Crystals of 5-[{6-(2-fluorobenzyl)oxy-2-naphthyl}methyl]-2,4-thiazolidinedione
    1.
    发明授权
    Crystals of 5-[{6-(2-fluorobenzyl)oxy-2-naphthyl}methyl]-2,4-thiazolidinedione 失效
    5 - [{6-(2-氟苄基)氧基-2-萘基}甲基] -2,4-噻唑烷二酮的晶体

    公开(公告)号:US06541493B1

    公开(公告)日:2003-04-01

    申请号:US09856295

    申请日:2001-08-20

    IPC分类号: C07D27734

    CPC分类号: C07D277/34

    摘要: The invention relates to type A crystal of 5-[{6-(2-fluorobenzyl)oxy-2-naphthyl}methyl]-2,4-thiazolidinedione characterized to have characteristic absorption peaks (2&thgr;) at 11.5°±0.3°, 14.5°±0.2°, 16.2°±0.3°, 17.0°±0.3°, 17.7°±0.2°, 18.6°±0.3°, 19.1°±0.2°, 21.3°±0.4°, 22.4°±0.5°, 25.7°±0.5° and 28.3°±0.5° in a powder X-ray diffraction pattern, and also to a method for preparation thereof, and a pharmaceutical composition comprising the same. The crystal is excellent in stability, and has advantages in handling, storage, and pharmaceutical preparation. The invention also relates to type B, C and D crystals of said compound.

    摘要翻译: 本发明涉及5 - [{6-(2-氟苄基)氧基-2-萘基}甲基] -2,4-噻唑烷二酮的A型晶体,其特征在于在11.5°±0.3°,14.5°具有特征吸收峰(2θ) °±0.2°,16.2°±0.3°,17.0°±0.3°,17.7°±0.2°,18.6°±0.3°,19.1°±0.2°,21.3°±0.4°,22.4°±0.5°,25.7°± 粉末X射线衍射图中为0.5°和28.3°±0.5°,以及其制备方法,以及包含该方法的药物组合物。 该晶体的稳定性优异,在处理,储存和制药方面具有优势。 本发明还涉及所述化合物的B,C和D型晶体。

    Crystals of 5-[{6-(2-fluorobenzyl)oxy-2-naphthyl}methyl]-2,4-thiazolidinedione
    2.
    发明申请
    Crystals of 5-[{6-(2-fluorobenzyl)oxy-2-naphthyl}methyl]-2,4-thiazolidinedione 审中-公开
    5 - [{6-(2-氟苄基)氧基-2-萘基}甲基] -2,4-噻唑烷二酮的晶体

    公开(公告)号:US20060149075A1

    公开(公告)日:2006-07-06

    申请号:US11357208

    申请日:2006-02-21

    IPC分类号: C07D277/34

    CPC分类号: C07D277/34

    摘要: The invention relates to type A crystal of 5-[{6-(2-fluorobenzyl)oxy-2-naphtyl}methyl]-2,4-thiazolidinedione characterized to have characteristic absorption peaks (2θ) at 11.5°±0.3°, 14.5°±0.2°, 16.2°±0.3°, 17.0°±0.3°, 17.7°±0.2°, 18.6°±0.3°, 19.1°±0.2°, 21.3°±0.4°, 22.4°±0.5°, 25.7°±1.5° and 28.3°±10.5° in a powder X-ray diffraction pattern, and also to a method for preparation thereof, and a pharmaceutical composition comprising the same. The crystal is excellent in stability, and has advantages in handling, storage, and pharmaceutical preparation. The invention also relates to type B, C and D crystals of said compound.

    摘要翻译: 本发明涉及5 - [{6-(2-氟苄基)氧基-2-萘基}甲基] -2,4-噻唑烷二酮的A型晶体,其特征在于在11.5°±0.3°,14.5°具有特征吸收峰(2θ) °±0.2°,16.2°±0.3°,17.0°±0.3°,17.7°±0.2°,18.6°±0.3°,19.1°±0.2°,21.3°±0.4°,22.4°±0.5°,25.7°± 在粉末X射线衍射图中为1.5°和28.3°±10.5°,以及其制备方法,以及包含该方法的药物组合物。 该晶体的稳定性优异,在处理,储存和制药方面具有优势。 本发明还涉及所述化合物的B,C和D型晶体。

