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1.发明授权公开(公告)号：US08273781B2
公开(公告)日：2012-09-25
申请号：US13255345
申请日：2010-03-08
申请人： Tatsumi Suzuki , Tadashi Sugiura , Yoshikazu Ito
发明人： Tatsumi Suzuki , Tadashi Sugiura , Yoshikazu Ito
IPC分类号： A61K31/41 , C07D257/04
CPC分类号： C07D257/04
摘要： The present invention provides a process for preparation of 1-alkyl-5-benzoyl-1H-tetrazole derivative including a step 1 of reacting a ketoamide derivative represented by formula (I) (in formula (I), A represents a halogen atom or the like; n represents an integer of 0 to 5; Y represents an alkyl group) with a halogenating agent to obtain an imidoyl halide derivative represented by formula (II) (in formula (II), A, n and Y are as defined above; X represents a halogen atom); and a step 2 of reacting the imidoyl halide derivative represented by formula (II) with an azide represented by formula (III) (in formula (III), M represents an alkali metal or the like; m represents 1 or 2) to obtain a 1-alkyl-5-benzoyl-1H-tetrazole derivative represented by formula (IV) (in formula (IV), A, n and Y are as defined above).
摘要翻译： 本发明提供一种制备1-烷基-5-苯甲酰基-1H-四唑衍生物的方法，其包括使式（I）表示的酮酰胺衍生物（式（I）中的A表示卤素原子或 （II）表示的亚氨基卤化物衍生物（式（II）中，A，n和Y如上所定义），卤素化合物与式（II）表示的亚氨基卤化物衍生物相同，式中，n表示0〜5的整数，Y表示烷基，Y表示烷基） X表示卤素原子）; 和式（II）表示的亚氨基卤衍生物与式（III）表示的叠氮化物（式（III）中的M表示碱金属等，m表示1或2）反应，得到 由式（IV）表示的1-烷基-5-苯甲酰基-1H-四唑衍生物（式（IV）中，A，n和Y如上所定义）。
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2.发明申请公开(公告)号：US20120004420A1
公开(公告)日：2012-01-05
申请号：US13255345
申请日：2010-03-08
申请人： Tatsumi Suzumi , Tadashi Sugiura , Yoshikazu Ito
发明人： Tatsumi Suzumi , Tadashi Sugiura , Yoshikazu Ito
IPC分类号： C07D257/04
CPC分类号： C07D257/04
摘要： The present invention provides a process for preparation of 1-alkyl-5-benzoyl-1H-tetrazole derivative including a step 1 of reacting a ketoamide derivative represented by formula (I) (in formula (I), A represents a halogen atom or the like; n represents an integer of 0 to 5; Y represents an alkyl group) with a halogenating agent to obtain an imidoyl halide derivative represented by formula (II) (in formula (II), A, n and Y are as defined above; X represents a halogen atom); and a step 2 of reacting the imidoyl halide derivative represented by formula (II) with an azide represented by formula (III) (in formula (III), M represents an alkali metal or the like; m represents 1 or 2) to obtain a 1-alkyl-5-benzoyl-1H-tetrazole derivative represented by formula (IV) (in formula (IV), A, n and Y are as defined above).
摘要翻译： 本发明提供一种制备1-烷基-5-苯甲酰基-1H-四唑衍生物的方法，其包括使式（I）表示的酮酰胺衍生物（式（I）中的A表示卤素原子或 （II）表示的亚氨基卤化物衍生物（式（II）中，A，n和Y如上所定义），卤素化合物与式（II）表示的亚氨基卤化物衍生物相同，式中，n表示0〜5的整数，Y表示烷基，Y表示烷基） X表示卤素原子）; 和式（II）表示的亚氨基卤衍生物与式（III）表示的叠氮化物（式（III）中的M表示碱金属等，m表示1或2）反应，得到 由式（IV）表示的1-烷基-5-苯甲酰基-1H-四唑衍生物（式（IV）中，A，n和Y如上所定义）。
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公开(公告)号：US20090171540A1
公开(公告)日：2009-07-02
申请号：US12314819
申请日：2008-12-17
CPC分类号： F16H61/21 , F16H59/44 , F16H61/0213 , F16H61/0248 , F16H2059/183
摘要： A control device for an automatic transmission capable of operating in an automatic shift mode in which a gear ratio is automatically selected based on driving conditions of a vehicle, and also capable of operating in a manual shift mode in which the gear ratio is changed based on an upshift command or a downshift command by manual operation of a manual operation device, the control device includes a manual shift control unit that changes and sets the gear ratio after downshift depending on a degree of requirement for deceleration based on a driving operation when the downshift command has been operated by the manual operation device in the manual shift mode, and performs the downshift to the gear ratio that has been changed and set.
