公开(公告)号：US5369116A

公开(公告)日：1994-11-29

申请号：US85060

申请日：1993-07-02

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyashi Tsutsumiuchi ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyashi Tsutsumiuchi ,  Yoshinori Yamanaka

IPC分类号： A01N43/78 ,  C07D277/20 ,  C07D277/42 ,  C07D277/44 ,  C07D417/12

CPC分类号： C07D417/12 ,  A01N43/78 ,  C07D277/42

摘要： Disclosed are a polyfluorinated thiazoline compound represented by the following formula (I): ##STR1## wherein Q represents a phenyl group; a phenyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; a pyridyl group; or a pyridyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; andR represents a hydrogen atom, a lower alkyl group or an acetyl group,and a chemical for controlling noxious organisms containing the same as an active ingredient.

摘要翻译： 公开了由下式（I）表示的多氟化噻唑啉化合物：其中Q表示苯基; 由卤素原子，卤代低级烷基，硝基，氰基，甲酰基，低级烷氧基羰基或苯甲酰基取代的苯基; 吡啶基; 或被卤素原子，卤代低级烷基，硝基，氰基，甲酰基，低级烷氧基羰基或苯甲酰基取代的吡啶基; R表示氢原子，低级烷基或乙酰基，以及用于控制含有活性成分的有害生物的化学物质。

公开(公告)号：US5221685A

公开(公告)日：1993-06-22

申请号：US828110

申请日：1992-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi ,  Yoshinori Yamanaka

IPC分类号： C07D277/46 ,  C07D277/48 ,  C07D417/12

CPC分类号： C07D417/12 ,  C07D277/46 ,  C07D277/48

摘要： Disclosed are a thiazoline compound represented by the following formula (I): ##STR1## wherein R represents hydrogen atom or a lower alkyl group, X represents oxygen atom or sulfur atom, and Q represents Ar (where Ar represents a substituted or unsubstituted phenyl group or a substituted or unsubstituted naphthyl group) or ##STR2## (where Y represents a halogen atom, a lower alkyl group, a lower alkoxy group, a lower haloalkyl group, a lower haloalkoxy group, nitro group, acetyl group or cyano group and n represents an integer of 0 to 5),a process for preparing the same and a chemical for controlling noxious organisms containing the same as an active ingredient.

公开(公告)号：US5081144A

公开(公告)日：1992-01-14

申请号：US503684

申请日：1990-04-02

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Yasuhisa Fukuda ,  Kiyoshi Tsutsumiuchi

IPC分类号： C07D231/22

CPC分类号： C07D231/22

摘要： A compound represented by the formula: ##STR1## wherein R.sub.1 represents hydrogen atom, a halogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.2 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.3 represents an alkyl group having 1 to 8 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or an aralkyl group which may be also substituted; R.sub.4 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; n represents an integer of 4 and when R.sub.2 is an alkyl group, n represents an integer of 1 to 3; A represents an alkylene group having 1 to 5 carbon atoms; and X represents an oxygen atom or a sulfur atom and an insecticide, acaricide or fungicide comprising a compound of the formula (I) as the active ingredient.

公开(公告)号：US5498612A

公开(公告)日：1996-03-12

申请号：US380717

申请日：1995-01-30

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Yoshinori Yamanaka

IPC分类号： A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D239/42 ,  C07D401/12 ,  C07D405/12 ,  C07F7/18 ,  C07D239/30

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N47/06 ,  A01N55/00 ,  C07D401/12 ,  C07D405/12 ,  C07F7/1856

摘要： Disclosed are a 4-phenethylaminopyrimidine compound represented by the formula (I): ##STR1## wherein R.sup.1 represents halogen, hydroxyl, acyloxy, alkoxy, haloalkoxy, alkylthio, benzyloxycarbonyloxy, alkyloxycarbonyloxy, alkylsulfonyloxy, tri(alkyl)silyloxy or alkyloxycarbonylalkyloxy;R.sup.2 represents hydrogen, alkyl, alkoxy, halogen, haloalkyl, haloalkoxy, unsubstituted or substituted benzoyl, hydroxyl, haloalkylcarbonyl, alkylsulfonyloxy, haloalkylsulfonyloxy, alkylsulfonyl, alkylsulfinyl, haloalkylsulfinyl, tri(alkyl)silylalkoxy, alkylthio, unsubstituted or substituted pyridyloxy, unsubstituted or substituted phenoxy, alkenyloxy, haloalkenyloxy, unsubstituted or substituted benzyl, 2-phenyl-2-1,3-dioxolanyl, alkoxyiminobenzyl, nitro, haloalkylthio or alkynyloxy; n is an integer of 1 to 5 and * represents an asymmetric carbon atom.a process for preparing the same and an agricultural and horticultural chemical for controlling noxious organisms which contains the same as an active ingredient.

