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公开(公告)号:US07279582B2
公开(公告)日:2007-10-09
申请号:US10280652
申请日:2002-10-25
申请人: Eric J. Stoner , Arthur J. Cooper , Lawrence Kolaczkowski , Ketan M. Patel , Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Daniel A. Dickman , Patricia A. Oliver , Jien-Heh J. Tien
发明人: Eric J. Stoner , Arthur J. Cooper , Lawrence Kolaczkowski , Ketan M. Patel , Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Daniel A. Dickman , Patricia A. Oliver , Jien-Heh J. Tien
IPC分类号: C07D233/32 , C07D239/10 , C07D239/12
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
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公开(公告)号:US07968707B2
公开(公告)日:2011-06-28
申请号:US11679227
申请日:2007-02-27
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D219/04 , C07D291/06 , C07D243/04 , C07D265/12 , C07D413/12 , C07D239/02
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
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公开(公告)号:US06472529B2
公开(公告)日:2002-10-29
申请号:US09837280
申请日:2001-04-18
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D23332
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
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公开(公告)号:US06313296B1
公开(公告)日:2001-11-06
申请号:US09511390
申请日:2000-02-23
申请人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
发明人: Hing Leung Sham , Daniel W. Norbeck , Xiaoqi Chen , David A. Betebenner , Dale J. Kempf , Thomas R. Herrin , Gondi N. Kumar , Stephen L. Condon , Arthur J. Cooper , Daniel A. Dickman , Steven M. Hannick , Lawrence Kolaczkowski , Patricia A. Oliver , Daniel J. Plata , Peter J. Stengel , Eric J. Stoner , Jieh-Heh J. Tien , Jih-Hua Liu , Ketan M. Patel
IPC分类号: C07D23902
CPC分类号: C07D207/27 , C07D207/404 , C07D207/408 , C07D223/10 , C07D233/32 , C07D233/42 , C07D239/10 , C07D239/22 , C07D241/08 , C07D241/18 , C07D253/06 , C07D263/22 , C07D307/20 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D417/12
摘要: A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.
摘要翻译: 公开了下式的化合物作为HIV蛋白酶抑制剂。 还公开了用于抑制HIV感染的方法和组合物。
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公开(公告)号:US6022989A
公开(公告)日:2000-02-08
申请号:US671893
申请日:1996-06-28
申请人: Patricia A. Oliver , Arthur J. Cooper , Joseph B. Paterson, Jr. , Denton C. Langridge , Jieh-Heh J. Tien
发明人: Patricia A. Oliver , Arthur J. Cooper , Joseph B. Paterson, Jr. , Denton C. Langridge , Jieh-Heh J. Tien
IPC分类号: C07D277/28 , C07C269/04 , C07C271/54 , C07C261/00
CPC分类号: C07C269/04
摘要: A process is disclosed for the preparation of an N-acylated activated derivative of an amino acid or a salt thereof.
摘要翻译: 公开了制备氨基酸或其盐的N-酰化活化衍生物的方法。
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公开(公告)号:US6160122A
公开(公告)日:2000-12-12
申请号:US673445
申请日:1996-06-28
申请人: Patricia A. Oliver , Arthur J. Cooper , John E. Lallaman , Denton C. Langridge , Jieh-Heh J. Tien
发明人: Patricia A. Oliver , Arthur J. Cooper , John E. Lallaman , Denton C. Langridge , Jieh-Heh J. Tien
IPC分类号: C07D277/28 , C07D277/30
CPC分类号: C07D277/28
摘要: A process is disclosed for the preparation of N-((N-Methyl-N-((2-isopropyl-4-thiazolyl)methyl)amino)carbonyl)-amino acid derivatives.
摘要翻译: 公开了制备N - ((N-甲基-N - ((2-异丙基-4-噻唑基)甲基)氨基)羰基) - 氨基酸衍生物的方法。
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