-
公开(公告)号:US5041459A
公开(公告)日:1991-08-20
申请号:US535270
申请日:1990-06-08
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D249/08 , C07D403/06 , C07D405/06 , C07D409/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Microbicidal hydroxy-keto-azoles of the formula ##STR1## in which R.sup.1 represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl or optionally substituted aryl,R.sup.2 represents optionally substituted aryl or a five- or six-membered heterocyclic radical having up to 3 hetero-atoms, which is optionally substituted and optionally fused to benzene, andX represents a nitrogen atom or a CH group,and addition products thereof with acids and metal salts.
摘要翻译: 其中R 1表示任选取代的烷基,任选取代的烯基,任选取代的环烷基或任选取代的芳基,其中R 1表示任选取代的芳基或五元或六元杂环基的式(I)的杀微生物羟基 - 酮 - 具有至多3个杂原子,其任选被取代并任选地与苯稠合,X表示氮原子或CH基团,以及其与酸和金属盐的加成产物。
-
公开(公告)号:US5081140A
公开(公告)日:1992-01-14
申请号:US384595
申请日:1989-07-24
申请人: Manfred Jautelat , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Astrid Mauler , Wilfried Paulus , Monika Frie
发明人: Manfred Jautelat , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Astrid Mauler , Wilfried Paulus , Monika Frie
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D249/08 , C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: New halogenovinyl-azole derivatives of the formula ##STR1## in which R.sup.1 represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl or optionally substituted aryl, or represents optionally substituted heteroaryl,R.sup.2 represents hydrogen, alkyl, alkenyl, acyl or aralkylX.sup.1 represents halogen,X.sup.2 represents halogen,X.sup.3 represents hydrogen or halogenY represents nitrogen or a CH group,and acid addition salts and metal salt complexes thereofare very effective for combating microbes in plant protection and in the preservation of materials.
摘要翻译: 式(I)的新的卤代乙烯基 - 唑衍生物,其中R 1表示任选取代的烷基,任选取代的烯基,任选取代的环烷基或任选取代的芳基,或表示任选取代的杂芳基,R 2表示氢,烷基,烯基,酰基或 芳烷基X1表示卤素,X2表示卤素,X3表示氢或卤素,Y表示氮或CH基,其酸加成盐和金属盐络合物对于防治植物保护和保存材料中的微生物非常有效。
-
公开(公告)号:US5143932A
公开(公告)日:1992-09-01
申请号:US645951
申请日:1991-01-25
申请人: Manfred Jautelat , Klaus Stroech , Gerd Hanssler , Stefan Dutzmann , Karl-Heinz Kuck , Wilhelm Brandes
发明人: Manfred Jautelat , Klaus Stroech , Gerd Hanssler , Stefan Dutzmann , Karl-Heinz Kuck , Wilhelm Brandes
IPC分类号: A01N43/50 , A01N43/653 , B27K3/34 , C07D233/60 , C07D233/64 , C07D249/08 , C07D521/00
CPC分类号: C07D249/08 , A01N43/50 , A01N43/653 , C07D231/12 , C07D233/56
摘要: Microbicidal halogenoallyl-azolyl derivatives of the formula ##STR1## in which R.sup.1 represents a radical of the formula ##STR2## R.sup.2 represents hydrogen, alkyl, alkenyl, acyl or aralkyl, X.sup.1 represents halogen,X.sup.2 represents halogen,X.sup.3 represents hydrogen or halogen andY represents nitrogen or a CH group,and addition products thereof with acids and metal salts.
摘要翻译: 式(I)的杀微生物卤代烯丙基 - 唑基衍生物,其中R 1表示下式的基团:其中R 1表示下式的基团: 烷基,烯基,酰基或芳烷基,X 1表示卤素,X 2表示卤素,X 3表示氢或卤素,Y表示氮或CH基团,并且其与酸和金属盐的加成产物。
-
公开(公告)号:US5122532A
公开(公告)日:1992-06-16
申请号:US645936
申请日:1991-01-25
申请人: Manfred Jautelat , Klaus Stroech , Gerd Hanssler , Stefan Dutzmann , Karl-Heinz Kuck , Wilhelm Brandes
发明人: Manfred Jautelat , Klaus Stroech , Gerd Hanssler , Stefan Dutzmann , Karl-Heinz Kuck , Wilhelm Brandes
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D233/64 , C07D249/08 , C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06 , C07D521/00
CPC分类号: C07D249/08 , A01N43/50 , A01N43/653 , C07D231/12 , C07D233/56
摘要: A microbicidal halogenoallyl-azolyl derivatives of the formula ##STR1## in which R.sup.1 represents halogenoallyl, propargyl, substituted cycloalkyl or optionally substituted heteroaryl, or represents a radical of the formula ##STR2## where R.sup.3 represents hydrogen, halogen, or phenyl which is optionally substituted by halogen, phenoxy which is optionally substituted by halogen or phenoxymethyl which is optionally substituted by halogen,R.sup.4 represents hydrogen or halogen, andR.sup.5 represents iso-propyl, or phenyl which is optionally substituted by halogen or phenoxy which is optionally substituted by halogen or phenoxy which is optionally substituted by halogen,R.sup.2 represents hydrogen, alkyl, alkenyl, acyl or aralkyl,X.sup.1 represents halogen,X.sup.2 represents halogen,X.sup.3 represents hydrogen or halogen andY represents nitrogen or a CH group,and addition products thereof with acids and metal salts.
