Pyrimidine derivatives, process for preparing the same and herbicide
using the same
    1.
    发明授权
    Pyrimidine derivatives, process for preparing the same and herbicide using the same 失效
    嘧啶衍生物,其制备方法和使用其的除草剂

    公开(公告)号:US5387575A

    公开(公告)日:1995-02-07

    申请号:US894557

    申请日:1992-06-05

    摘要: Disclosed are a pyrimidine or triazine compound represented by the following formula (I): ##STR1## wherein R.sup.1 represents cyano group, a halogen atom, hydroxy group or --O--R.sup.7 where R.sup.7 represents a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a halo-lower alkyl group or a cyano-lower alkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom or a lower alkyl group; R.sup.4 represents a 1-imidazolyl group, --NHSO.sub.2 --R.sup.8 where R.sup.8 represents a lower alkyl group or a phenyl group which may have a substituent, hydroxy group, a lower alkoxy group or a benzyloxy group when Z is nitrogen atom; or a 1-imidazolyl group, --NHSO.sub.2 --R.sup.8 where R.sup.8 has the same meaning as defined above, hydroxy group, OK, a lower alkoxy group which may have a substituent, a lower alkenyloxy group, a lower alkynyloxy group, a cycloalkoxy group which may have a substituent, a phenoxy group, a benzyloxy group, a lower alkylthio group, a phenylthio group or an alkylsulfonylamino group when Z is --CH.dbd. group; R.sup.5 represents a lower alkoxy group; R.sup.6 represents a lower alkoxy group or a lower alkyl group; X represents oxygen atom or sulfur atom; and Z represents nitrogen atom or --CH.dbd. group. processes for preparing the same and a herbicide containing the same as an active ingredient(s).

    摘要翻译: 公开了由下式(I)表示的嘧啶或三嗪化合物:其中R 7表示低级烷基,低级烯基,低级炔基,卤代烷基, 低级烷基或氰基 - 低级烷基; R2代表氢原子或低级烷基; R3表示氢原子或低级烷基; R 4表示当Z为氮原子时,可以具有取代基,羟基,低级烷氧基或苄氧基的低级烷基或苯基,-NHSO 2 -R 8, 或1-咪唑基,-NHSO 2 -R 8,其中R8具有与上述相同的含义,羟基,OK,可具有取代基的低级烷氧基,低级链烯氧基,低级炔氧基,环烷氧基 当Z为-CH =基团时,可具有取代基,苯氧基,苄氧基,低级烷硫基,苯硫基或烷基磺酰基氨基; R5代表低级烷氧基; R6代表低级烷氧基或低级烷基; X表示氧原子或硫原子; Z表示氮原子或-CH =基团。 其制备方法和含有其作为活性成分的除草剂。

    Triazine derivative, process for preparing the same and herbicide using
the same
    2.
    发明授权
    Triazine derivative, process for preparing the same and herbicide using the same 失效
    三嗪衍生物,其制备方法和使用其的除草剂

    公开(公告)号:US5529977A

    公开(公告)日:1996-06-25

    申请号:US326830

    申请日:1994-10-21

    摘要: Disclosed are a pyrimidine or triazine compound represented by the following formula (I): ##STR1## wherein R.sup.1 represents cyano group, a halogen atom, hydroxy group or --O--R.sup.7 where R.sup.7 represents a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a halo-lower alkyl group or a cyano-lower alkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom or a lower alkyl group; R.sup.4 represents a 1-imidazolyl group, --NHSO.sub.2 --R.sup.8 where R.sup.8 represents a lower alkyl group or a phenyl group which may have a substituent, hydroxy group, a lower alkoxy group or a benzyloxy group when Z is nitrogen atom; or a 1-imidazolyl group, --NHSO.sub.2 --R.sup.8 where R.sup.8 has the same meaning as defined above, hydroxy group, OK, a lower alkoxy group which may have a substituent, a lower alkenyloxy group, a lower alkynyloxy group, a cycloalkoxy group which may have a substituent, a phenoxy group, a benzyloxy group, a lower alkylthio group, a phenylthio group or an alkylsulfonylamino group when Z is --CH.dbd. group; R.sup.5 represents a lower alkoxy group; R.sup.6 represents a lower alkoxy group or a lower alkyl group; X represents oxygen atom or sulfur atom; and Z represents nitrogen atom or --CH.dbd. group.processes for preparing the same and a herbicide containing the same as an active ingredient(s).

