Azolyl-derivatives endowed with antifungal activity
    7.
    发明授权
    Azolyl-derivatives endowed with antifungal activity 失效
    具有抗真菌活性的唑基衍生物

    公开(公告)号:US5036094A

    公开(公告)日:1991-07-30

    申请号:US408945

    申请日:1989-09-18

    摘要: Disclosed are compounds, having the general formula: ##STR1## wherein: m=0, 1, 2; n=0, 1 with the condition that when m=0, also n=0;p=0, 1; q=1, 2;X is either oxygen or sulphur;A=N, CH;R is H, CH.sub.3, F;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phe=nyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, haloalkyl=thio, wherein the halogen is Cl, Br, F;R.sub.2 is selected from H, chlorine, bromine, fluorine;R.sub.f is selected from the group formed by alkyls containing from 2 to 4 carbon atoms, and containing at least 4 atoms of halogen selected from F, Cl and Br, of which at least 3 are F atoms; alkenyls and alkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected between Cl and Br.The present invention relates to azolyl-derivatives, more particularly to substituted azolyldioxanes and azolyldioxolanes, endowed with high fungicidal activity, to the process for their preparation, and to their related use in the agrarian field.

    摘要翻译: 公开了具有以下通式的化合物:其中:m = 0,1,2; n = 0,1,条件是当m = 0时,n = 0; p = 0,1, q = 1,2; X是氧或硫; A = N,CH; R为H,CH 3,F; R 1选自氯,溴,氟,CF 3,phe = nyl,C 1 -C 2 - 烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷基=硫代,其中卤素是Cl,Br,F; R2选自H,氯,溴,氟; Rf选自由含有2至4个碳原子的烷基形成的基团,并且含有至少4个选自F,Cl和Br的卤素,其中至少3个是F原子; 含有至多4个碳原子的烯基和炔基,其含有至少2个F原子,以及任选的选自Cl和Br之间的其它卤素。 本发明涉及唑类衍生物,更具体地涉及具有高杀真菌活性的取代的azolyldioxanes和azolyldioxolanes,其制备方法及其在土地领域的相关用途。