公开(公告)号：US06521627B1

公开(公告)日：2003-02-18

申请号：US09673494

申请日：2000-10-16

申请人： Katsutoshi Fujii ,  Yoshinori Yamanaka ,  Kiyoshi Tsutsumiuchi ,  Youichi Yoshida

发明人： Katsutoshi Fujii ,  Yoshinori Yamanaka ,  Kiyoshi Tsutsumiuchi ,  Youichi Yoshida

IPC分类号： C07D23942

CPC分类号： C07D239/42 ,  A01N43/54 ,  C07D239/30

摘要： The present invention is to provide a novel 5-iodo-4-phenethylaminopyrimidine derivative represented by the following formula (1): wherein R1 represents a halogen atom, a C2-4 acyloxy group or a hydroxyl group; R2 represents a hydrogen atom, a halogen atom, a C1-4 alkyl group, a C1-4 haloalkyl group, a C1-4 alkoxy group or a C1-4 haloalkoxy group; n is an integer of 1 to 3; and * represents an asymmetric carbon atom, useful as pesticides, a synthetic intermediate thereof and processes for producing these compounds, and pesticides containing the 5-iodo-4-phenethylaminopyrimidine derivative(s).

摘要翻译： 本发明提供由下式（1）表示的新的5-碘-4-苯乙基氨基嘧啶衍生物：其中R1表示卤素原子，C2-4酰氧基或羟基; R 2表示氢原子，卤素原子，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基; n为1〜3的整数。 和*表示可用作农药的不对称碳原子，其合成中间体及其制备方法，以及含有5-碘-4-苯乙基氨基嘧啶衍生物的农药。

公开(公告)号：US5221685A

公开(公告)日：1993-06-22

申请号：US828110

申请日：1992-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

IPC分类号： C07D277/46 ,  C07D277/48 ,  C07D417/12

CPC分类号： C07D417/12 ,  C07D277/46 ,  C07D277/48

摘要： Disclosed are a thiazoline compound represented by the following formula (I): ##STR1## wherein R represents hydrogen atom or a lower alkyl group, X represents oxygen atom or sulfur atom, and Q represents Ar (where Ar represents a substituted or unsubstituted phenyl group or a substituted or unsubstituted naphthyl group) or ##STR2## (where Y represents a halogen atom, a lower alkyl group, a lower alkoxy group, a lower haloalkyl group, a lower haloalkoxy group, nitro group, acetyl group or cyano group and n represents an integer of 0 to 5),a process for preparing the same and a chemical for controlling noxious organisms containing the same as an active ingredient.

公开(公告)号：US5498612A

公开(公告)日：1996-03-12

申请号：US380717

申请日：1995-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

IPC分类号： A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D239/42 ,  C07D401/12 ,  C07D405/12 ,  C07F7/18 ,  C07D239/30

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D401/12 ,  C07D405/12 ,  C07F7/1856

摘要： Disclosed are a 4-phenethylaminopyrimidine compound represented by the formula (I): ##STR1## wherein R.sup.1 represents halogen, hydroxyl, acyloxy, alkoxy, haloalkoxy, alkylthio, benzyloxycarbonyloxy, alkyloxycarbonyloxy, alkylsulfonyloxy, tri(alkyl)silyloxy or alkyloxycarbonylalkyloxy;R.sup.2 represents hydrogen, alkyl, alkoxy, halogen, haloalkyl, haloalkoxy, unsubstituted or substituted benzoyl, hydroxyl, haloalkylcarbonyl, alkylsulfonyloxy, haloalkylsulfonyloxy, alkylsulfonyl, alkylsulfinyl, haloalkylsulfinyl, tri(alkyl)silylalkoxy, alkylthio, unsubstituted or substituted pyridyloxy, unsubstituted or substituted phenoxy, alkenyloxy, haloalkenyloxy, unsubstituted or substituted benzyl, 2-phenyl-2-1,3-dioxolanyl, alkoxyiminobenzyl, nitro, haloalkylthio or alkynyloxy; n is an integer of 1 to 5 and * represents an asymmetric carbon atom.a process for preparing the same and an agricultural and horticultural chemical for controlling noxious organisms which contains the same as an active ingredient.

