6-Substituted 2,4-diamino-1,3,5-triazine derivatives having at least two asymmetrically substituted carbon atoms, the production thereof, and their use as herbicides
    4.
    发明授权
    6-Substituted 2,4-diamino-1,3,5-triazine derivatives having at least two asymmetrically substituted carbon atoms, the production thereof, and their use as herbicides 失效
    具有至少两个不对称取代的碳原子的6-取代的2,4-二氨基-1,3,5-三嗪衍生物,其制备及其作为除草剂的用途

    公开(公告)号:US06358886B1

    公开(公告)日:2002-03-19

    申请号:US09623612

    申请日:2000-11-03

    IPC分类号: C07D25118

    摘要: The invention relates to novel substituted optically active aminotriazines having at least two asymmetrically substituted carbon atoms of the formula (I), in which A represents a single bond or represents in each case straight-chain or branched alkanediyl or oxaalkanediyl having in each case up to 6 carbon atoms, Z represents certain carbocyclic or heterocyclic radicals and the substituents R1, R2, R3, R4 and Y are as defined in the description,  with the proviso that in each individual case R2, R3 and Y are different from one another and that the substituents at the two carbon atoms to which R2 and R3 or R4 are attached are configured as follows: (a) R configuration at the carbon atom to which R2 and R3 are attached and R configuration at the carbon atom to which R4 is attached (“R,R-diastereomers”), (b) R configuration at the carbon atom to which R2 and R3 are attached and S configuration at the carbon atom to which R4 is attached (“R,S-diastereomers”), (c) S configuration at the carbon atom to which R2 and R3 are attached and R configuration at the carbon atom to which R4 is attached (“S,R-diastereomers”), (d) S configuration at the carbon atom to which R2 and R3 are attached and S configuration at the carbon atom to which R4 is attached (“S,S-diastereomers”), (e) R configuration at the carbon atom to which R2 and R3 are attached and racemic configuration at the carbon atom to which R4 is attached (“R,racdiastereomers”), (f) S configuration at the carbon atom to which R2 and R3 are attached and racemic configuration at the carbon atom to which R4 is attached (“S,rac-diastereomers”), and to a process for preparing the compounds of the formula (I) and to their use as herbicides.

    摘要翻译: 本发明涉及具有式(I)的至少两个不对称取代的碳原子的新的取代的光学活性氨基三嗪,其中A表示单键或表示在每种情况下为直链或支链烷二基或氧杂烷二基,在每种情况下最多为6 碳原子,Z表示某些碳环或杂环基团,并且取代基R 1,R 2,R 3,R 4和Y如说明书中所定义,条件是在各个别情况下,R 2,R 3和Y彼此不同, R2和R3或R4连接的两个碳原子上的取代基配置如下:(a)R 2和R 3连接的碳原子上的R构型,R 4连接的碳原子上的R构型(“ R,R非对映异构体“),(b)R 2和R 3连接的碳原子上的R构型,R 4连接的碳原子上的S构型(”R,S-非对映异构体“),(c)S 配置在碳ato m与R 2相连的碳原子上的R构型(“S,R-非对映异构体”),(d)在R2和R3所连接的碳原子上的S构型, R 4连接的碳原子(“S,S-非对映异构体”),(e)R 2和R 3所连接的碳原子上的R构型,R 4连接的碳原子上的外消旋构型(“R” 外消旋异构体“),(f)R 2和R 3所连接的碳原子上的S构型以及与R4连接的碳原子上的外消旋构型(”S,外消旋 - 非对映体“),以及制备该化合物的方法 的式(I)和它们作为除草剂的用途。

    Substituted thiazol(in) ylideneamino sulfonylamino (thio)carbonyl-triazolinones
    9.
    发明授权
    Substituted thiazol(in) ylideneamino sulfonylamino (thio)carbonyl-triazolinones 失效
    取代的噻唑(亚)氨基磺酰基氨基(硫代)羰基 - 三唑啉酮

    公开(公告)号:US06403535B1

    公开(公告)日:2002-06-11

    申请号:US09787479

    申请日:2001-04-27

    IPC分类号: A01N4738

    CPC分类号: C07D417/12 A01N47/38

    摘要: The invention relates to novel substituted thiazol(in)ylidenaminosulphonyl-amino(thio)carbonyl-triazolinones of the formula (I) in which Q represents oxygen or sulphur, R1 represents hydrogen, amino, alkylideneamino or represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkylamino, dialkylamino, alkanoylamino, alkenyl, alkinyl, alkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl and arylalkyl, R2 represents hydrogen, cyano, halogen or represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, alkenyl, alkinyl, alkenyloxy, alkenylthio, alkenylamino, cycloalkyl, cycloalkylalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, aryl, aryloxy, arylthio, arylamino, arylalkyl, arylalkoxy, arylalkylthio and arylalkylamino, R3 represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl and arylalkyl, R4 represents hydrogen, cyano, halogen or optionally substituted alkyl, R5 represents hydrogen, cyano, halogen or optionally substituted alkyl, and to salts of compounds of the formula (I), to processes for preparing the novel compounds and to their use as herbicides.

    摘要翻译: 本发明涉及式(I)中的新的取代的噻唑(亚氨基)磺酰基 - 氨基(硫代)羰基 - 三唑啉酮,其中Q表示氧或硫,R 1表示氢,氨基,亚烷基氨基或代表任意取代的基团, 由烷基,烷氧基,烷基氨基,二烷基氨基,烷酰基氨基,烯基,炔基,烯基氧基,环烷基,环烷基烷基,环烷基氨基,芳基和芳基烷基组成的基团,R 2表示氢,氰基,卤素或表示任意取代的基团, 烷基磺酰基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基,二烷基氨基,烯基,炔基,烯基氧基,烯基硫基,烯基氨基,环烷基,环烷基烷基,环烷氧基,环烷基硫基,环烷基氨基,芳基,芳氧基,芳硫基,芳基氨基,芳基烷基,芳基烷氧基,芳基烷硫基和芳烷基氨基, R 3表示在每种情况下任选取代的基团,其由烷基,烷氧基, 烯基,环烷基,环烷基烷基,芳基和芳烷基,R 4表示氢,氰基,卤素或任选取代的烷基,R 5表示氢,氰基,卤素或任选取代的烷基,以及式(I)化合物的盐, 用于制备新化合物及其作为除草剂的用途。