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1.FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTS 失效
标题翻译: 功能选择性ALPHA2C ADRENORECEPTOR AGONISTS公开(公告)号:US20100197562A1
公开(公告)日:2010-08-05
申请号:US12525641
申请日:2008-02-11
申请人: Manuel De lera Ruiz , Kevin D. McCormick , Christopher W. Boyce , Robert G. Aslanian , Younong Yu , Pietro Mangiaracina , Junying Zheng , Michael Y. Berlin , Stephanie L. Ciesla , Chia-yu Huang , Bo Liang
发明人: Manuel De lera Ruiz , Kevin D. McCormick , Christopher W. Boyce , Robert G. Aslanian , Younong Yu , Pietro Mangiaracina , Junying Zheng , Michael Y. Berlin , Stephanie L. Ciesla , Chia-yu Huang , Bo Liang
IPC分类号: A61K31/506 , C07D403/14 , A61K31/4178 , C07D401/10 , C07D487/04 , A61K31/519 , C07D401/14 , A61K31/4439 , A61K31/56 , A61K38/02 , A61P11/00 , A61P29/00 , A61P1/12 , A61P9/00 , A61P25/00 , A61P25/24 , A61P25/22 , A61P25/18 , A61P3/10 , A61P19/02
CPC分类号: C07D403/14 , C07D233/10 , C07D401/14 , C07D403/06 , C07D403/10 , C07D405/14 , C07D407/14 , C07D409/14 , C07D413/14
摘要: In its many embodiments, the present invention provides a novel class of biaryl compounds as inhibitors of ÿ2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the ÿ2C adrenergic receptors using such compounds or pharmaceutical compositions.
摘要翻译: 在其许多实施方案中,本发明提供了一类新颖的联芳基化合物作为ÿ2C肾上腺素能受体激动剂的抑制剂,制备此类化合物的方法,含有一种或多种此类化合物的药物组合物,制备包含一种或多种此类化合物的药物制剂的方法, 以及使用这些化合物或药物组合物治疗,预防,抑制或改善与ÿ2C肾上腺素能受体相关的一种或多种病症的方法。
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2.Substituted spirocyclic piperidine derivatives as histamine-3 (H3) receptor ligands 失效
标题翻译: 取代的螺环哌啶衍生物作为组胺-3(H3)受体配体公开(公告)号:US08513232B2
公开(公告)日:2013-08-20
申请号:US12846100
申请日:2010-07-29
申请人: Edward R. Bacon , Nadine C. Becknell , Reddeppa reddy Dandu , Lisa Guise-Zawacki , Tao Guo , Chia-yu Huang , Robert L. Hudkins , Babu G. Sundar , Ming Tao , Minglang Wu , Allison L. Zulli
发明人: Edward R. Bacon , Nadine C. Becknell , Reddeppa reddy Dandu , Lisa Guise-Zawacki , Tao Guo , Chia-yu Huang , Robert L. Hudkins , Babu G. Sundar , Ming Tao , Minglang Wu , Allison L. Zulli
IPC分类号: C07D491/10 , C07D401/14 , C07D471/10 , A61K31/397 , A61K31/438 , A61K31/506 , A61P11/00 , A61P1/00 , A61P25/00 , A61P29/00
CPC分类号: C07D491/10
摘要: The present invention provides compounds of Formula (I): their use as H3 antagonists/inverse agonists, processes for their preparation, and pharmaceuticals compositions thereof.
摘要翻译: 本发明提供式(I)化合物:其用作H3拮抗剂/反向激动剂,其制备方法及其药物组合物。
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3.Substituted Spirocyclic Piperidine Derivatives as Histamine-3 (H3) Receptor Ligands 失效
标题翻译: 取代的螺环哌啶衍生物作为组胺-3(H3)受体配体公开(公告)号:US20110071131A1
公开(公告)日:2011-03-24
申请号:US12846100
申请日:2010-07-29
申请人: Edward R. Bacon , Nadine C. Becknell , Reddeppa reddy Dandu , Lisa Guise-Zawacki , Tao Guo , Chia-yu Huang , Robert L. Hudkins , Babu G. Sundar , Ming Tao , Minglang Wu , Allison L. Zulli
发明人: Edward R. Bacon , Nadine C. Becknell , Reddeppa reddy Dandu , Lisa Guise-Zawacki , Tao Guo , Chia-yu Huang , Robert L. Hudkins , Babu G. Sundar , Ming Tao , Minglang Wu , Allison L. Zulli
IPC分类号: A61K31/397 , C07D471/10 , A61K31/438 , C07D413/14 , A61K31/5377 , C07D401/14 , A61K31/506 , A61P25/00 , A61P1/00 , A61P11/00 , A61P9/00 , A61P29/00
CPC分类号: C07D491/10
摘要: The present invention provides compounds of Formula (I): their use as H3 antagonists/inverse agonists, processes for their preparation, and pharmaceuticals compositions thereof.
摘要翻译: 本发明提供式(I)化合物:其用作H3拮抗剂/反向激动剂,其制备方法及其药物组合物。
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