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1.发明申请NOVEL AZACYCLYL-SUBSTITUTED ARYLDIHYDROISOQUINOLINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS 有权新乙酰胆碱取代的芳基二氢喹啉酮，其制备方法及其作为药物使用公开(公告)号：US20090264403A1
公开(公告)日：2009-10-22
申请号：US12191662
申请日：2008-08-14
申请人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
发明人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
IPC分类号： A61K31/4725 , C07D401/10 , C07D405/14 , A61K31/55
CPC分类号： A61K31/4725 , A61K31/496 , A61K31/5377 , A61K31/541 , A61K31/551 , C07D401/10 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/14 , C07D417/14 , C07D471/04 , C07D487/04 , C07D487/10 , C07D491/04 , C07D495/04 , C07D513/04
摘要： The invention relates to azacyclyl-substituted aryldihydroisoquinolinones and their derivatives, and their physiologically tolerated salts and physiologically functional derivatives, their preparation, medicaments comprising at least one azacyclyl-substituted aryldihydroisoquinolinone of the invention or its derivative, and the use of the azacyclyl-substituted aryidihydroisoquinolinones of the invention and their derivatives as MCH antagonists.
摘要翻译： 本发明涉及氮杂环酰基取代的芳基二氢异喹啉酮及其衍生物及其生理上耐受的盐和生理功能衍生物，其制备方法，包含至少一种本发明的氮杂环酰基取代的芳基二氢异喹啉酮或其衍生物的药物，以及使用偶氮基酰基取代的芳酰基异喹啉酮 的本发明及其衍生物作为MCH拮抗剂。
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2.发明申请NOVEL AMINOALCOHOL-SUBSTITUTED ARYLDIHYDROISOQUINOLINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS 有权新型氨基醇取代的芳基二氢喹啉酮，其制备方法及其作为药物使用公开(公告)号：US20090082391A1
公开(公告)日：2009-03-26
申请号：US12191697
申请日：2008-08-14
申请人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
发明人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
IPC分类号： A61K31/4365 , C07D495/04
CPC分类号： C07D471/04 , C07D217/24 , C07D401/12 , C07D451/06 , C07D453/02 , C07D455/06
摘要： The invention relates to aminoalcohol-substituted aryldihydroisoquinolinones and their derivatives, and their physiologically tolerated salts and physiologically functional derivatives, their preparation, medicaments comprising at least one aminoalcohol-substituted aryldihydroisoquinolinone of the invention or its derivative, and the use of the aminoalcohol-substituted aryldihydroisoquinolinones of the invention and their derivatives as MCH antagonists.
摘要翻译： 本发明涉及氨基醇取代的芳基二氢异喹啉酮及其衍生物及其生理上耐受的盐和生理功能衍生物，其制备方法，包含至少一种本发明的氨基醇取代的芳基二氢异喹啉酮或其衍生物的药物，以及氨基醇取代的芳基二氢异喹啉酮的用途 的本发明及其衍生物作为MCH拮抗剂。
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3.发明申请NOVEL AZACYCLYL-SUBSTITUTED ARYLTHIENOPYRIMIDINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS 有权新乙酰胆碱取代的芳香族二亚胺，其制备方法及其作为药物使用公开(公告)号：US20090082339A1
公开(公告)日：2009-03-26
申请号：US12191630
申请日：2008-08-14
申请人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
发明人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
IPC分类号： A61K31/551 , C07D495/04 , C07D243/08 , A61K31/517 , C07D239/91 , A61K31/519
CPC分类号： C07D491/04 , C07D239/91 , C07D403/10 , C07D495/04 , C12N9/99
摘要： The invention relates to azacyclyl-substituted arylthienopyrimidinones and their derivatives, and their physiologically tolerated salts and physiologically functional derivatives, their preparation, medicaments comprising at least one azacyclyl-substituted arylthienopyrimidinone of the invention or its derivative, and the use of the azacyclyl-substituted arylthienopyrimidinones of the invention and their derivatives as MCH antagonists.
