Iminothiazolines, their production and use as herbicides
    3.
    发明授权
    Iminothiazolines, their production and use as herbicides 失效
    异噻唑啉,其生产和用作除草剂

    公开(公告)号:US5292715A

    公开(公告)日:1994-03-08

    申请号:US936516

    申请日:1992-08-28

    摘要: There is disclosed an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(lower)alkyl, halo(lower)alkoxy or halo(lower)alkylthio; R.sup.2 is methyl, ethyl, chlorine, bromine or iodine; R.sup.3 is lower alkyl, lower cycloalkyl, lower alkoxy, lower cycloalkoxy, lower alkylamino, phenylamino or phenyl, all of which are optionally substituted with at least one substituent selected from halogen, lower alkyl, lower alkoxy, halo(lower)alkyl, lower cycloalkyl and lower cycloalkoxy; and R.sup.4 is hydrogen or halogen. Also disclosed are a process for producing this compound, a herbicidal composition comprising this compound as an active ingredient, and a method for controlling undesired weeds by use of this compound as a herbicide.

    摘要翻译: 公开了下式的亚氨基噻唑啉化合物:(*化学结构*)(I)其中R1是卤素,卤代(低级)烷基,卤代(低级)烷氧基或卤代(低级)烷硫基; R2是甲基,乙基,氯,溴或碘; R3是低级烷基,低级环烷基,低级烷氧基,低级环烷氧基,低级烷基氨基,苯基氨基或苯基,它们全部被至少一个选自卤素,低级烷基,低级烷氧基,卤代(低级)烷基,低级环烷基 和低级环烷氧基; R4是氢或卤素。 还公开了制备该化合物的方法,包含该化合物作为活性成分的除草组合物,以及通过使用该化合物作为除草剂来控制不需要的杂草的方法。

    Herbicidal composition
    7.
    发明授权
    Herbicidal composition 失效
    除草成分

    公开(公告)号:US5312798A

    公开(公告)日:1994-05-17

    申请号:US944084

    申请日:1992-09-11

    CPC分类号: A01N43/78 A01N47/18

    摘要: There is disclosed a herbicidal composition comprising as active ingredients a herbicidally effective amount of (a) an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(C.sub.1 -C.sub.2)alkyl, halo(C.sub.1 -C.sub.2)alkoxy or halo(C.sub.1 -C.sub.2)alkylthio; R.sup.2 is C.sub.1 -c.sub.2 alkyl, chroline, bromine or iodine; R.sup.3 is C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkoxy or C.sub.1 -C.sub.6 alkoxy, all of which are optionally substituted with at least one substituent selected from halogen, C.sub.1 -C.sub.2 alkyl and C.sub.1 -C.sub.2 alkoxy; R.sup.4 is hydrogen or halogen; and (b) at least one of herbicidal triazine compounds, herbicidal uracil compounds, herbicidal urea compounds, herbicidal dinitro aniline compounds, norflurazon, dimethazon, imazaquin and imazethapyr. Also disclosed is a method for controlling undesired weeds by use of the herbicidal composition.

    摘要翻译: 公开了除草组合物,其包含除草有效量的(a)下式的亚氨基噻唑啉化合物:其中R 1是卤素,卤代(C 1 -C 2)烷基,卤代(C 1 -C 2)烷氧基或卤素 (C1-C2)烷硫基; R2是C1-C2烷基,氯原子,溴或碘; R3是C1-C6烷基,C3-C6环烷基,C3-C6环烷氧基或C1-C6烷氧基,它们全部被至少一个选自卤素,C 1 -C 2烷基和C 1 -C 2烷氧基的取代基取代; R4是氢或卤素; 和(b)至少一种除草三嗪化合物,除草尿嘧啶化合物,除草脲化合物,除草二硝基苯胺化合物,诺氟拉津,二甲基噻唑,咪唑啉酮和咪草烟。 还公开了通过使用除草组合物来控制不需要的杂草的方法。

    Oligosaccharide derivatives and process for producing the same
    9.
    发明授权
    Oligosaccharide derivatives and process for producing the same 失效
    寡糖衍生物及其制备方法

    公开(公告)号:US06518249B1

    公开(公告)日:2003-02-11

    申请号:US09485978

    申请日:2000-02-18

    IPC分类号: A61K3170

    CPC分类号: C07H15/04

    摘要: An oligosaccharide derivative, at higher homogeneity than fucose polysaccharide and rhamnose polysaccharide and with greater antiulcer effects, which is represented by the following general formula: Y—OCH(CH2NHR)2 wherein, Y represents an oligofucose or oligorhamnose at a polymerization number of 2 to 20, where the hydroxyl groups may or may not be partially modified in the form of sulfate ester, and R represents phenyl group, a higher alkylphenyl group, a higher alkyl group or —(CH2)n—NHX wherein n is an integer of 1 to 10 and X represents a higher alkanoyl group or an alkylamino group.

    摘要翻译: 一种低聚糖衍生物,其比岩藻糖多糖和鼠李糖多糖具有更高的均一性,并且具有较大的抗溃疡作用,其由以下通式表示:其中Y表示聚合数为2至20的寡聚核糖或寡鼠李糖,其中羟基可以 或可以不以硫酸酯的形式部分修饰,R代表苯基,高级烷基苯基,高级烷基或 - (CH2)n-NHX,其中n为1至10的整数,X表示较高的 烷酰基或烷基氨基。

    Antibacterial agents and process for producing the same
    10.
    发明授权
    Antibacterial agents and process for producing the same 失效
    抗菌剂及其制造方法

    公开(公告)号:US07498317B2

    公开(公告)日:2009-03-03

    申请号:US11049423

    申请日:2005-02-02

    IPC分类号: A61K31/731 A61K31/737

    摘要: An antibacterial agent showing a high affinity for Helicobactor pyroli and having an antibacterial effect specific to H. Pyroli. The agent has a chemical structure wherein an antibacterial substance is bonded to a sulfated polysaccharide or an oligosaccharide prepared by partial decomposition of the sulfated polysaccharide. Preferable embodiments are those having the chemical structure represented by Y—OCH(AH2NHR)n or Y—BH2NHR, wherein Y represents a sulfated polysaccharide or an oligosaccharide prepared by partial decomposition of the sulfated polysaccharide; A a carbon derived from aldehyde group occurring through the reduction of the reduced end sugar of Y and subsequent oxidation of the resulting product with an oxidant; B a carbon derived from the aldehyde group at the reduced end sugar of Y; R an antibacterial substance with a primary amino group or with an amino group introduced therein or represents an antibacterial substance derivative prepared by bonding an antibacterial substance through a spacer to the carbon A or the carbon B; and n=1 or 2.

    摘要翻译: 对Helicobactor pyroli具有高亲和力并具有对H. Pyroli特异性的抗菌作用的抗菌剂。 该药剂具有抗菌物质与通过硫酸化多糖的部分分解制备的硫酸化多糖或寡糖结合的化学结构。 优选的实施方案是具有由Y-OCH(AH2NHR)n或Y-BH2NHR表示的化学结构的那些,其中Y表示硫酸化多糖或通过硫酸化多糖的部分分解制备的寡糖; 衍生自醛基的碳通过还原末端糖的Y而发生,随后用氧化剂氧化所得产物; B是衍生自Y的还原末端糖的醛基的碳; R是具有伯氨基或在其中引入氨基的抗菌物质,或代表通过间隔剂将抗菌物质与碳A或碳B结合而制备的抗菌物质衍生物; n = 1或2。