摘要翻译： 公开了由式（I）表示的4-苯乙基氨基嘧啶化合物：其中R 1表示卤素，羟基，酰氧基，烷氧基，卤代烷氧基，烷硫基，苄氧羰基氧基，烷氧基羰氧基，烷基磺酰氧基，三（烷基）甲硅烷氧基或烷氧基羰基烷氧基。 R 2表示氢，烷基，烷氧基，卤素，卤代烷基，卤代烷氧基，未取代或取代的苯甲酰基，羟基，卤代烷基羰基，烷基磺酰氧基，卤代烷基磺酰氧基，烷基磺酰基，烷基亚磺酰基，卤代烷基亚磺酰基，三（烷基）甲硅烷基烷氧基，烷硫基，未取代或取代的吡啶氧基，未取代或取代的苯氧基 ，烯氧基，卤代烯氧基，未取代或取代的苄基，2-苯基-2,3-二氧戊环，烷氧基亚氨基苄基，硝基，卤代烷硫基或炔氧基; n为1〜5的整数，*表示不对称碳原子。 其制备方法以及用于控制含有与活性成分相同的有害生物的农业和园艺化学品。

公开(公告)号：US5369116A

公开(公告)日：1994-11-29

申请号：US85060

申请日：1993-07-02

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyashi Tsutsumiuchi ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyashi Tsutsumiuchi ,  Yoshinori Yamanaka

IPC分类号： A01N43/78 ,  C07D277/20 ,  C07D277/42 ,  C07D277/44 ,  C07D417/12

CPC分类号： C07D417/12 ,  A01N43/78 ,  C07D277/42

摘要： Disclosed are a polyfluorinated thiazoline compound represented by the following formula (I): ##STR1## wherein Q represents a phenyl group; a phenyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; a pyridyl group; or a pyridyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; andR represents a hydrogen atom, a lower alkyl group or an acetyl group,and a chemical for controlling noxious organisms containing the same as an active ingredient.

摘要翻译： 公开了由下式（I）表示的多氟化噻唑啉化合物：其中Q表示苯基; 由卤素原子，卤代低级烷基，硝基，氰基，甲酰基，低级烷氧基羰基或苯甲酰基取代的苯基; 吡啶基; 或被卤素原子，卤代低级烷基，硝基，氰基，甲酰基，低级烷氧基羰基或苯甲酰基取代的吡啶基; R表示氢原子，低级烷基或乙酰基，以及用于控制含有活性成分的有害生物的化学物质。

公开(公告)号：US06881863B2

公开(公告)日：2005-04-19

申请号：US10468880

申请日：2002-02-21

申请人： Katsumasa Harada ,  Yasuhisa Fukuda ,  Yoshinori Yamanaka

发明人： Katsumasa Harada ,  Yasuhisa Fukuda ,  Yoshinori Yamanaka

IPC分类号： C07C249/12 ,  C07C251/44 ,  C07B61/00

CPC分类号： C07C249/12 ,  C07C2601/20 ,  C07C251/44

摘要： The present invention relates to a process for preparing 2-halogenocycloalkanone oxime which comprises subjecting a 2-halogenocycloalkenone oxime compound to reduction with hydrogen in the presence of a platinum-carried catalyst.

摘要翻译： 本发明涉及一种2-卤代环烷酮肟的制备方法，该方法包括在铂载体催化剂存在下，用氢气还原2-卤代环烯酮肟化合物。

公开(公告)号：US06689895B2

公开(公告)日：2004-02-10

申请号：US10363415

申请日：2003-03-03

申请人： Katsumasa Harada ,  Yasuhisa Fukuda ,  Yoshinori Yamanaka ,  Tadashi Murakami ,  Kenji Hirotsu

发明人： Katsumasa Harada ,  Yasuhisa Fukuda ,  Yoshinori Yamanaka ,  Tadashi Murakami ,  Kenji Hirotsu

IPC分类号： C07C25509

CPC分类号： C07C255/09

摘要： The present invention relates to a novel compound 4,8-dodecadienedinitrile represented by the following formula (1): wherein means a cis or trans bond, and a process for preparing 4,8-dodecadienedinitrile which comprises reacting a 2-alkoxy-5,9-cyclododecadienone oxime or a 2-halogeno-5,9-cyclododecadienone oxime with formic acid and hydroxylamine.

摘要翻译： 本发明涉及由下式（1）表示的新化合物4,8-十二烷二腈：其中为顺式或反式键，以及制备4,8-十二二氰基腈的方法，其包括使2-烷氧基-5,9 - 环十二碳二烯酮肟或2-卤代-5,9-环十二碳二烯肟与甲酸和羟胺。