摘要翻译： 一种用于自动变速器的控制装置，其能够在自动变速模式下操作，其中根据车辆的驾驶状况自动选择齿轮比，并且还能够以基于以下方式改变齿轮比的手动变速模式进行操作 通过手动操作装置的升档命令或降档命令，所述控制装置包括手动变速控制单元，所述手动变速控制单元根据所述降档时的驱动操作根据减速度的要求来改变和设定所述换低档后的档位比 指令由手动操作装置在手动换档模式下操作，并且执行降档到变速比设定。
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公开(公告)号：US08116952B2
公开(公告)日：2012-02-14
申请号：US12314822
申请日：2008-12-17
CPC分类号： F16H61/0213 , F16H61/0248 , Y10T477/69367
摘要： A control system for an automatic transmission is provided with a manual shift mode capable of performing a shift command made by manual operation. While in the manual shift mode and during the operation of a downshift command generated by a shift lever, a manual shift control unit calculates a degree of power required by a driver that, for example, takes into consideration an operation intent of the driver and a road condition. A post-downshift shift speed is then determined in accordance with the degree of required power and downshifting performed. By performing only one downshift command through manual operation, downshifting in accordance with the degree of power required by the driver is performed. Downshifting to a shift speed desired by the driver can thus be promptly performed, without the operation becoming a burden.
摘要翻译： 用于自动变速器的控制系统具有能够执行通过手动操作进行的换档指令的手动换挡模式。 在手动换挡模式下，在换挡杆产生的降挡指令的操作期间，手动变速控制单元计算驾驶员要求的功率，例如考虑驾驶员的操作意图和 道路状况。 然后根据所需功率和降档的程度来确定降档换档速度。 通过手动操作仅执行一个降档指令，执行根据驾驶员所需功率的降档。 因此可以迅速地执行降档到驾驶员期望的换档速度，而不会使操作变成负担。
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公开(公告)号：US08068963B2
公开(公告)日：2011-11-29
申请号：US12318226
申请日：2008-12-23
IPC分类号： B60W10/10
CPC分类号： F16H61/0213 , F16H59/66 , F16H61/0248 , F16H2059/663 , Y10T477/69367
摘要： A control device for an automatic transmission capable of operating in an automatic shift mode in which a gear ratio is automatically selected based on driving conditions of a vehicle, and also capable of operating in a manual shift mode in which the gear ratio is changed based on an upshift command or a downshift command by manual operation of a manual operation device, the control device includes a manual shift control unit that changes and sets the gear ratio after downshift depending on road conditions when the downshift command has been operated by the manual operation device in the manual shift mode, and performs the downshift to the gear ratio that has been changed and set.