    摘要翻译: 公开了由下式(I)表示的嘧啶或三嗪化合物:其中R 1表示氰基,卤素原子,羟基或-O-R 7,其中R 7表示低级烷基,低级烯基 基,低级炔基,卤代低级烷基或氰基 - 低级烷基; R2表示氢原子或低级烷基; R3表示氢原子或低级烷基; R 4表示当Z为氮原子时,可以具有取代基,羟基,低级烷氧基或苄氧基的低级烷基或苯基,-NHSO 2 -R 8, 或1-咪唑基,-NHSO 2 -R 8,其中R8具有与上述相同的含义,羟基,OK,可具有取代基的低级烷氧基,低级链烯氧基,低级炔氧基,环烷氧基 当Z为-CH =基团时,可具有取代基,苯氧基,苄氧基,低级烷硫基,苯硫基或烷基磺酰基氨基; R5代表低级烷氧基; R6代表低级烷氧基或低级烷基; X表示氧原子或硫原子; Z表示氮原子或-CH =基团。 其制备方法和含有其作为活性成分的除草剂。

    Sulfonamide derivative, process for preparing the same and herbicide
using the same
    3.
    发明授权
    Sulfonamide derivative, process for preparing the same and herbicide using the same 失效
    磺酰胺衍生物,其制备方法和使用其的除草剂

    公开(公告)号:US5376620A

    公开(公告)日:1994-12-27

    申请号:US41998

    申请日:1993-04-02

    摘要: Disclosed are a sulfonamide compound represented by the following formula (I): ##STR1## wherein Y represents a lower akyl group, a lower alkenyl group, a lower alkynyl group, a halo-lower alkyl group, a cyano-lower alkyl group or --C(CH.sub.3).sub.2 (OR.sup.1) where R.sup.1 represents a lower akyl group, a lower alkenyl group, a lower alkynyl group, a halo-lower alkyl group or a cyano-lower alkyl group; Q represents a substituted or unsubstituted pyridyl group or --NR.sup.2 R.sup.3 where R.sup.2 represents a hydrogen atom, a lower alkyl group, a lower alkoxy group; and R.sup.3 represents a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a phenyl group or a benzyl group; or R.sup.2 and R.sup.3 may be combined to form a cycloamino group; X represents an oxygen atom or a sulfur atom; and Z represents a nitrogen atom or --CH.dbd. group;processes for preparing the same and a herbicide containing the same as an active ingredient(s).

    摘要翻译: 公开了由下式(I)表示的磺酰胺化合物:其中Y表示低级烷基,低级烯基,低级炔基,卤代低级烷基,氰基 - 低级烷基 基团或-C(CH 3)2(OR 1),其中R 1表示低级烷基,低级烯基,低级炔基,卤代低级烷基或氰基 - 低级烷基; Q表示取代或未取代的吡啶基或-NR2R3,其中R2表示氢原子,低级烷基,低级烷氧基; R3表示低级烷基,低级烯基,低级炔基,苯基或苄基。 或者R 2和R 3可以组合形成环氨基; X表示氧原子或硫原子; Z表示氮原子或-CH =基团; 其制备方法和含有其作为活性成分的除草剂。

    Pyrimidine derivatives and a pharmaceutical composition containing them
    6.
    发明授权
    Pyrimidine derivatives and a pharmaceutical composition containing them 失效
    嘧啶衍生物和含有它们的药物组合物

