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157 条记录 (耗时 0.036 秒)

    Insecticidal and acaricidal plant-protection agents containing substituted 1,2,4-oxadiazole derivatives
    3.
    发明授权
    Insecticidal and acaricidal plant-protection agents containing substituted 1,2,4-oxadiazole derivatives 失效
    含有取代的1,2,4-恶二唑衍生物的杀虫和杀螨植物保护剂

    公开(公告)号：US5428049A

    公开(公告)日：1995-06-27

    申请号：US182124

    申请日：1994-01-13

    申请人： Peter Jeschke ,  Werner Lindner ,  Ulrike Wachendorff-Neumann ,  Christoph Erdelen

    发明人： Peter Jeschke ,  Werner Lindner ,  Ulrike Wachendorff-Neumann ,  Christoph Erdelen

    IPC分类号： A01N43/82 ,  A01N43/824 ,  A01N43/836 ,  A01N47/02 ,  C07D271/06 ,  C07D413/04

    CPC分类号： C07D271/06 ,  A01N43/82 ,  A01N47/02 ,  C07D413/04

    摘要： The present invention relates to the use of 1,2,4-oxadiazole derivatives, some of which are already known, as insecticides and acaricides in plant protection.The compounds, used in accordance with the invention, have the formula (I) ##STR1## in which R.sup.1 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aryl or heterocyclyl,R.sup.2 represents hydrogen, nitro, cyano, carboxyl, carbamoyl or halogen, or represents in each case optionally substituted alkyl, alkoxy or alkylthio,R.sup.3 represents hydrogen, nitro, cyano, carboxyl, carbamoyl or halogen, or represents in each case optionally substituted alkyl, alkoxy or alkylthio, andR.sup.4 has the meaning given in the text of the application.

    摘要翻译： PCT No.PCT / EP92 / 01525 Sec。 371日期1994年1月13日 102（e）日期1994年1月13日PCT提交1992年7月6日PCT公布。 第WO93 / 01719号公报 日期：1993年2月4日。本发明涉及1,2,4-恶二唑衍生物在植物保护中的用途，其中有些已知是杀虫剂和杀螨剂。 根据本发明使用的化合物在每种情况下具有式（I）nts任选取代的烷基，环烷基，芳基或杂环基，R 2表示氢，硝基，氰基，羧基，氨基甲酰基或卤素，或表示 每种情况下任选取代的烷基，烷氧基或烷硫基，R 3表示氢，硝基，氰基，羧基，氨基甲酰基或卤素，或在各种情况下表示任选取代的烷基，烷氧基或烷硫基，R4具有本申请案文中给出的含义。

    Ectoparasiticide agents
    4.
    发明授权
    Ectoparasiticide agents 有权
    杀寄生虫剂

    公开(公告)号：US06630569B1

    公开(公告)日：2003-10-07

    申请号：US09719626

    申请日：2000-12-14

    申请人： Peter Jeschke ,  Andreas Turberg ,  Norbert Mencke ,  Olaf Hansen

    发明人： Peter Jeschke ,  Andreas Turberg ,  Norbert Mencke ,  Olaf Hansen

    IPC分类号： C07K750

    CPC分类号： A01N43/84 ,  A01N43/72

    摘要： The present invention relates to the ectoparasiticidal use of cyclic depsipeptides of the formula (I) in which R1, R2, R3, R4, X1, X2, X3 and X4 are substituents described herein, which are effective for controlling ectoparasites, and to ectoparasiticidal compositions containing the depsipeptides.

    摘要翻译： 本发明涉及式（I）的环状缩肽，其中R 1，R 2，R 3，R 4，X 1，X 2，X 2， 3＆gt;和X 4是本文描述的对控制外寄生物有效的取代基，以及含有脱脂肽的外寄生植物杀伤组合物。

    Octacyclodepsipeptides having an endoparasiticidal action
    7.
    发明授权
    Octacyclodepsipeptides having an endoparasiticidal action 失效
    具有内寄生性杀伤作用的Octacyclodepsipeptide

    公开(公告)号：US06369028B1

    公开(公告)日：2002-04-09

    申请号：US08246029

    申请日：1994-05-19

    申请人： Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    发明人： Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    IPC分类号： A61K3800

    CPC分类号： C07D273/00 ,  C07C235/12 ,  C07C235/34

    摘要： The present invention relates to compounds of the general formula (I) in which R1, R2, R11 and R12 represent the same or different radicals selected from the group of C1-8-alkyl, C1-8-halogenoalkyl, C3-6-cycloalkyl, aralkyl or aryl, R3, R5, R7, R9, represent the same or different radicals selected from the group of hydrogen or straight-chain C1-5-alkyl or branched C4-7-alkyl which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl  carboxamide,  imidazolyl, indolyl, guanidino, —SH or C1-4-alkylthio, and furthermore represents aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, nitro or a —NR13R14 group in which R13 and R14 independently from each other represent hydrogen or alkyl or together with the adjoining nitrogen atom forms a 5, 6 or 7-membered ring which is optionally interrupted by O, S or N and which is optionally C1-4-alkyl substituted, R4, R6, R8, R10 represent the same or different radicals selected from the group of hydrogen, straight-chain C1-5-alkyl and represents isopropyl, sec.-butyl, t-butyl, C2-6-alkenyl, C3-7-cycloalkyl, which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl, carboxamide, imidazolyl, indolyl, guanidino, SH or C1-4-alkylthio and represent aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, and stereoisomers thereof, to processes for their preparation and to their use as endoparasiticides.