摘要翻译： 公开了由式（I）表示的4-苯乙基氨基嘧啶化合物：其中R 1表示卤素，羟基，酰氧基，烷氧基，卤代烷氧基，烷硫基，苄氧羰基氧基，烷氧基羰氧基，烷基磺酰氧基，三（烷基）甲硅烷氧基或烷氧基羰基烷氧基。 R 2表示氢，烷基，烷氧基，卤素，卤代烷基，卤代烷氧基，未取代或取代的苯甲酰基，羟基，卤代烷基羰基，烷基磺酰氧基，卤代烷基磺酰氧基，烷基磺酰基，烷基亚磺酰基，卤代烷基亚磺酰基，三（烷基）甲硅烷基烷氧基，烷硫基，未取代或取代的吡啶氧基，未取代或取代的苯氧基 ，烯氧基，卤代烯氧基，未取代或取代的苄基，2-苯基-2,3-二氧戊环，烷氧基亚氨基苄基，硝基，卤代烷硫基或炔氧基; n为1〜5的整数，*表示不对称碳原子。 其制备方法以及用于控制含有与活性成分相同的有害生物的农业和园艺化学品。

公开(公告)号：US5124333A

公开(公告)日：1992-06-23

申请号：US558798

申请日：1990-07-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Isamu Narita ,  Shoji Shikita

IPC分类号： A01N43/54 ,  A01N43/90 ,  A01N47/38 ,  C07D239/42 ,  C07D239/70 ,  C07D239/94 ,  C07D403/12 ,  C07D491/048 ,  C07D495/04

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/90 ,  A01N47/38 ,  C07D239/70 ,  C07D239/94 ,  C07D403/12 ,  C07D495/04

摘要： An aminopyrimidine compound of the formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, an alkyl group, a cycloalkyl group or a halogen atom;R.sup.2 and R.sup.3 each represent an alkyl group or a halogen atom, or R.sup.2 and R.sup.3 represent a saturated or unsaturated 5- or 6-membered ring;R.sup.4 represents a hydrogen atom or --CONR.sup.6 R.sup.7, where R.sup.6 and R.sup.7 represent an unsaturated 5-membered ring; andR.sup.5 represents ##STR2## where m represents an integer of 1 to 10; m' represents an integer of 1 to 15;n represents an integer of 0, 1 or 2;R.sup.8 represents a hydrogen atom, an alkyl group or a cycloalkyl group;R.sup.9 represents an alkyl group, an alkenyl group, an alkynyl group, a substituted or unsubstituted phenyl group, a substituted or unsubstituted aralkyl group or an alkyl group,and acid addition salts thereof. Such compound is useful for combatting insects, acarids, nematodes and fungus.

公开(公告)号：US4895849A

公开(公告)日：1990-01-23

申请号：US105403

申请日：1987-10-05

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

IPC分类号： A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/42 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/08

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/0812

摘要： There are disclosed a compound represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom or a lower alkyl group; R.sub.2 and R.sub.3 each independently represent a halogen atom or a lower alkyl group; R.sub.4 represents a hydrogen atom, a halogen atom or a lower alkyl group; n represents an integer of 1 or 2; Q represents a phenyl group or a heterocyclic group; a substituted or unsubstituted alkyl group; an allyl group; a geranyl group; a farnesyl group; a cycloalkylmethyl group; a substituted ethyl group; a glycidyl group; an acetonyl group; a substituted dioxoranyl group; a 2,2-diethoxyethyl group, a 1-ethoxycarbonylethyl group, a trimethylsilylmethyl group or a 1-pyridylethyl group; A represents a lower alkylene group; and B represents a direct bond, an oxygen atom, a sulfur atom, a straight or branched lower alkylene group or a lower alkyleneoxy group;or an acid addition salt thereof, a process for producing the same, and an insecticide, an acaricide and a fungicide containing the derivative as the active ingredient.

摘要翻译： 公开了下式表示的化合物：其中R 1表示氢原子或低级烷基; R2和R3各自独立地表示卤素原子或低级烷基; R4表示氢原子，卤素原子或低级烷基; n表示1或2的整数; Q表示苯基或杂环基; 取代或未取代的烷基; 烯丙基; 香叶基 法呢基 环烷基甲基; 取代的乙基; 缩水甘油基; 丙酮基; 取代的二氧杂环戊烷基; 2,2-二乙氧基乙基，1-乙氧基羰基乙基，三甲基甲硅烷基甲基或1-吡啶基乙基; A表示低级亚烷基; B表示直接键，氧原子，硫原子，直链或支链低级亚烷基或低级亚烷基氧基; 或其酸加成盐，其制备方法，以及含有该衍生物作为活性成分的杀虫剂，杀螨剂和杀真菌剂。

