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1.发明申请SULFONAMIDE SUBSTITUTED PYRAZOLINE COMPOUNDS, THEIR PREPARATION AND USE AS CB1 MODULATORS 失效磺酰胺取代的吡咯啉化合物，其制备和用作CB1调节剂公开(公告)号：US20100184772A1
公开(公告)日：2010-07-22
申请号：US12445260
申请日：2007-10-10
IPC分类号： C07D231/06 , A61K31/415 , A61K31/4178 , C07D403/12 , C07D409/12 , A61K31/4155 , A61K31/428 , C07D417/12 , C07D405/12 , C07D413/12 , A61K31/422 , A61K31/513 , C07D401/12 , A61K31/4709 , A61K31/4439 , A61K31/4245 , A61K31/433 , A61K31/427 , A61K31/4725 , A61K31/498 , C07D513/04 , A61K31/429 , A61P5/00 , A61P9/00 , A61P11/00 , A61P25/00 , A61P37/00 , A61P15/00 , A61P1/00 , A61P35/00 , A61P19/00 , A61P3/00
CPC分类号： C07D231/06 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D513/04
摘要： The present invention relates to substituted pyrazoline compounds of general formula (I), methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及通式（I）的取代吡唑啉化合物，其制备方法，包含这些化合物的药物及其制备用于治疗人和动物的药物的用途。
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2.发明授权Sulfonamide substituted pyrazoline compounds, their preparation and use as CB1 modulators 失效磺酰胺取代的吡唑啉化合物，其制备和用作CB1调节剂公开(公告)号：US08044053B2
公开(公告)日：2011-10-25
申请号：US12445260
申请日：2007-10-10
IPC分类号： A61K31/501 , A61K31/496 , A61K31/497 , A61K31/437 , A61K31/4523 , A61K31/415 , A61K31/4178 , A61K31/4245 , A61K31/426 , A61K31/433 , C07D237/02 , C07D239/02 , C07D241/02 , C07D221/02 , C07D221/00 , C07D401/02 , C07D277/20 , C07D263/30 , C07D271/08 , C07D285/10 , C07D233/54 , C07D231/10
CPC分类号： C07D231/06 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D513/04
摘要： The present invention relates to substituted pyrazoline compounds of general formula (I), methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及通式（I）的取代吡唑啉化合物，其制备方法，包含这些化合物的药物及其制备用于治疗人和动物的药物的用途。
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3.发明授权公开(公告)号：US07829581B2
公开(公告)日：2010-11-09
申请号：US11995708
申请日：2006-07-17
IPC分类号： A61K31/454 , A61K31/4155 , C07D401/02 , C07D403/02
CPC分类号： C07D231/06 , C07D403/12
摘要： The present invention relates to prodrugs of pyrazoline compounds of formula I, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及式I的吡唑啉化合物的前药，其制备方法，包含这些化合物的药物及其用于制备用于治疗人和动物的药物的用途。
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4.发明申请SUBSTITUTED PYRAZOLINE COMPOUNDS WITH ACAT INHIBITION ACTIVITY, THEIR PREPARATION AND USE AS MEDICAMENTS 审中-公开具有ACAT抑制活性的取代的吡唑化合物，其制备和用作药物公开(公告)号：US20100069364A1
公开(公告)日：2010-03-18
申请号：US12523451
申请日：2008-01-17
IPC分类号： C07D231/06 , A61K31/415 , A61K31/55 , C07D401/12 , A61K31/454 , A61P3/00 , A61P3/10 , A61P3/06
CPC分类号： C07D231/06
摘要： The present invention relates to substituted pyrazoline compounds, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals, especially in dyslipidaemia.
