-
公开(公告)号:USD695283S1
公开(公告)日:2013-12-10
申请号:US29406400
申请日:2011-11-14
申请人: Igor Duc , John Brunner
设计人: Igor Duc , John Brunner
-
公开(公告)号:USD679674S1
公开(公告)日:2013-04-09
申请号:US29408210
申请日:2011-12-08
申请人: Igor Duc , John Brunner
设计人: Igor Duc , John Brunner
-
3.Indazoles, benzisoxazoles and benzisothiazoles and their use as estrogenic agents 有权
标题翻译: 吲唑,苯并异恶唑和苯并异噻唑及其作为雌激素剂的用途公开(公告)号:US07977364B2
公开(公告)日:2011-07-12
申请号:US11664887
申请日:2005-10-14
申请人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
发明人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
IPC分类号: A61K31/423 , A61K31/416 , C07D261/20 , C07D231/56
CPC分类号: C07D231/56 , C07D261/20 , C07D275/04 , C07D275/06 , C07D491/06
摘要: The present invention relates to compounds of formula (I): in which R1, R2, R3, X, Y and A are as defined in the specification. The compounds are modulators of the estrogen receptors.
摘要翻译: 本发明涉及式(I)化合物:其中R1,R2,R3,X,Y和A如说明书中所定义。 这些化合物是雌激素受体的调节剂。
-
4.1-N-phenyl-amino-1h-imidazole derivatives and pharmaceutical compositions containing them 失效
标题翻译: 1-N-苯基 - 氨基-1h-咪唑衍生物和含有它们的药物组合物公开(公告)号:US20070112009A1
公开(公告)日:2007-05-17
申请号:US10582778
申请日:2004-12-15
申请人: Jean Lafay , Benoit Rondot , Paule Bonnet , Thierry Clerc , Jaqueline Shields , Igor Duc , Eric Duranti , Francois Puccio , Christian Blot , Philippe Maillos
发明人: Jean Lafay , Benoit Rondot , Paule Bonnet , Thierry Clerc , Jaqueline Shields , Igor Duc , Eric Duranti , Francois Puccio , Christian Blot , Philippe Maillos
IPC分类号: A61K31/513 , A61K31/497 , A61K31/4152 , A61K31/501 , A61K31/4439 , C07D409/02 , C07D403/02
CPC分类号: C07D233/54 , C07D409/12 , C07D419/12
摘要: The invention relates to the compounds of formula (I): in which R1, R2, R3, R4, Q and Z are as defined in the specification. The invention also relates to the pharmaceutical compositions containing these compounds.
摘要翻译: 本发明涉及式(I)化合物:其中R 1,R 2,R 3,R 4, / SUB,Q和Z如说明书中所定义。 本发明还涉及含有这些化合物的药物组合物。
-
5.1-N-phenyl-amino-1h-imidazole derivatives and pharmaceutical compositions containing them 失效
标题翻译: 1-N-苯基 - 氨基-1h-咪唑衍生物和含有它们的药物组合物公开(公告)号:US08476455B2
公开(公告)日:2013-07-02
申请号:US10582778
申请日:2004-12-15
申请人: Jean Lafay , Benoit Rondot , Paule Bonnet , Thierry Clerc , Jacqueline Shields , Igor Duc , Eric Duranti , Francois Puccio , Christian Blot , Philippe Maillos
发明人: Jean Lafay , Benoit Rondot , Paule Bonnet , Thierry Clerc , Jacqueline Shields , Igor Duc , Eric Duranti , Francois Puccio , Christian Blot , Philippe Maillos
IPC分类号: C07D233/44 , A61K31/4164
CPC分类号: C07D233/54 , C07D409/12 , C07D419/12
摘要: The invention relates to the compounds of formula (I): in which R1, R2, R3, R4, Q and Z are as defined in the specification. The invention also relates to the pharmaceutical compositions containing these compounds.
摘要翻译: 本发明涉及式(I)化合物:其中R1,R2,R3,R4,Q和Z如说明书中所定义。 本发明还涉及含有这些化合物的药物组合物。
-
6.Indazoles, benzisoxazoles and benzisothiazoles and their use as estrogenic agents 有权
标题翻译: 吲唑,苯并异恶唑和苯并异噻唑及其作为雌激素剂的用途公开(公告)号:US20090023779A1
公开(公告)日:2009-01-22
申请号:US11664887
申请日:2005-10-14
申请人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
发明人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
IPC分类号: C07D231/56 , A61K31/416 , C07D413/02 , A61K31/454 , A61K31/42 , C07D261/20 , C07D275/04 , A61K31/428 , A61P35/00
CPC分类号: C07D231/56 , C07D261/20 , C07D275/04 , C07D275/06 , C07D491/06
摘要: The present invention relates to compounds of formula (I): in which R1, R2, R3, X, Y and A are as defined in the specification.The compounds are modulators of the estrogen receptors.
摘要翻译: 本发明涉及式(I)化合物:其中R1,R2,R3,X,Y和A如说明书中所定义。 这些化合物是雌激素受体的调节剂。
-
7.Indazoles, benzisoxazoles and benzisothiazoles and their use as estrogenic agents 失效
标题翻译: 吲唑,苯并异恶唑和苯并异噻唑及其作为雌激素剂的用途公开(公告)号:US08173679B2
公开(公告)日:2012-05-08
申请号:US13152433
申请日:2011-06-03
申请人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
发明人: Benoit Rondot , Jean Lafay , Paule Bonnet , Thierry Clerc , Igor Duc , Eric Duranti , Francois Puccio , Jacqueline Shields , Christian Blot , Philippe Maillos
IPC分类号: A61K31/454 , A61K31/428 , A61K31/423 , A61K31/416 , C07D261/20 , C07D401/06 , C07D275/04 , C07D413/12 , C07D231/56
CPC分类号: C07D231/56 , C07D261/20 , C07D275/04 , C07D275/06 , C07D491/06
摘要: The present invention relates to compounds of formula (I): in which R1, R2, R3, X, Y and A are as defined in the specification. The compounds are modulators of the estrogen receptors.
摘要翻译: 本发明涉及式(I)化合物:其中R1,R2,R3,X,Y和A如说明书中所定义。 这些化合物是雌激素受体的调节剂。
-
8.Sulfamate benzothiophene derivatives as steroid sulfatase inhibitors 失效
标题翻译: 磺胺基苯并噻吩衍生物作为类固醇硫酸酯酶抑制剂公开(公告)号:US07476691B2
公开(公告)日:2009-01-13
申请号:US10555780
申请日:2003-05-16
申请人: Jean Lafay , Benoît Rondot , Denis Carniato , Paule Bonnet , Thierry Clerc , Jacqueline Shields , Igor Duc , Eric Duranti
发明人: Jean Lafay , Benoît Rondot , Denis Carniato , Paule Bonnet , Thierry Clerc , Jacqueline Shields , Igor Duc , Eric Duranti
IPC分类号: A61K31/381 , C07D333/64 , C07D333/66
CPC分类号: C07D333/54 , C07D333/76
摘要: The present invention relates to sulfamate benzothiophene compounds of the formula: (I) wherein R1, R2, R3, m and n are as defined in the specification. The invention also relates to pharmaceutical compositions containing these compounds and to methods of using them.
摘要翻译: 本发明涉及式(I)的氨基磺酸苯并噻吩化合物,其中R 1,R 2,R 3,m和n如说明书中所定义。 本发明还涉及含有这些化合物的药物组合物及其使用方法。
-
-
-
-
-
-
-