摘要翻译： 本发明涉及氮杂环酰基取代的芳基噻吩并嘧啶酮及其衍生物及其生理上耐受的盐和生理功能衍生物，其制备方法，包含至少一种本发明的氮杂环酰基取代的芳基噻吩并嘧啶酮或其衍生物的药物，以及使用偶氮酰基取代的芳基噻吩并嘧啶酮 的本发明及其衍生物作为MCH拮抗剂。
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4.发明申请NOVEL AMINO ALCOHOL-SUBSTITUTED ARYLTHIENOPYRIMIDINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS 有权新型氨基醇取代的芳香族二亚胺，其制备方法及其作为药物使用公开(公告)号：US20090076002A1
公开(公告)日：2009-03-19
申请号：US12191678
申请日：2008-08-14
申请人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
发明人： Lothar SCHWINK , Siegfried STENGELIN , Matthias GOSSEL , Gerhard HESSLER , Torsten HAACK , Petra LENNIG
IPC分类号： A61K31/5377 , C07D495/04 , A61K31/519
CPC分类号： C07D495/04 , C07D519/00
摘要： The invention relates to amino alcohol-substituted arylthienopyrimidinones and their derivatives, and their physiologically tolerated salts and physiologically functional derivatives, their preparation, medicaments comprising at least one amino alcohol-substituted arylthienopyrimidinone of the invention or its derivative, and the use of the amino alcohol-substituted arylthienopyrimidinones of the invention and their derivatives as MCH antagonists.
摘要翻译： 本发明涉及氨基醇取代的芳基噻吩并嘧啶酮及其衍生物及其生理上耐受的盐和生理功能衍生物，其制备方法，包含至少一种本发明的氨基醇取代的芳基噻吩并嘧啶酮或其衍生物的药物，以及氨基醇的用途 - 取代的芳基噻吩并嘧啶酮及其衍生物作为MCH拮抗剂。
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5.发明申请公开(公告)号：US20100249097A1
公开(公告)日：2010-09-30
申请号：US12705140
申请日：2010-02-12
IPC分类号： A61K31/397 , C07D405/12 , A61K31/4025 , A61P3/10 , A61P3/00 , A61K31/4709 , C07D413/12 , A61K31/5377 , C07D417/12 , A61K31/541 , A61K31/55
CPC分类号： C07D405/12 , A61K31/397 , A61K31/4025 , A61K31/4525 , A61K31/4709 , A61K31/496 , A61K31/5377 , A61K31/541 , A61K31/55 , A61K31/553 , A61K45/06 , C07D307/12
摘要： The invention relates to substituted tetrahydronaphthalenes and derivatives thereof, and also to the physiologically compatible salts and physiologically functional derivatives thereof, to preparation thereof, to medicaments comprising at least one inventive substituted tetrahydronaphthalene or derivative thereof, and to the use of the inventive substituted tetrahydronaphthalenes and derivatives thereof as medicaments.
摘要翻译： 本发明涉及取代的四氢萘及其衍生物，以及其生理上相容的盐和生理功能衍生物及其制备方法，涉及包含至少一种本发明取代的四氢化萘或其衍生物的药物，以及本发明取代的四氢萘和 其衍生物作为药物。
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6.发明申请ARYL-SUBSTITUTED POLYCYCLIC AMINES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT 有权芳基取代的多环酰胺，其生产方法及其作为药物的用途公开(公告)号：US20100298378A1
公开(公告)日：2010-11-25
申请号：US12846075
申请日：2010-07-29
IPC分类号： A61K31/4545 , C07D487/08 , A61K31/407 , C07D401/14 , A61K31/454 , C07D498/10 , A61K31/424 , A61K31/4439 , C07D417/14 , A61K31/427 , A61P3/06 , A61P3/10
CPC分类号： C07D471/04 , C07D471/08 , C07D487/04
摘要： The invention relates to aryl-substituted polycyclic amines of formula I, especially bicyclic amines, and to the physiologically tolerated salts and physiologically functional derivatives thereof; where the symbols and radicals are explained in the description, as well as to pharmaceutical compositions containing them and to methods of treatment using them.
