摘要:
This invention provides novel isatin compounds which are useful as therapeutic agents. The invention isatin compounds and the pharmaceutically acceptable salts thereof exhibit anti-ulcer activities which are applicable for propylaxis and treatment of ulcer diseases in the digestive tract of animals.
摘要:
The imidazole derivatives of the general formula: ##STR1## wherein A and B may be the same or different, and each is a straight- or branched-chain alkylene or alkenylene group having 1 to 8 carbon atoms, D is an acyl group having 2 to 10 carbon atoms, an alkoxycarbonyl group having 2 to 7 carbon atoms or a dialkoxymethyl group having 3 to 13 carbon atoms, Q is a cyano group or an alkoxycarbonyl group having 2 to 7 carbon atoms, X is a halogen atom, Z is ##STR2## (wherein E is a hydrogen atom, a halogen atom, an alkyl group having 1 to 6 carbon atoms or an alkoxy group having 1 to 6 carbon atoms, Y is an oxygen atom or a sulfur atom and may be connected with either A or B), n is zero or 1, with the proviso that n is 1 when Y connects with B.These compounds are novel compounds and are useful as intermediates in producing 1-substituted imidazole derivatives which possess strong and specific inhibitory effects on thromboxane synthetase and thus are useful as therapeutically active agents for treatment of diseases caused by thromboxane A.sub.2.
摘要:
There is provided a flat antenna apparatus in which a low-noise amplifier provided therein does not generate an abnormal oscillation, and a case and a ground pattern formed on a circuit board are reliably connected to each other by means of a simple construction. A flat antenna element is mounted on a circuit board. The circuit board has an amplifying circuit for amplifying a radio frequency received from the flat antenna element. A case and the flat antenna element are attached to opposite sides of the circuit board. A tab formed on a peripheral edge of the case is inserted into a slot formed on the circuit board, the tab being soldered to fix the case on the circuit board.
摘要:
A novel low thermal expansion cast alloy is provided. The alloy consists of, by percents by weight, 0.02 to 0.25% of C, 30.5 to 33.3% of Ni, 4.0 to 6.0% of Co, 0.005 to 0.70% of Mn, 0.005-0.50% of Si and the balance substantially of Fe, with the proviso that % C.gtoreq.3.0285-0.0936 x % Ni (% C and % Ni are weight % of C and Ni). By such composition, micro-segregation of Ni can be reduced and the Ni content range showing the low thermal expansion coefficient can be broadened to an extent of substantially enabling mass production by a casting process in place of the conventional forging or rolling process. The average thermal expansion coefficient at the temperature range from - 50 to 120.degree. C. of the cast alloy is not more than 1.5.times.10.sup.-6 /.degree.C.
摘要:
A mobile communication method includes a mobile station transmitting a location registration request on the basis of a pilot signal, a network device judging, in response to the received location registration request, whether or not access to a specific radio base station from the mobile station is permitted, the network device rejecting location registration processing when the access is judged not to be permitted, and the network device making a determination so that the transmission power of the pilot signal in the specific radio base station is reduced when the number of rejections of location registration processing exceeds a predetermined number of times.
摘要:
In preferred embodiments this invention provides a pharmaceutical composition and a method for the treatment of allergic conjunctivitis or allergic rhinitis. The composition is an aqueous solution containing N-(3,4-dimethoxycinnamoyl)anthranilic acid or a pharmaceutically acceptable salt thereof as an active ingredient. The composition additionally contains as essential components polyvinylpyrrolidone, a basic compound and a surface active agent in prescribed quantities, and the composition has a pH of about 6.5-8.5.
摘要:
1,3-Disubstituted imidazoles of the general formula (I): ##STR1## wherein A and B may be the same or different, and each is a straight- or branched-chain alkylene or alkenylene group having 1 to 8 carbon atoms, Y is an acyl group having 2 to 10 carbon atoms, an alkoxycarbonyl group having 2 to 7 carbon atoms or an dialkoxymethyl group having 3 to 13 carbon atoms, Z is a cyano group or an alkoxycarbonyl group having 2 to 7 carbon atoms, X is a halogen atom, n is zero or 1. The said compounds are intermediates for producing the imidazole derivatives of the general formula (V) above which possess strong and specific inhibitory effects on thromboxane synthetase and thus are useful as therapeutical agents for treatment of diseases caused by thromboxane A.sub.2.
摘要:
A mobile communication method according to the present invention includes a step A of causing a mobile station in a standby mode in a first cell to transmit a communication start request signal, a step B of judging whether or not to measure communication quality of a second cell on the basis of judgment as to whether or not the particular service is provided in each of the cells and judgment as to whether or not communication quality of the second cell is included in the communication start request signal, the second cell overlaid by the first cell in a different frequency band and a step C of starting communication of the mobile station in either one of the first cell and the second cell on the basis of the measured communication quality of the second cell.
摘要:
A mobile communication method according to the present invention includes a step A of causing a mobile station in a standby mode in a first cell to transmit a communication start request signal, a step B of judging whether or not to measure communication quality of a second cell on the basis of judgment as to whether or not the particular service is provided in each of the cells and judgment as to whether or not communication quality of the second cell is included in the communication start request signal, the second cell overlaid by the first cell in a different frequency band and a step C of starting communication of the mobile station in either one of the first cell and the second cell on the basis of the measured communication quality of the second cell.
摘要:
The present invention provides an improved method for producing a nuclear substituted cinnamoylanthranilic acid compound.Illustrative of the process is the reaction of 3-hydroxy-4-methoxybenzaldehyde with 2-carboxymalonanilic acid in an inert solvent medium in the presence of a molar excess of piperidine to provide a high purity intermediate salt precipitate, and the salt is treated with an acidic reagent to yeild N-(3-hydroxy-4-methoxycinnamoyl)anthranilic acid product.