-
公开(公告)号:US09481698B2
公开(公告)日:2016-11-01
申请号:US14436493
申请日:2013-09-27
Applicant: SANDOZ AG
Inventor: Hubert Sturm , Josef Wieser
IPC: C07F9/6561 , C07F9/6539
CPC classification number: C07F9/65613 , C07F9/65397 , C07F9/65615
Abstract: The present invention relates to a novel process for preparing ceftaroline fosamil as well as to intermediates of this process.
Abstract translation: 本发明涉及一种制备头孢洛林粉剂的新方法以及该方法的中间体。
-
公开(公告)号:US09382278B2
公开(公告)日:2016-07-05
申请号:US14863982
申请日:2015-09-24
Applicant: Sandoz AG
Inventor: Peter Kremminger , Hubert Sturm
IPC: C07D501/08 , C07F9/6561 , C07D417/04 , C07D501/59 , C07C51/41 , C07C303/22 , C07D501/04
CPC classification number: C07F9/65613 , C07C51/41 , C07C303/22 , C07D417/04 , C07D501/04 , C07D501/08 , C07D501/59
Abstract: The present invention relates to a novel process for preparing ceftaroline fosamil via intermediates of Formulae (1), (3) or (4) of this process.
Abstract translation: 本发明涉及通过该方法的式(1),(3)或(4)的中间体制备头孢罗林粉剂的新方法。
-
公开(公告)号:US09534004B2
公开(公告)日:2017-01-03
申请号:US14653122
申请日:2013-12-19
Applicant: Sandoz AG
Inventor: Josef Wieser , Hubert Sturm , Arthur Pichler , Andreas Hotter , Nolwenn Martin , Christoph Langes , Ulrich Griesser
IPC: C07F9/6561
CPC classification number: C07F9/6561 , C07F9/65613
Abstract: The present invention relates to novel crystalline forms of ceftaroline fosamil and to methods for their preparation. Furthermore the present invention relates to the use of the novel forms of ceftaroline fosamil for the preparation of an antibiotic medicament. In addition the present invention relates to pharmaceutical compositions comprising an effective amount of the novel forms of ceftaroline fosamil and to methods of preparing the same. Finally the present invention relates to pharmaceutical combinations comprising an effective amount of the novel forms of ceftaroline fosamil and β-lactamase inhibitors.
Abstract translation: 本发明涉及头孢洛林粉末的新型结晶形式及其制备方法。 此外,本发明涉及新型形式的头孢洛林粉剂用于制备抗生素药物的用途。 此外,本发明涉及包含有效量的头孢洛罗松受体的新形式的药物组合物及其制备方法。 最后,本发明涉及包含有效量的新型形式的头孢噻吩福沙米和β-内酰胺酶抑制剂的药物组合。
-
4.
公开(公告)号:US20160200750A1
公开(公告)日:2016-07-14
申请号:US14653122
申请日:2013-12-19
Applicant: SANDOZ AG
Inventor: Josef Wieser , Hubert Sturm , Arthur Pichler , Andreas Hotter , Nolwenn Martin , Christoph Langes , Ulrich Griesser
IPC: C07F9/6561
CPC classification number: C07F9/6561 , C07F9/65613
Abstract: The present invention relates to novel crystalline forms of ceftaroline fosamil and to methods for their preparation. Furthermore the present invention relates to the use of the novel forms of ceftaroline fosamil for the preparation of an antibiotic medicament. In addition the present invention relates to pharmaceutical compositions comprising an effective amount of the novel forms of ceftaroline fosamil and to methods of preparing the same. Finally the present invention relates to pharmaceutical combinations comprising an effective amount of the novel forms of ceftaroline fosamil and β-lactamase inhibitors.
Abstract translation: 本发明涉及头孢洛林粉末的新型结晶形式及其制备方法。 此外,本发明涉及新型形式的头孢洛林粉剂用于制备抗生素药物的用途。 此外,本发明涉及包含有效量的头孢洛罗松受体的新形式的药物组合物及其制备方法。 最后,本发明涉及药物组合,其包含有效量的新型形式的头孢洛罗Fosamil和β-内酰胺酶抑制剂。
-
公开(公告)号:USRE47787E1
公开(公告)日:2019-12-31
申请号:US16058177
申请日:2018-08-08
Applicant: SANDOZ AG
Inventor: Hubert Sturm , Josef Wieser
IPC: C07F9/6561 , C07F9/6539
Abstract: The present invention relates to a novel process for preparing ceftaroline fosamil as well as to intermediates of this process.
-
公开(公告)号:US20160264628A1
公开(公告)日:2016-09-15
申请号:US15162253
申请日:2016-05-23
Applicant: SANDOZ AG
Inventor: Roland Barth , Kerstin Knepper , Hubert Sturm
IPC: C07K7/64
CPC classification number: C07K7/64 , C07D261/08 , C07D413/12 , C07D413/14 , C07D417/12 , C07F9/653 , C07K7/56
Abstract: The present invention relates to the preparation of compounds, in particular to the preparation of compounds of formula (I), which may be used with a compound of formula (VI), or a salt thereof as intermediates for the preparation of antifungal agents, preferably micafungin (MICA) or a salt thereof.
-
7.
公开(公告)号:US20160046655A1
公开(公告)日:2016-02-18
申请号:US14436493
申请日:2013-09-27
Applicant: SANDOZ AG
Inventor: Hubert Sturm , Josef Wieser
IPC: C07F9/6561
CPC classification number: C07F9/65613 , C07F9/65397 , C07F9/65615
Abstract: The present invention relates to a novel process for preparing ceftaroline fosamil as well as to intermediates of this process.
Abstract translation: 本发明涉及一种制备头孢洛林粉剂的新方法以及该方法的中间体。
-
-
-
-
-
-