    摘要翻译： 本发明涉及通式（I）的化合物，其中R 1，R 2，R 11和R 12表示相同或不同的选自C 1-8 - 烷基，C 1-8 - 卤代烷基，C 3-6 - 环烷基， 芳烷基或芳基，R 3，R 5，R 7，R 9表示相同或不同的选自氢或直链C 1-5烷基或支链C 4-7 - 烷基的基团，其可任选被羟基，C 1-4 烷氧基，羧基羧酰胺，咪唑基，吲哚基，胍基，-SH或C 1-4 - 烷硫基，此外表示可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基，硝基取代的芳基，芳烷基或杂芳基甲基 或-NR 13 R 14基团，其中R 13和R 14彼此独立地表示氢或烷基或与相邻的氮原子一起形成可选地被O，S或N中断的5,6或7-元环，并且其任选地为C1 R 4，R 6，R 8，R 10表示选自该基团的相同或不同的基团 的氢，直链C1-5 - 烷基，代表异丙基，仲丁基，叔丁基，C 2-6 - 烯基，C 3-7 - 环烷基，其可任选被羟基，C 1-4 - 烷氧基， 羧基，羧酰胺，咪唑基，吲哚基，胍基，SH或C 1-4 - 烷硫基，代表可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基及其立体异构体取代的芳基，芳烷基或杂芳基甲基， 其制备方法及其作为内寄生物杀虫剂的用途。

    Substituted 1,2,4-oxadiazole derivatives
    9.
    发明授权
    Substituted 1,2,4-oxadiazole derivatives 失效
    取代的1,2,4-恶二唑衍生物

    公开(公告)号：US5371231A

    公开(公告)日：1994-12-06

    申请号：US57584

    申请日：1993-05-05

    申请人： Peter Jeschke ,  Werner Lindner ,  Achim Harder ,  Norbert Mencke ,  Axel Haberkorn

    发明人： Peter Jeschke ,  Werner Lindner ,  Achim Harder ,  Norbert Mencke ,  Axel Haberkorn

    IPC分类号： A61K31/41 ,  A01N43/82 ,  A01N43/836 ,  A61K31/4245 ,  A61P33/00 ,  A61P33/10 ,  C07D271/06

    CPC分类号： C07D271/06 ,  A01N43/82

    摘要： The present invention relates to new substituted 1,2,4-oxadiazole derivatives of the formula (I) and to their stereoisomers ##STR1## in which formula R.sup.4 represents OH, SH, halogenoalkoxy, halogenoalkylthio, halogenoalkylsulphinyl, halogenoalkylsulphonyl, aryloxy, aralkoxy, arylthio, aralkylthio, alkylenedioxy, halogenoalkylenedioxy, amino, alkylamino, dialkylamino, acylamino, carbamoyl, alkylsulphinyl, alkylsulphonyl, arylsuphinyl, arylsulphonyl, sulphonylamino, alkoxycarbonyl, alkylcarbonyl, alkylcarbonyloxy, alkoxyalkyl, alkoxyalkoxy or hydroxyalkoxy, where in the event that at least one of the radicals R.sup.2 or R.sup.3 is other than hydrogen, R.sup.4 additionally represents halogen, alkyl, halogenoalkyl, alkoxy or thioalkyl, where, in the event that R.sup.1 represents optionally substituted C.sub.1-8 -alkyl, R.sup.4 additionally represents alkoxy,processes for their preparation, and their use as endoparasiticides.

    摘要翻译： 本发明涉及式（I）的新的取代的1,2,4-恶二唑衍生物及其立体异构体，其中式R4代表OH，SH，卤代烷氧基，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基，芳氧基， 芳烷氧基，芳硫基，芳烷硫基，亚烷基二氧基，卤代亚烷基二氧基，氨基，烷基氨基，二烷基氨基，酰基氨基，氨基甲酰基，烷基亚磺酰基，烷基磺酰基，芳基亚乙基，芳基磺酰基，磺酰基氨基，烷氧基羰基，烷基羰基，烷基羰基氧基，烷氧基烷基，烷氧基烷氧基或羟基烷氧基，其中在至少一个 基团R2或R3不是氢，R4另外表示卤素，烷基，卤代烷基，烷氧基或硫代烷基，其中，在R 1表示任选取代的C 1-8 - 烷基的情况下，R 4另外表示烷氧基，其制备方法， 并将其用作内寄生物杀灭剂。