摘要翻译: 式(I)的杀微生物卤代烯丙基 - 唑基衍生物,其中R 1表示卤代烯丙基,炔丙基,取代的环烷基或任选取代的杂芳基,或表示下式的基团,其中R 3表示氢,卤素或苯基, 任选被卤素取代的苯氧基或任选被卤素取代的苯氧基甲基,R 4代表氢或卤素,R 5代表异丙基,或任选被卤素或苯氧基取代的苯基,任选被卤素或苯氧基任意地被 卤素或苯氧基,其任选被卤素取代,R 2表示氢,烷基,烯基,酰基或芳烷基,X 1表示卤素,X 2表示卤素,X 3表示氢或卤素,Y表示氮或CH基团, 和金属盐。
-
公开(公告)号:US5175169A
公开(公告)日:1992-12-29
申请号:US761087
申请日:1991-09-17
申请人: Manfred Jautelat , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Astrid Mauler , Wilfried Paulus , Monika Frie
发明人: Manfred Jautelat , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Astrid Mauler , Wilfried Paulus , Monika Frie
IPC分类号: A01N43/50 , A01N43/653 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: New halogenovinyl-azole derivatives of the formula ##STR1## in which R.sup.1 represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl or optionally substituted aryl, or represents optionally substituted heteroaryl,R.sup.2 represents hydrogen, alkyl, alkenyl, acyl or aralkylX.sup.1 represents halogen,X.sup.2 represents halogen,X.sup.3 represents hydrogen or halogenY represents nitrogen or a CH group,and acid addition salts and metal salt complexes thereofare very effective for combating microbes in plant protection and in the preservation of materials.
摘要翻译: 式(I)的新的卤代乙烯基 - 唑衍生物,其中R 1表示任选取代的烷基,任选取代的烯基,任选取代的环烷基或任选取代的芳基,或表示任选取代的杂芳基,R 2表示氢,烷基,烯基,酰基或 芳烷基X1表示卤素,X2表示卤素,X3表示氢或卤素,Y表示氮或CH基,其酸加成盐和金属盐络合物对于防治植物保护和保存材料中的微生物非常有效。
-
6.
公开(公告)号:US4917720A
公开(公告)日:1990-04-17
申请号:US256808
申请日:1988-10-12
申请人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
发明人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
IPC分类号: C07C43/225 , A01N43/50 , A01N43/653 , C07C41/00 , C07C45/00 , C07C49/167 , C07C49/175 , C07C67/00 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulfur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.
-
公开(公告)号:US4826865A
公开(公告)日:1989-05-02
申请号:US175467
申请日:1988-03-30
申请人: Gerhard Jager , Manfred Jautelat , Dieter Arlt , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler
发明人: Gerhard Jager , Manfred Jautelat , Dieter Arlt , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler
IPC分类号: A01N43/50 , A01N43/64 , A01N43/653 , C07D233/60 , C07D249/08 , C07D521/00 , C07D233/54
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Novel fungicidally active compounds of the formula ##STR1## in which X is nitrogen or the CH group,Y is hydrogen, bromine or iodine,Z is oxygen, sulphur, the --SO-- group or the --SO.sub.2 -- group, andAr is optionally substituted aryl,or physiologically tolerated addition products thereof with acids or metal salts.