公开(公告)号：US5252596A

公开(公告)日：1993-10-12

申请号：US903940

申请日：1992-06-26

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Akira Ooka ,  Shoji Shikita

IPC分类号： A01N43/56 ,  C07D231/54 ,  A61K43/56

CPC分类号： C07D231/54

摘要： Disclosed are a novel phenoxyalkylamine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a lower alkyl group or a lower haloalkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom, a lower alkyl group or a halogen atom; R.sup.4 represents a lower alkenyl group or --S--O--R.sup.6 where A represents a lower alkylene group and R.sup.6 represents a lower alkyl group, a lower alkenyl group or a lower alkynyl group; R.sup.5 represents hydrogen atom, a lower alkyl group or a halogen atom,a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

公开(公告)号：US5039692A

公开(公告)日：1991-08-13

申请号：US539965

申请日：1990-06-15

申请人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

发明人： Tokio Obata ,  Katsutoshi Fujii ,  Toshinobu Tanaka ,  Akira Ooka ,  Shoji Shikita

IPC分类号： C07D233/64 ,  A01N43/56 ,  C07D231/14 ,  C07D231/16 ,  C07D233/68

CPC分类号： C07D231/16 ,  C07D231/14

摘要： There are disclosed a phenoxyalkylamine derivative represented by the formula: ##STR1## wherein A.sup.1 represents an alkylene group having 2 to 5 carbon atoms, R.sup.1 and R.sup.2 each represent hydrogen atom or a lower alkyl group having 1 to 5 carbon atoms, R.sup.3, R.sup.4 and R.sup.5 each represent hydrogen atom, an alkyl group having 1 to 5 carbon atoms or a halogen atom, R.sup.6 represents hydrogen atom, an alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms or a group --A.sup.2 --X--R.sup.7, A.sup.2 represents an alkylene group having 1 to 5 carbon atoms, X represents oxygen atom or sulfur atom, R.sup.7 represents a lower alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a substituted or unsubstituted aralkyl group,and an insecticide, an acaricide and a fungicide for agriculture and horticulture, which comprises a carrier and the above phenoxyalkylamine derivative represented as the active ingredient.

公开(公告)号：US4985426A

公开(公告)日：1991-01-15

申请号：US435937

申请日：1989-11-13

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Kiyoshi Tsutsumiuchi ,  Haruo Yoshiya

IPC分类号： A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/42 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/08

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/58 ,  A01N43/66 ,  A01N43/78 ,  A01N49/00 ,  A01N55/00 ,  C07D239/56 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07F7/0812

摘要： There is disclosed a compound represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom or a lower alkyl group; R.sub.2 and R.sub.3 each independently represent a halogen atom or a lower alkyl group; R.sub.4 represents a hydrogen atom, a halogen atom or a lower alkyl group; n represents an integer of 1 or 2; Q represents a phenyl group or a heterocyclic group; a substituted or unsubstituted alkyl group; an allyl group, a geranyl group; a farnesyl group; a cycloalkylmethyl group; a substituted ethyl group; a glycidyl group; an acetonyl group; a substituted dioxoranyl group; a 2,2-diethoxyethyl group, a 1-ethoxycarbonylethyl group, a trimethylsilylmethyl group or a 1-pyridylethyl group; A represents a lower alkylene group; and B represents a direct bond, an oxygen atom, a sulfur atom, a straight or branched lower alkylene group or a lower alkyleneoxy group;or an acid addition salt thereof, a process for producing the same, and an insecticide, an acaricide and a fungicide containing the derivative as the active ingredient.

公开(公告)号：US4931455A

公开(公告)日：1990-06-05

申请号：US289626

申请日：1988-12-22

申请人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Haruo Yoshiya ,  Kiyoshi Tsutsumiuchi ,  Shoji Shikita

发明人： Hirosuke Yoshioka ,  Tokio Obata ,  Katsutoshi Fujii ,  Haruo Yoshiya ,  Kiyoshi Tsutsumiuchi ,  Shoji Shikita

IPC分类号： A01N43/54 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  A01N47/20 ,  A01N47/28 ,  A01N49/00 ,  A01N53/00 ,  C07D239/42 ,  C07D403/12 ,  C07D405/12 ,  C07D413/12

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  A01N47/20 ,  A01N47/28 ,  A01N49/00 ,  A01N53/00 ,  C07D403/12 ,  C07D405/12 ,  C07D413/12

摘要： There are described an alkylaminopyrimidine derivative represented by the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom, a halogen atom, a lower alkyl group, a cycloalkyl group having 3 to 6 carbon atoms, a halogenated lower alkyl group or a substituted or unsubstituted phenyl group; R.sub.2 represents a halogen atom; R.sub.3 represents a hydrogen atom, a lower alkyl group or a cycloalkyl group having 3 to 6 carbon atoms; and R.sub.4 represents a straight or branched alkyl group having 1 to 20 carbon atoms which may have substituents,or an acid addition salt thereof, a process for preparing the same and an insecticide, an acaricide or a fungicide containing the compound as an active ingredient.