    Salt or Solvate of 5-Methyl-2(Piperazin-1-Yl)Benzenesulfonic Acid
    3.
    发明申请
    Salt or Solvate of 5-Methyl-2(Piperazin-1-Yl)Benzenesulfonic Acid 审中-公开
    盐酸盐或5-甲基-2(哌嗪-1-基)苯磺酸的溶剂合物

    公开(公告)号:US20100004266A1

    公开(公告)日:2010-01-07

    申请号:US12309487

    申请日:2007-07-20

    申请人: Katsuhiko Masuda

    发明人: Katsuhiko Masuda

    CPC分类号: C07D295/08

    摘要: The present invention provides a novel salt form or solvate of 5-methyl-2-(piperazin-1-yl)benzenesulfonic acid.The present invention provides 5-methyl-2-(piperazin-1-yl)benzenesulfonic acid hydrochloride, calcium 5-methyl-2-(piperazin-1-yl)benzenesulfonate and 5-methyl-2-(piperazin-1-yl)benzenesulfonic acid 2,2,2-tetrafluoroethanolate.

    摘要翻译: 本发明提供5-甲基-2-(哌嗪-1-基)苯磺酸的新型盐形式或溶剂合物。 本发明提供5-甲基-2-(哌嗪-1-基)苯磺酸盐酸盐,5-甲基-2-(哌嗪-1-基)苯磺酸钙和5-甲基-2-(哌嗪-1-基) 苯磺酸2,2,2-四氟乙醇盐。

    Flying spherical body measuring apparatus
    4.
    发明授权
    Flying spherical body measuring apparatus 失效
    飞球体测量仪

    公开(公告)号:US5481355A

    公开(公告)日:1996-01-02

    申请号:US102345

    申请日:1993-08-05

    摘要: The initial movement of a spherical body is detected by detecting the intersection with a light beam emitted from trigger light illuminating portion 2 to trigger light-receiving portion 3, and as a result, measurement of time by an arithmetic processing unit is started. During flight, spherical body 1 intersects light beams emitted from surface velocity sensors 4 and 5, the reflected light therein is detected by these surface velocity sensors 4 and 5, and the surface velocity of spherical body 1 is then measured. Spherical body 1 continues in flight and intersects at least two light beams irradiated from multi-beam illuminating portion 6 which are detected by multi-beam light-receiving portion 7. Based on a signal from multi-beam light-receiving portion 7 the arithmetic processing unit measures the time of intersection of spherical body 1 with a light beam, and then calculates the angle of elevation, horizontal angle, velocity and surface velocity of spherical body 1 based on the aforementioned measured time period. Furthermore, this arithmetic processing unit also calculates the amount of directional rotation of spherical body 1 based on the aforementioned calculated angle of elevation, horizontal angle, velocity and surface velocity of spherical body 1.

    摘要翻译: 通过检测与从触发光照射部分2发射的光束的交点来触发光接收部分3来检测球体的初始移动,结果,开始由算术处理单元测量时间。 在飞行中,球体1与表面速度传感器4和5发射的光束相交,其中的反射光被这些表面速度传感器4和5检测,然后测量球体1的表面速度。 球形体1在飞行中继续,并与由多光束照射部分6照射的至少两个光束相交,由多光束光接收部分7检测。根据来自多光束光接收部分7的信号,算术处理 单位测量球体1与光束的交叉时间,然后根据上述测量时间周期计算球体1的仰角,水平角,速度和表面速度。 此外,该算术处理单元还基于上述计算的球体1的仰角,水平角,速度和表面速度来计算球体1的定向旋转量。

    Metal ion laser protected against the deposition of metal vapor on
brewster windows
    5.
    发明授权
    Metal ion laser protected against the deposition of metal vapor on brewster windows 失效
    金属离子激光器防止金属蒸气沉积在布鲁斯特窗口上