    公开(公告)号:US4450162A

    公开(公告)日:1984-05-22

    申请号:US384416

    申请日:1982-06-02

    CPC分类号: C07D239/42 C07D239/70

    摘要: New 4-anilinopyrimidine derivatives of formula (I): ##STR1## (wherein: R.sup.1 and R.sup.2 are the same or different and each represents a C.sub.1 -C.sub.6 alkyl group or R.sup.1 and R.sup.2 together represent a C.sub.3 -C.sub.5 alkylene group;R.sup.3 represents a hydrogen atom or a C.sub.1 -C.sub.6 alkyl group;n is 0, 1 or 2; andR.sup.4 represents a C.sub.1 -C.sub.6 alkyl group, a C.sub.1 -C.sub.6 alkoxy group, a C.sub.1 -C.sub.6 haloalkyl group, a halogen atom, a nitro group, a C.sub.1 -C.sub.6 alkanesulphonyl group, a cyano group, a carboxy group or a C.sub.2 -C.sub.7 alkoxycarbonyl group and, when n is 2, the two groups represented by R.sup.4 may be the same or different or they may together represent a methylenedioxy group)and pharmaceutically acceptable acid addition salts thereof have been found to have strong antidepressant activity, with low toxicity and very few side-effects. The compounds may be formulated in conventional pharmaceutical compositions for administration by various routes and may be prepared by reacting a 4-halopyrimidine with aniline or an aniline derivative.

    摘要翻译: 式(I)的新的4-苯胺基嘧啶衍生物:其中:R 1和R 2相同或不同,各自表示C 1 -C 6烷基或R 1和R 2一起代表C 3 -C 5亚烷基; R3表示氢原子或C1-C6烷基; n为0,1或2; R4表示C1-C6烷基,C1-C6烷氧基,C1-C6卤代烷基,卤素原子, 硝基,C1-C6烷磺酰基,氰基,羧基或C2-C7烷氧基羰基,当n为2时,由R4表示的两个基团可以相同或不同,或者它们可以一起代表亚甲二氧基 组)及其药学上可接受的酸加成盐被发现具有强的抗抑郁活性,毒性低,副作用非常少。 化合物可以配制成用于通过各种途径给药的常规药物组合物,并且可以通过4-卤代嘧啶与苯胺或苯胺衍生物反应来制备。

    Image forming apparatus and image forming method used in the same
    8.
    发明授权
    Image forming apparatus and image forming method used in the same 失效
    图像形成装置及其形成方法

    公开(公告)号:US5953134A

    公开(公告)日:1999-09-14

    申请号:US731778

    申请日:1996-10-18

    摘要: An image forming method for use in image forming apparatus including on the right surface thereof a discharge opening connectable with a post-processing device, the image forming method comprising the steps of:a first step of delivering one or more documents to a read position sequentially starting from the first document to read the documents at the read position, and outputting the documents in the form of images of the same posture as document images to be read on the documents;a second step of reading a document at a position where the same is placed and outputting the document in the form of an image of the same posture of a document image to be read on the document;a third step of forming, on the upper surface of a sheet to be supplied from the left surface side of the image forming apparatus, the images output in the first or second step in the order that they are read, and delivering the formed images in a direction of the right surface of the image forming apparatus; anda fourth step of reversing the sheet in such a manner that the upper surface of the sheet on which the images are formed in the third step is turned over to the lower surface of the sheet, and discharging the reversed sheet to the discharge opening.

    摘要翻译: 一种用于图像形成装置的图像形成方法,在其右表面上包括可与后处理装置连接的排出口,所述图像形成方法包括以下步骤:顺序地将一个或多个文档递送到读取位置的第一步骤 从第一文档开始,在读取位置读取文档,并且以文档的相同姿势的图像的形式输出要读取的文档的文档; 在放置相同位置的文档的位置读取文档的第二步骤,并以要读取的文档图像的相同姿态的图像的形式输出文档; 第三步骤,在从图像形成装置的左表面侧供给的片材的上表面上,以第一或第二步骤中输出的图像,以读取顺序形成,并将形成的图像输送到 图像形成装置的右表面的方向; 以及第四步骤,使得片材的第三步骤中形成图像的片材的上表面被翻转到片材的下表面,并将反转的片材排出到排出口。