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    Isoxazoline derivatives as insecticidal compounds
    1.
    发明授权
    Isoxazoline derivatives as insecticidal compounds 有权
    异恶唑啉衍生物作为杀虫剂

    公开(公告)号：US09247740B2

    公开(公告)日：2016-02-02

    申请号：US14240428

    申请日：2012-08-24

    申请人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    发明人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    IPC分类号： C07D413/12 ,  C07D331/04 ,  A01N43/20 ,  A01N43/80 ,  A01N43/40 ,  A01N43/54

    CPC分类号： A01N43/20 ,  A01N43/40 ,  A01N43/54 ,  A01N43/80 ,  C07D331/04 ,  C07D413/12

    摘要： The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译： 本发明提供式（I）化合物，其中G1是氧; R1是氢; R2是基团P（P）L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R4）R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6，CH或氮; Y2和Y3独立地是CH或氮; 其中Y1，Y2和Y3中不超过两个是氮，并且其中Y 2和Y 3不都是氮; R5是氢，卤素，氰基，硝基，NH2，C1-C2烷基，C1-C2卤代烷基，C3-C5环烷基，C3-C5卤代环烷基，C1-C2烷氧基，C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式（I）化合物的中间体，以及使用式（I）化合物控制昆虫，螨虫，线虫或软体动物的方法。

    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS
    2.
    发明申请
    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 有权
    异辛唑衍生物作为杀虫剂化合物

    公开(公告)号：US20140206606A1

    公开(公告)日：2014-07-24

    申请号：US14240428

    申请日：2012-08-24

    申请人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    发明人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    IPC分类号： A01N43/80 ,  A01N43/40 ,  A01N43/54 ,  A01N43/20

    CPC分类号： A01N43/20 ,  A01N43/40 ,  A01N43/54 ,  A01N43/80 ,  C07D331/04 ,  C07D413/12

    摘要： The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译： 本发明提供式（I）化合物，其中G1是氧; R1是氢; R2是基团P（P）L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R4）R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6，CH或氮; Y2和Y3独立地是CH或氮; 其中Y1，Y2和Y3中不超过两个是氮，并且其中Y 2和Y 3不都是氮; R5是氢，卤素，氰基，硝基，NH2，C1-C2烷基，C1-C2卤代烷基，C3-C5环烷基，C3-C5卤代环烷基，C1-C2烷氧基，C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式（I）化合物的中间体，以及使用式（I）化合物控制昆虫，螨虫，线虫或软体动物的方法。

    Process for the preparation of dihydropyrrole derivatives
    8.
    发明授权
    Process for the preparation of dihydropyrrole derivatives 有权
    二氢吡咯衍生物的制备方法

    公开(公告)号：US09233920B2

    公开(公告)日：2016-01-12

    申请号：US13703630

    申请日：2011-06-14

    申请人： Myriem El Qacemi ,  Helmars Smits ,  Jerome Yves Cassayre ,  Nicholas Phillip Mulholland ,  Peter Renold ,  Edouard Godineau ,  Thomas Pitterna

    发明人： Myriem El Qacemi ,  Helmars Smits ,  Jerome Yves Cassayre ,  Nicholas Phillip Mulholland ,  Peter Renold ,  Edouard Godineau ,  Thomas Pitterna

    IPC分类号： C07D207/46 ,  C07D207/20 ,  C07D401/04 ,  C07D413/12 ,  C07D413/14 ,  C07D417/14 ,  A01N43/36

    CPC分类号： C07D207/46 ,  A01N43/36 ,  C07D207/20 ,  C07D401/04 ,  C07D413/12 ,  C07D413/14 ,  C07D417/14

    摘要： The present invention provides stereoselective processes for the preparation of compounds of formula (I) wherein P is phenyl, naphthyl, a 6-membered heteroaryl group containing one or two nitrogen atoms as ring members, or a 10-membered bicyclic heteroaryl group containing one or two nitrogen atoms as ring members, and wherein the phenyl, naphthyl and heteroaryl groups are optionally substituted; R1 is chlorodifluoromethyl or trifluoromethyl; R2 is optionally substituted aryl or optionally substituted heteroaryl; n is 0 or 1; including the process comprising (a-i) reacting a compound of formula II wherein P, R1 and R2 are as defined for the compound of formula I; with nitromethane in the presence a chiral catalyst to give a compound of formula III Wherein P, R1 and R2 are as defined for the compound of formula I; and (a-ii) reductively cyclizing the compound of formula III to give the compound of formula I. The invention also provides intermediates useful for processes for the synthesis of compounds of formula (I).

    摘要翻译： 本发明提供了制备式（I）化合物的立体选择性方法，其中P是苯基，萘基，含有一个或两个氮原子作为环成员的6元杂芳基或含有一个或多个氮原子的10元双环杂芳基 两个氮原子作为环成员，并且其中苯基，萘基和杂芳基任选被取代; R1是氯二氟甲基或三氟甲基; R2是任选取代的芳基或任选取代的杂芳基; n为0或1; 包括（a-i）使式II化合物与式Ⅰ化合物反应的方法，其中P，R 1和R 2如对式I化合物所定义; 在硝基甲烷中存在手性催化剂，得到式III化合物，其中P，R 1和R 2如式I化合物所定义; 和（a-ii）将式III化合物还原性环化得到式I化合物。本发明还提供了可用于合成式（I）化合物的方法的中间体。

    Isoxazoline derivatives as insecticides
    9.
    发明授权
    Isoxazoline derivatives as insecticides 有权
    异恶唑啉衍生物作为杀虫剂

    公开(公告)号：US08754053B2

    公开(公告)日：2014-06-17

    申请号：US13579637

    申请日：2011-02-17

    申请人： Thomas Pitterna ,  Myriem El Qacemi ,  Jerome Yves Cassayre ,  Peter Renold ,  Vladimir Bobosik

    发明人： Thomas Pitterna ,  Myriem El Qacemi ,  Jerome Yves Cassayre ,  Peter Renold ,  Vladimir Bobosik

    IPC分类号： A01N43/80 ,  C07D261/04 ,  C07D413/10 ,  C07D413/12 ,  C07D417/12

    CPC分类号： C07D261/04 ,  A01N43/80 ,  C07D413/10 ,  C07D413/12 ,  C07D417/12

    摘要： The present invention relates to compounds formula (I), wherein P is P1, P2, heterocyclyl or heterocyclyl substituted by one to five Z; and wherein A1, A2, A3, A4, G1, R1, R2, R3, R4, R5, R6, R17, R18, R19 and R20 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.

    摘要翻译： 本发明涉及式（I）化合物，其中P为P1，P2，被1至5个Z取代的杂环基或杂环基; 并且其中A1，A2，A3，A4，G1，R1，R2，R3，R4，R5，R6，R17，R18，R19和R20如权利要求1中所定义; 或其盐或N-氧化物。 此外，本发明涉及制备式（I）化合物的方法和中间体，其包含式（I）化合物的杀虫，杀螨，杀线虫和杀软体动物的组合物和使用式（I）化合物控制的方法 昆虫，螨虫，线虫和软体动物害虫。