Sulphonyltriazol derivatives and their use for combating micro-organisms
    6.
    发明授权
    Sulphonyltriazol derivatives and their use for combating micro-organisms 失效
    磺酰三唑衍生物及其对抗微生物的用途

    公开(公告)号:US06384066B1

    公开(公告)日:2002-05-07

    申请号:US09787650

    申请日:2001-03-20

    IPC分类号: A07N4380

    摘要: Novel sulphonyltriazole derivatives of the formula in which Hal represents fluorine, chlorine or bromine, R1 represents hydrogen, alkyl, alkoxyalkyl, cycloalkyl, alkylaminocarbonyl, optionally substituted phenyl, optionally substituted phenoxy or represents optionally substituted heterocyclyl and R2 represents alkyl or represents optionally substituted heterocyclyl or represents a radical of the formula in which R3 represents halogen, alkyl or phenyl, R4 represents hydrogen or alkyl and R5 represents alkyl or optionally substituted phenyl, or R4 and R5 together with the nitrogen atom to which they are attached form a heterocyclic ring which may be substituted and which may also contain an additional heteroatom, a process for preparing these substances and their use for controlling undesirable microorganisms.

    摘要翻译: 烷基,烷氧基烷基,环烷基,烷基氨基羰基,任选取代的苯基,任选取代的苯氧基或任选取代的杂环基,R 2表示烷基或代表任选取代的杂环基或代表基团 的化合物,其中R 3表示卤素,烷基或苯基,R 4表示氢或烷基,R 5表示烷基或任选取代的苯基,或R 4和R 5与它们所连接的氮原子一起形成可被取代的杂环, 另外的杂原子,这些物质的制备方法及其控制不良微生物的用途。

    2-cyanobenzimidazoles and their use, and new precursors
    10.
    发明授权
    2-cyanobenzimidazoles and their use, and new precursors 失效
    2-氰基苯并咪唑及其用途和新前体

    公开(公告)号:US5510364A

    公开(公告)日:1996-04-23

    申请号:US981035

    申请日:1992-11-24

    CPC分类号: C07D491/04 A01N43/90

    摘要: New 2-cyanobenzimidazoles of the formula (I) ##STR1## in which R.sup.1, R.sup.2 and A have the meaning given in the description, a preparation process, their use in agriculture, for example against fungi, insects etc., and new intermediates.Formula (I) provides a definition of the compounds; for example they are obtained from suitable 2-cyanobenzimidazoles which are unsubstituted in the 1-position with N,N-dimethylsulphamoyl halide. The 2-cyanobenzimidazoles which are unsubstituted in the 1-position are equally new and can be reacted from suitable phenylenediamines of the formula (IV) with methyl 2,2,2-trichloroacetimidate of the formula (V) to give the 2-trichloromethylbenzimidazoles of the formula (VI), which are equally new and from which the compounds of the formula (II) can subsequently be obtained with ammonia.

    摘要翻译: 式(I)的新的2-氰基苯并咪唑其中R1,R2和A具有说明书中给出的含义,制备方法,它们在农业中的用途,例如抗真菌,昆虫等,以及 新中间体 式(I)提供化合物的定义; 例如,它们可由合适的2-氰基苯并咪唑得到,其中N,N-二甲基氨磺酰卤在1位未被取代。 在1-位未被取代的2-氰基苯并咪唑是同等新的,并且可以由适当的式(Ⅳ)亚苯基二胺与式(Ⅴ)的2,2,2-三氯乙酰亚氨酸甲酯反应得到2-(三氟甲基)苯并咪唑 式(VI)同样新,随后可以用氨获得式(II)化合物。