摘要翻译： 本发明涉及式I的芳基取代的多环胺，特别是双环胺，以及其生理上耐受的盐和生理功能衍生物; 在说明书中解释符号和自由基以及含有它们的药物组合物以及使用它们的治疗方法。
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7.发明申请ARYL-SUBSTITUTED POLYCYCLIC AMINES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT 有权芳基取代的多环酰胺，其生产方法及其作为药物的用途公开(公告)号：US20090258881A1
公开(公告)日：2009-10-15
申请号：US12489653
申请日：2009-06-23
IPC分类号： A61K31/4985 , C07D455/02 , A61K31/435 , A61P3/04 , A61K31/46 , C07D451/02 , C07D403/12 , A61K31/454 , C07D487/04 , C07D401/14 , C07D401/12 , C07D405/14
CPC分类号： C07D471/04 , C07D471/08 , C07D487/04
摘要： The invention relates to aryl-substituted polycyclic amines of the formula I, especially bicyclic amines, and to the physiologically tolerated salts and physiologically functional derivatives thereof; where the symbols and radicals are explained in the description as well as to pharmaceutical compositions and medical treatments employing these compounds.
摘要翻译： 本发明涉及式I的芳基取代的多环胺，特别是双环胺，以及其生理上耐受的盐和生理功能衍生物; 在说明书中解释符号和基团以及使用这些化合物的药物组合物和医疗处理。
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公开(公告)号：US20090258872A1
公开(公告)日：2009-10-15
申请号：US12489648
申请日：2009-06-23
IPC分类号： A61K31/5377 , A61K31/4375 , A61P3/04 , A61K31/439
CPC分类号： C07D471/04 , C07D471/08 , C07D487/04
摘要： The invention relates to therapeutic use of aryl-substituted polycyclic amines of the formula I, especially bicyclic amines, and to the physiologically tolerated salts and physiologically functional derivatives thereof; where the symbols and radicals are explained in the description.
摘要翻译： 本发明涉及式I的芳基取代的多环胺，特别是双环胺，以及其生理上耐受的盐和生理功能衍生物的治疗用途; 在描述中解释符号和基团。
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9.发明申请ARYL-SUBSTITUTED POLYCYCLIC AMINES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT 有权芳基取代的多环酰胺，其生产方法及其作为药物的用途公开(公告)号：US20070299077A1
公开(公告)日：2007-12-27
申请号：US11674353
申请日：2007-02-13
IPC分类号： A61K31/495 , A61K31/40 , A61K31/404 , A61K31/407 , A61K31/415 , A61K31/496 , A61P3/04 , C07D209/00 , C07D211/00 , C07D295/00 , C07D277/02 , C07D263/02 , C07D241/36 , C07D231/02 , C07D221/00 , C07D213/00 , C07D209/04 , A61P3/10 , A61P3/00 , A61K31/421 , A61K31/426 , A61K31/44 , A61K31/4523
CPC分类号： C07D471/04 , C07D471/08 , C07D487/04
摘要： The invention relates to aryl-substituted polycyclic amines of formula I, especially bicyclic amines, and to the physiologically tolerated salts and physiologically functional derivatives thereof; where the symbols and radicals are explained in the description, as well as to pharmaceutical compositions containing them and to methods of treatment using them.
摘要翻译： 本发明涉及式I的芳基取代的多环胺，特别是双环胺，以及其生理上耐受的盐和生理功能衍生物; 在说明书中解释符号和自由基以及含有它们的药物组合物以及使用它们的治疗方法。
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10.发明申请ARYL-SUBSTITUTED POLYCYCLIC AMINES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT 有权芳基取代的多环酰胺，其生产方法及其作为药物的用途公开(公告)号：US20070197584A1
公开(公告)日：2007-08-23
申请号：US11675646
申请日：2007-02-16
IPC分类号： A61K31/47
CPC分类号： C07D471/04 , C07D471/08 , C07D487/04
摘要： The invention relates to aryl-substituted polycyclic amines of the formula I, especially bicyclic amines, and to the physiologically tolerated salts and physiologically functional derivatives thereof; where the symbols and radicals are explained in the description as well as to pharmaceutical compositions and medical treatments employing these compounds.
摘要翻译： 本发明涉及式I的芳基取代的多环胺，特别是双环胺，以及其生理上耐受的盐和生理功能衍生物; 在说明书中解释符号和基团以及使用这些化合物的药物组合物和医疗处理。
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