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公开(公告)号:US08097594B2
公开(公告)日:2012-01-17
申请号:US12379539
申请日:2009-02-24
申请人: Milind Dattatraya Sindkhedkar , Vijaya Narayan Desai , Rajesh Maganlal Loriya , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Rajesh Onkardas Bora , Santosh Devidas Diwakar , Ganesh Rajaram Jadhav , Shivaji Sampatrao Pawar
发明人: Milind Dattatraya Sindkhedkar , Vijaya Narayan Desai , Rajesh Maganlal Loriya , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Rajesh Onkardas Bora , Santosh Devidas Diwakar , Ganesh Rajaram Jadhav , Shivaji Sampatrao Pawar
CPC分类号: C07D493/04
摘要: The present invention provides compounds having antimicrobial activity for preventing and treating diseases caused by microbial infections. Thus, the present invention relates to novel semi-synthetic 11,12-γ lactone macrolides and ketolides having antimicrobial activity, processes for making compounds as well as pharmaceutical compositions containing said compounds as active ingredients and methods of treating microbial infections with the compounds.
摘要翻译: 本发明提供具有抗微生物活性的化合物,其用于预防和治疗由微生物感染引起的疾病。 因此,本发明涉及具有抗微生物活性的新型半合成11,12-γ内酯大环内酯和酮内酯,以及制备化合物的方法以及含有所述化合物作为活性成分的药物组合物以及用该化合物治疗微生物感染的方法。
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公开(公告)号:US20090247478A1
公开(公告)日:2009-10-01
申请号:US12379539
申请日:2009-02-24
申请人: Milind Dattatraya Sindkhedkar , Vijaya Narayan Desai , Rajesh Maganlal Loriya , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Rajesh Onkardas Bora , Santosh Devidas Diwakar , Ganesh Rajaram Jadhav , Shivaji Sampatrao Pawar
发明人: Milind Dattatraya Sindkhedkar , Vijaya Narayan Desai , Rajesh Maganlal Loriya , Mahesh Vithalbhai Patel , Bharat Kalidas Trivedi , Rajesh Onkardas Bora , Santosh Devidas Diwakar , Ganesh Rajaram Jadhav , Shivaji Sampatrao Pawar
IPC分类号: A61K31/7048 , C07H17/08
CPC分类号: C07D493/04
摘要: The present invention provides compounds having antimicrobial activity for preventing and treating diseases caused by microbial infections. Thus, the present invention relates to novel semi-synthetic 11,12-γ lactone macrolides and ketolides having antimicrobial activity, processes for making compounds as well as pharmaceutical compositions containing said compounds as active ingredients and methods of treating microbial infections with the compounds.
摘要翻译: 本发明提供具有抗微生物活性的化合物,其用于预防和治疗由微生物感染引起的疾病。 因此,本发明涉及具有抗微生物活性的新型半合成的11,12-γ-内酯大环内酯和酮内酯,以及制备化合物的方法以及含有所述化合物作为活性成分的药物组合物以及用该化合物治疗微生物感染的方法。
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公开(公告)号:US20120309770A1
公开(公告)日:2012-12-06
申请号:US13310863
申请日:2011-12-05
IPC分类号: A61K31/343 , A61P31/14 , A61K31/443 , A61K31/506 , C07D307/84 , C07D405/14
CPC分类号: C07D405/14 , C07D407/12
摘要: The disclosure provides compounds of formula I, including their salts, as well as compositions and methods of using the compounds. The compounds have activity against hepatitis C virus (HCV) and may be useful in treating those infected with HCV.
摘要翻译: 本公开提供式I化合物,包括其盐,以及使用该化合物的组合物和方法。 该化合物具有抗丙型肝炎病毒(HCV)的活性,可用于治疗HCV感染者。
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公开(公告)号:US08507683B2
公开(公告)日:2013-08-13
申请号:US13310863
申请日:2011-12-05
IPC分类号: C07D471/04 , A61K31/437
CPC分类号: C07D405/14 , C07D407/12
摘要: The disclosure provides compounds of formula I, including their salts, as well as compositions and methods of using the compounds. The compounds have activity against hepatitis C virus (HCV) and may be useful in treating those infected with HCV.
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