摘要翻译： 本发明涉及取代的吡唑啉化合物，其制备方法，包含这些化合物的药物及其用于制备用于治疗人和动物，特别是血脂异常的药物的用途。
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5.发明申请公开(公告)号：US20080300278A1
公开(公告)日：2008-12-04
申请号：US11995708
申请日：2006-07-17
IPC分类号： A61K31/415 , A61P25/00 , A61P37/00 , A61P9/00 , A61P11/00 , A61P1/00 , A61P3/00 , A61P35/00 , C07D403/12 , C07D401/02 , C07D231/06 , A61K31/454
CPC分类号： C07D231/06 , C07D403/12
摘要： The present invention relates to prodrugs of pyrazoline compounds of formula I, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及式I的吡唑啉化合物的前药，其制备方法，包含这些化合物的药物及其用于制备用于治疗人和动物的药物的用途。
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公开(公告)号：US20090318524A1
公开(公告)日：2009-12-24
申请号：US12226559
申请日：2007-04-30
申请人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
发明人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
IPC分类号： C07D209/52 , A61K31/403 , A61P3/06 , A61P29/00 , A61P1/00 , A61P25/28 , A61P19/02 , A61P9/00 , A61P25/30
CPC分类号： A61K31/403 , C07D209/52 , C07D209/94
摘要： The present invention relates to substituted bicyclic tetrahydropyrrole compounds of general formula (I), methods for their preparation, medicaments comprising these compounds as well their use in the manufacture of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及通式（I）的取代的双环四氢吡咯化合物，其制备方法，包含这些化合物的药物及其在制备用于治疗人和动物的药物中的用途。
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公开(公告)号：US20090306403A1
公开(公告)日：2009-12-10
申请号：US12226310
申请日：2007-04-30
申请人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
发明人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
IPC分类号： C07F7/02 , C07D209/52
CPC分类号： C07D209/52
摘要： The present invention relates to a process using the Pauson-Khand Reaction to produce substituted bicyclic tetrahydropyrrole compounds of general formula (I)
摘要翻译： 本发明涉及使用Pauson-Khand反应制备通式（I）的取代的双环四氢吡咯化合物的方法，
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公开(公告)号：US08372990B2
公开(公告)日：2013-02-12
申请号：US12226559
申请日：2007-04-30
申请人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
发明人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobés , Carmen Garcia Granda
IPC分类号： C07D209/52 , A61K31/403 , A61P3/06 , A61P29/00 , A61P1/00 , A61P25/28 , A61P19/02 , A61P9/00 , A61P25/30
CPC分类号： A61K31/403 , C07D209/52 , C07D209/94
摘要： The present invention relates to substituted bicyclic tetrahydropyrrole compounds of general formula (I), methods for their preparation, medicaments comprising these compounds as well their use in the manufacture of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及通式（I）的取代的双环四氢吡咯化合物，其制备方法，包含这些化合物的药物及其在制备用于治疗人和动物的药物中的用途。
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公开(公告)号：US08299113B2
公开(公告)日：2012-10-30
申请号：US12226626
申请日：2007-04-30
申请人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobes , Carmen Garcia Granda
发明人： Miguel Angel Pericas-Brondo , Antonio Torrens-Jover , Susana Yenes-Minguez , Félix Cuevas Cordobes , Carmen Garcia Granda
IPC分类号： A01N43/38 , A61K31/40 , C07D209/00
CPC分类号： C07D209/52 , C07D207/20
摘要： The present invention relates to substituted bicyclic tetrahydropyrrole compounds of general formula (I), methods for their preparation, medicaments comprising these compounds as well their use in the manufacture of a medicament for the treatment of humans and animals.
摘要翻译： 本发明涉及通式（I）的取代的双环四氢吡咯化合物，其制备方法，包含这些化合物的药物及其在制备用于治疗人和动物的药物中的用途。
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公开(公告)号：US20100099712A1
公开(公告)日：2010-04-22
申请号：US12523394
申请日：2008-01-17
IPC分类号： A61K31/454 , C07D401/12 , C07D231/06 , A61K31/415 , A61P3/10 , A61P3/06
CPC分类号： C07D401/12 , C07D231/06
摘要： The present invention relates to substituted pyrazoline compounds, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals, especially in dyslipidaemia.
摘要翻译： 本发明涉及取代的吡唑啉化合物，其制备方法，包含这些化合物的药物及其用于制备用于治疗人和动物，特别是血脂异常的药物的用途。
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