摘要翻译: 新型杀真菌活性化合物,其中X是氮或CH基,Y是氢,溴或碘,Z是氧,硫,-SO-基或-SO 2 - 基,Ar是任选的 取代的芳基或其与酸或金属盐的生理上耐受的加成产物。
-
公开(公告)号:US5254693A
公开(公告)日:1993-10-19
申请号:US788007
申请日:1991-11-05
IPC分类号: A01N43/74 , C07D277/32 , C07D277/34 , C07D277/42 , C07D277/56 , C07D263/38 , C07D263/48
CPC分类号: C07D277/42 , A01N43/74 , C07D277/56
摘要: Fungicidal substituted acrylic esters of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or alkenyl, or represents in each case optionally substituted aralkyl, aralkenyl, aryl or heteroaryl,R.sup.2 represents halogen, cyano, nitro, formyl, halogenoalkyl, alkoxyalkyl or alkylthioalkyl, or represents hydroximinoalkyl, alkoximinoalkyl, N-alkyliminoalkyl, N-aryliminoalkyl or N,N-dialkylhydrazonoalkyl, or represents alkoxy, alkylthio, halogenoalkoxy or halogenoalkylthio, or represents aryloxy or arylthio, or represents alkanoyl, alkoxycarbonyl, N,N-dialkylcarbamoyl or heterocyclylcarbonyl,R.sup.3 represents alkyl, or represents optionally substituted aralkyl,R.sup.4 represents dialkylamino or represents a radical --Z--R.sup.5,X represents oxygen or sulphur andY represents oxygen or sulphur or represents a radical ##STR2## where R.sup.5 represents alkyl or represents optionally substituted aralkyl,R.sup.6 represents hydrogen, alkyl or alkanoyl, or represents in each case optionally substituted aralkyl or aryl, andZ represents oxygen or sulphur.
摘要翻译: 式(I)的杀真菌取代的丙烯酸酯,其中R 1表示氢,烷基或烯基,或在每种情况下表示任选取代的芳烷基,芳烯基,芳基或杂芳基,R 2表示卤素,氰基,硝基,甲酰基,卤代烷基, 烷氧基烷基或烷硫基烷基,或代表肟基烷基,烷肟基烷基,N-烷基亚氨基烷基,N-芳基亚氨基烷基或N,N-二烷基肼基烷基,或代表烷氧基,烷硫基,卤代烷氧基或卤代烷硫基,或代表芳氧基或芳硫基,或代表烷酰基,烷氧羰基,N, 二烷基氨基甲酰基或杂环基羰基,R3代表烷基,或代表任意取代的芳烷基,R4代表二烷基氨基或代表基团-Z-R5,X代表氧或硫,Y代表氧或硫,或代表基团,其中R5代表烷基或代表 任选取代的芳烷基,R 6表示氢,烷基或烷酰基,或在每种情况下表示任选取代的芳烷基 R芳基,Z表示氧或硫。
-
9.
公开(公告)号:US4988729A
公开(公告)日:1991-01-29
申请号:US423607
申请日:1989-10-17
申请人: Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
发明人: Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
IPC分类号: A01N43/08 , A01N43/28 , C07D307/14 , C07D307/22 , C07D317/28 , C07D327/04 , C07D407/12 , C07D417/12
CPC分类号: C07D407/12 , A01N43/08 , A01N43/28 , C07D307/14 , C07D317/28 , C07D327/04
摘要: Combattting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid additon salts thereof. Many of the compounds wherein R.sup.1 has a narrower meaning are new.
摘要翻译: 用下式(Ⅰ)的氨基甲基杂环化合物与R1代表氢,烷基,烯基,各取代四氢萘基,十氢萘基,环烷基或环烯基,以及被环烷基,环烯基,环烷氧基 或环烷硫基,其中环状基团可任选被取代,此外任选取代的芳基,另外被芳基,芳氧基,芳硫基,芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基,其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基,R 3表示烷基,烯基,炔基,烷氧基烷基,羟基烷基,羟基烷氧基烷基,二烷氧基烷基,或在每种情况下任选取代的环烷基,环烷基烷基,芳基,芳烷基,芳烯基,呋喃基烷基,四氢呋喃基烷基,四氢吡喃基烷基,二氧戊环烷基或二烷基烷基,X 代表氧,硫或CH2基,或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。
-
10.
公开(公告)号:US4878939A
公开(公告)日:1989-11-07
申请号:US258108
申请日:1988-10-13
申请人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
发明人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
IPC分类号: C07C43/225 , A01N43/50 , A01N43/653 , C07C41/00 , C07C45/00 , C07C49/167 , C07C49/175 , C07C67/00 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulphur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.
摘要翻译: 其中R 1和R 2各自独立地表示具有多于一个碳原子的烷基,或者R 1表示二氯甲基,三氯甲基,氯乙烯基或二氯乙烯基,并且R 2表示烷基,R 3表示烷基, 酮基或CH(OH)基,Z表示氮原子或CH基,X表示氧或硫,Ar表示任选取代的苯基,或其与酸和金属盐的加成产物对真菌有活性, 植物生长。 还显示了其新的中间体。
-
-
-
-
-
-
-
-
-