    公开(公告)号:US4710938A

    公开(公告)日:1987-12-01

    申请号:US873155

    申请日:1986-06-06

    IPC分类号: H01S3/03 H01S3/034 H01S3/22

    CPC分类号: H01S3/0346 H01S3/031

    摘要: A helium-cadmium ion laser is disclosed which has a tubular housing hermetically closed at both ends by Brewster windows and having a hollow cathode mounted therein. Disposed outside the hollow cathode and open to its interior are a row of primary anodes and a row of metal chambers containing a metal material to be vaporized. A pair of secondary anodes are further disposed adjacent the opposite ends of the hollow cathode for protecting the Brewster windows from contamination by the metal vapor by sending it back into the hollow cathode. In order to prevent the metal vapor from depositing on the ends of the hollow cathode on being thus sent back, a pair of tubular insulators are coaxially mounted next to the opposite ends of the hollow cathode for the passage of the metal vapor therethrough. Each tubular insulator has a bore including a smaller diameter portion away from the hollow cathode, and a larger diameter portion closer to the hollow cathode. Further, for impeding the flow of the metal vapor from the hollow cathode toward the Brewster windows, the laser housing has a pair of constrictions adjacent the Brewster windows.

    摘要翻译: 公开了一种氦 - 镉离子激光器,其具有通过布鲁斯特窗口在两端密封并具有安装在其中的中空阴极的管状外壳。 设置在空心阴极外面并向其内部开放的是一排主阳极和一排含有要蒸发的金属材料的金属室。 一对次级阳极进一步设置在中空阴极的相对端附近,用于通过将布鲁斯特窗口送回中空阴极来保护布鲁斯特窗口免受金属蒸气的污染。 为了防止金属蒸气沉积在中空阴极的端部上,因此这样一个管状的绝缘体被同轴地安装在中空阴极的相对端上,以使金属蒸汽通过。 每个管状绝缘体具有包括远离空心阴极的较小直径部分的孔和更接近空心阴极的较大直径部分。 此外,为了阻止金属蒸气从中空阴极朝向布鲁斯特窗口流动,激光器壳体具有与布鲁斯特窗口相邻的一对收缩部。

    IMAGE INFORMATION DETECTING APPARATUS
    6.
    发明申请
    IMAGE INFORMATION DETECTING APPARATUS 失效
    图像信息检测装置

    公开(公告)号:US20070256088A1

    公开(公告)日:2007-11-01

    申请号:US11668984

    申请日:2007-01-30

    IPC分类号: G11B17/04

    CPC分类号: G11B7/0037

    摘要: An image information detecting apparatus is disclosed that comprises: a semiconductor laser that emits a laser light beam; a light receiving unit that receives a reflected light beam of the laser light beam applied to a color changing layer of an optical disc, the color changing layer being formed from a photo-sensitive material of a heat-sensitive material, and that outputs an electrical signal corresponding to the level of the reflected light beam; and a detecting unit that detects image information based on the electric signal, wherein the image information detecting apparatus detects the image information indicating an image from the color changing layer after the image has been formed therein.

    摘要翻译: 公开了一种图像信息检测装置,包括:发射激光的半导体激光器; 光接收单元,其接收施加到光盘的变色层的激光束的反射光束,所述变色层由感光材料的感光材料形成,并且输出电 信号对应于反射光束的电平; 以及检测单元,其基于所述电信号检测图像信息,其中所述图像信息检测装置在形成所述图像之后检测指示来自所述变色层的图像的图像信息。

    Drive mode selecting system for four-wheel-drive motor vehicle
    7.
    发明授权
    Drive mode selecting system for four-wheel-drive motor vehicle 失效
    四轮驱动汽车的驱动模式选择系统

    公开(公告)号:US4890686A

    公开(公告)日:1990-01-02

    申请号:US247191

    申请日:1988-09-21

    摘要: A drive mode selecting system for a four-wheel-drive motor vehicle includes a drive system for driving a first axle drive mechanism and a second axle drive mechanism, a clutch for selectively rigidly connecting the first and second axle drive mechanisms through the drive system for transmitting relative torque between the first and second axle drive mechanisms, and disconnecting the first and second axle drive mechanisms, a brake operation detector for detecting operation of a brake of the motor vehicle, an accelerator operation detector for detecting operation of an accelerator of the motor vehicle, and a controller responsive to detected signals from the brake operation detecting means and the accelerator operation detecting means for applying a disengaging signal to the clutch means to disconnect the first and second axle drive mechanisms when the detected signals indicate that the brake is operated and the accelerator is not operated.

