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    4-amino-quinolines
    5.
    发明授权
    4-amino-quinolines 失效
    4-氨基喹啉

    公开(公告)号：US3808216A

    公开(公告)日：1974-04-30

    申请号：US24140572

    申请日：1972-04-05

    Applicant: ROUSSEL UCLAF

    Inventor： CEREDE J ,  ALLAIS A ,  MEIER J

    IPC: C07D409/12 ,  A61K31/47 ,  C07D417/12 ,  C07D33/60

    CPC classification number: A61K31/47

    Abstract: NOVEL 4-AMINO-QUINOLINES OF THE FORMULA

    4-(X-OOC-Y-NH-),R,R1-QUINOLINE

    WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, HALOGEN, -CF3, LOWER ALKYL, LOWER ALKOXY, LOWER ALKYLSULFONYLOXY, LOWER ALKYLTHIO, NITRO, LOWER ALKYLAMINO, LOWER ACYLAMINO AND CYANO, R1 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, CHLORINE AND METHYL, Y IS SELECTED FROM THE GROUP CONSISTING OF 2,3 AND 3,4-DISUBSTITUTED THIOPHENES OF THE FORMULA

    R2-THIEN-2,3-YLENE AND R2-THIEN-3,4-YLENE

    AND 4,5-DISUBSTITUTED THIAZOLES OF THE FORMULA

    2-Q-THIAZOL-4,5-YLENE

    WHEREIN R2 AND Q ARE SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND LOWER ALKYL AD X IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, LOWER ALKYL, A PHENYL, DILOWERALKYLAMINO LOWER ALKYLENE, N-MORPHOLINO LOWER ALKYLENE,

    -CH2-CH(-O-R3)-CH2-O-R4, 2-P2-1,3-DIOXAN-5-YL, AND

    -(CH2)N-N(+)(-M'')2-M Z(-),

    R3 AND R4 BEING HYDROGEN AND TAKEN TOGETHER FORM

    -C(-P)(-P1)-

    P AND P1 ARE LOWER ALKYL, P2 IS SELECTED FROM THE GROUP CONSISTING OF LOWER ALKYL AND MONOCYCLIC ARYL, M AND M'' ARE LOWER ALKYL, Z IS HALOGEN AND N IS AN INTEGER FROM 1 TO 6, AND THEIR NON-TOXIC, PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS HAVING ANALGESIC AND ANTI-INFLAMMATORY ACTIVITY AND THEIR PREPARATION. LOWER ALKYL MEANS HAVING 1 TO 6 CARBON ATOMS.

    Tetrahydropyranyl and tetrahydrothiapyranyl phenylacetic acid compounds
    6.
    发明授权
    Tetrahydropyranyl and tetrahydrothiapyranyl phenylacetic acid compounds 失效
    四氢呋喃和四氢萘甲酸苯甲酸化合物

    公开(公告)号：US3772332A

    公开(公告)日：1973-11-13

    申请号：US3772332D

    申请日：1972-04-12

    Applicant: ROUSSEL UCLAF

    Inventor： ALLAIS A ,  MEIER J ,  DUBE J

    IPC: C07D335/02 ,  C07D309/02 ,  C07D309/04 ,  C07D309/06 ,  A61K27/00 ,  C07D65/04

    CPC classification number: C07D309/06 ,  C07D309/04

    Abstract: NOVEL COMPOUNDS OF THE FORMULA

    (2-HAL,4-(R-OOC-Z-)PHENYL)-CH
    WHEREIN X IS SELECTED FROM THE GROUP CONSISTING OF OXYGEN, SULFUR, SO AND SO2, R IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ANION OF A NON-TOXIC; THERAPEUTICALLY ACCEPTABLE ORGANIC OR MINERAL BASE AND RESIDUE OF AN ALCOHOL, AN Z IS SELCETED FROM THE GROUP CONSISTING OF -CHR1- AND >C=R2 WHEREIN R1 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND STRAINGT OR BRANCHED ALKYL OF 1 TO 4 CARBON ATOMS, AND R2 IS A STRAIGHT OR BRANCHED ALKYLIDENE OF 1 TO 4 CARBON ATOMS AND HAL IS SELECTED FROM THE GROUP CONSISTING OF FLUORINE, BROMINE AND CHLORINE, WHICH COMPOUNDS WHICH CONTAIN AT LEAST ONE ASYMMETRIC CARBON ATOM CAN BE IN RACEMIC OR OPTICALLY ACTIVE GORM, AND THEIR PREPARATION WHICH COMPOUNDS HAVE ANALGESIC AND ANTIINFLAMMATORY ACTIVITY.

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