药学上可接受的盐，对映体形式，非对映异构体和外消旋体，这些化合物的制备，含有它们的药物组合物及其制备，以及这些化合物在控制或预防中的用途 的疾病，如癌症。
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6.发明申请Pyrazole Derivatives, Their Manufacture and Their Use as Pharmaceutical Agents 审中-公开吡唑衍生物，其制造及其作为药剂的用途公开(公告)号：US20090264485A1
公开(公告)日：2009-10-22
申请号：US11989218
申请日：2006-08-07
IPC分类号： A61K31/422 , C07D413/12 , A61P35/00
CPC分类号： C07D413/12
摘要： Objects of the present invention are the compounds of formula I their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of the above-mentioned compounds, pharmaceutical compositions containing them and their manufacture, as well as the use of the above-mentioned compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明的目的是式I化合物，其药学上可接受的盐，对映异构体形式，非对映异构体和外消旋物，上述化合物的制备，含有它们的药物组合物及其制备方法以及使用上述 控制或预防疾病如癌症的化合物。
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公开(公告)号：US20060211750A1
公开(公告)日：2006-09-21
申请号：US11226677
申请日：2005-09-14
IPC分类号： A61K31/422 , C07D413/02
CPC分类号： C07D413/12
摘要： The present invention relates to the compounds of formula I their pharmaceutically acceptable salts or esters, enantiomeric forms, diastereoisomers and racemates, the preparation of the above-mentioned compounds, compositions containing such compounds and their manufacture, as well as the use of such compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明涉及式I化合物的药学上可接受的盐或酯，对映体形式，非对映异构体和外消旋物，上述化合物的制备，含有这些化合物的组合物及其制备方法以及这些化合物在 控制或预防癌症等疾病。
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公开(公告)号：US20060069095A1
公开(公告)日：2006-03-30
申请号：US11232303
申请日：2005-09-21
IPC分类号： A61K31/5377 , A61K31/422 , C07D413/02 , C07D413/14
CPC分类号： C07D413/12
摘要： Compounds of formula I their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, are disclosed. Also disclosed are methods of preparation of the above-mentioned compounds, pharmaceutical compositions and salts and esters thereof containing them, as well as the use of the above-mentioned compounds in the treatment, control or prevention of illnesses such as cancer.
摘要翻译： 式I化合物
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公开(公告)号：US07288557B2
公开(公告)日：2007-10-30
申请号：US11226677
申请日：2005-09-14
IPC分类号： A61K31/422 , C07D263/32
CPC分类号： C07D413/12
摘要： The present invention relates to the compounds of formula I their pharmaceutically acceptable salts or esters, enantiomeric forms, diastereoisomers and racemates, the preparation of the above-mentioned compounds, compositions containing such compounds and their manufacture, as well as the use of such compounds in the control or prevention of illnesses such as cancer.
摘要翻译： 本发明涉及式I化合物的药学上可接受的盐或酯，对映体形式，非对映异构体和外消旋体，上述化合物的制备，含有这些化合物的组合物及其制备方法以及这些化合物在 控制或预防癌症等疾病。
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公开(公告)号：US20050113342A1
公开(公告)日：2005-05-26
申请号：US10961907
申请日：2004-10-12
IPC分类号： C07D401/14 , C07D403/04 , A61K31/675 , A61K31/506 , C07F9/6512 , C07D43/04
CPC分类号： C07D401/14 , C07D403/04
摘要： Compounds of the general formula (I) are presented which arevaluable therapeutics for the treatment of cancer and cancer related diseases.
摘要翻译： 提出了通式（I）的化合物，其用于治疗癌症和癌症相关疾病的有价值的治疗剂。
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