    摘要翻译: 用于四轮驱动的机动车辆的驱动模式选择系统包括用于驱动第一车轴驱动机构和第二车轴驱动机构的驱动系统,用于通过驱动系统选择性地刚性地连接第一和第二轴驱动机构的离合器, 在所述第一和第二轴驱动机构之间传递相对扭矩,以及断开所述第一和第二轴驱动机构,用于检测所述机动车辆的制动器的操作的制动操作检测器,用于检测所述电动机的加速器的操作的加速器操作检测器 车辆以及响应于来自制动操作检测装置和加速器操作检测装置的检测信号的控制器,用于当检测到的信号指示制动器被操作时,向离合器装置施加分离信号以断开第一和第二轴驱动机构, 加速器不工作。

    Drive power transmission device
    9.
    发明授权
    Drive power transmission device 失效
    驱动传动装置

    公开(公告)号:US4756209A

    公开(公告)日:1988-07-12

    申请号:US68568

    申请日:1987-06-30

    摘要: A drive power transmission device includes an input carrier having a front portion for receiving drive power from a drive source and a tubular rear portion, a planetary gear mechanism having a sun gear disposed coaxially in the tubular portion of the input carrier, a plurality of planet gears meshing with the sun gear and rotatably supported on a periphery of the tubular portion, and a ring gear mounted concentrically on the tubular portion and meshing with the planet gears, a first output shaft coupled to and supporting the sun gear, an intermediate tubular member connectable to the first output shaft and a rear end of the tubular rear portion of the input carrier and disposed concentrically with the first output shaft, an outer tubular member connectable to the ring gear and disposed concentrically with the intermediate tubular member, a viscous shear coupling mechanism interconnecting the outer tubular member and the intermediate tubular member, and a second output shaft coupled to and supporting the outer tubular member. The viscous shear coupling mechanism comprises two groups of mutually interleaves plates disposed in a fluid chamber defined between the intermediate tubular member and the outer tubular member and filled with a fluid and fixedly fitted over the intermediate tubular member and in the outer tubular member.

    摘要翻译: 一种驱动动力传递装置,包括:输入托架,具有用于从驱动源和管状后部接收驱动力的前部;行星齿轮机构,其具有同轴地布置在输入托架的管状部分中的太阳轮;多个行星 与太阳齿轮啮合的齿轮和可旋转地支撑在管状部分的周边上的齿轮,以及同心地安装在管状部分上并与行星齿轮啮合的环形齿轮,联接到太阳齿轮并支撑太阳齿轮的第一输出轴,中间管状部件 可连接到第一输出轴和输入托架的管状后部的后端并且与第一输出轴同心设置,外部管状构件,其可连接到环形齿轮并与中间管状构件同心设置,粘性剪切耦合 将外部管状构件和中间管状构件互连的机构,以及联接到该第二输出轴的第二输出轴 并支撑外管状构件。 粘性剪切耦合机构包括两组相互交错的板,它们设置在限定在中间管状构件和外部管状构件之间的流体室中,并填充有流体并固定地装配在中间管状构件和外部管状构件上。

    Image information detecting apparatus
    10.
    发明授权
    Image information detecting apparatus 失效
    图像信息检测装置

    公开(公告)号:US07791995B2

    公开(公告)日:2010-09-07

    申请号:US11668984

    申请日:2007-01-30

    IPC分类号: G11B7/00

    CPC分类号: G11B7/0037

    摘要: An image information detecting apparatus is disclosed that comprises: a semiconductor laser that emits a laser light beam; a light receiving unit that receives a reflected light beam of the laser light beam applied to a color changing layer of an optical disc, the color changing layer being formed from a photo-sensitive material of a heat-sensitive material, and that outputs an electrical signal corresponding to the level of the reflected light beam; and a detecting unit that detects image information based on the electric signal, wherein the image information detecting apparatus detects the image information indicating an image from the color changing layer after the image has been formed therein.

    摘要翻译: 公开了一种图像信息检测装置,包括:发射激光的半导体激光器; 光接收单元,其接收施加到光盘的变色层的激光束的反射光束,所述变色层由感光材料的感光材料形成,并且输出电 信号对应于反射光束的电平; 以及检测单元,其基于所述电信号检测图像信息,其中所述图像信息检测装置在形成所述图像之后检测指示来自所述变色层的图像的图像信息。