摘要翻译： 一种用于自动变速器的控制装置，其能够在自动变速模式下操作，其中根据车辆的驾驶状况自动选择齿轮比，并且还能够以基于以下方式改变齿轮比的手动变速模式进行操作 通过手动操作装置的手动操作的升档指令或降档指令，所述控制装置包括手动变速控制单元，所述手动变速控制单元根据所述手动操作装置操作了所述降档指令时的道路状况来改变并设定所述换档后的档位比 在手动换档模式下，执行降档到变速比设定。
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公开(公告)号：US06915970B2
公开(公告)日：2005-07-12
申请号：US10300750
申请日：2002-11-21
申请人： Yoshiji Iyoda , Akito Suzuki , Tadashi Sugiura
发明人： Yoshiji Iyoda , Akito Suzuki , Tadashi Sugiura
CPC分类号： B22C5/0404 , B02C17/14 , B02C17/16 , B22C5/0481 , B22D29/02 , Y10S241/10
摘要： An apparatus for vibratingly smashing sand masses, comprising a sand tank (30) elastically supported and having an inner tank (33) therein for holding sand masses; and vibrating means (21) having unbalanced weights for vibrating the sand tank, including the inner tank, by rotating the unbalanced weights, such that the vibrations of the sand tank draw a Lissajous's figure of approximately a circle. The inner tank (33) is defined by a wall (31) disposed in the sand tank apart from the inner surface (30A) of the sand tank (30), the wall (31) having a plurality of apertures (32).
摘要翻译： 一种用于振动粉碎沙粒的装置，包括：弹性支撑的砂箱（30），其中具有用于保持砂块的内罐（33）; 以及具有不平衡重物的振动装置（21），用于通过旋转不平衡的重物来振动包括内罐的砂箱，使得砂箱的振动吸收大约一圈的李萨如图。 内罐（33）由设置在沙箱中的与砂箱（30）的内表面（30A）分开的壁（31）限定，壁（31）具有多个孔（32）。
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公开(公告)号：US4648163A
公开(公告)日：1987-03-10
申请号：US766696
申请日：1985-08-19
CPC分类号： F16H55/49 , B21D53/261 , B21H1/04 , B23P15/00 , Y10T29/49456
摘要： A method of making a poly-V ribbed pulley engaged with a V-ribbed belt or V-ribbed belts. The method includes the steps of pressing two flanges or one circular projection between the two flanges in the cylinder, pressing a flange at the radially outer end of a thick circular plate, connecting one flange of the cylinder to the flange of the thick circular plate by welding, and performing rolling to form V-shaped grooves at the outside surface of the cylinder.
摘要翻译： 制造与V形肋带或V形肋带接合的多V肋带轮的方法。 该方法包括以下步骤：在气缸中的两个凸缘之间按压两个凸缘或一个圆形突起，在厚圆形板的径向外端处按压凸缘，将圆柱体的一个凸缘连接到厚圆形板的凸缘上 焊接并进行轧制以在气缸的外表面形成V形槽。
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8.发明授权Compound containing pyridine ring and method for producing halogenated picoline derivative and tetrazolyloxime derivative 有权含有吡啶环的化合物及卤代甲基吡啶衍生物和四唑基肟衍生物的制备方法公开(公告)号：US08841458B2
公开(公告)日：2014-09-23
申请号：US13583733
申请日：2011-03-11
申请人： Hidekazu Miyazaki , Satoru Yanaka , Shiro Tsubokura , Tadashi Sugiura , Kaoru Noda , Kengo Suzuki
发明人： Hidekazu Miyazaki , Satoru Yanaka , Shiro Tsubokura , Tadashi Sugiura , Kaoru Noda , Kengo Suzuki
IPC分类号： C07D213/75 , C07D401/12 , C07D405/12
CPC分类号： C07D213/75 , C07D401/12 , C07D405/12
摘要： Disclosed is a compound containing a pyridine ring that can be synthesized in an industrially advantageous manner, and is useful as an intermediate for producing tetrazolyloxime derivatives that exhibit fungicidal activity (wherein R0 represents a C1-6 alkoxy group, C1-6 alkoxy-C1-6 alkoxy group or the like, R1 represents a C1-2 alkoxycarbonyl group, acetyl group or the like, Z represents a halogen atom, cyano group or the like, X represents a halogen atom, and n represents an integer of 0 to 3), and industrially advantageous production methods for producing 2-substituted amino-6-halomethylpyridine derivatives and tetrazolyloxime derivatives.
摘要翻译： 公开了含有可以工业上有利的方式合成的吡啶环的化合物，可用作生产具有杀真菌活性的四唑基肟衍生物的中间体（其中R 0表示C1-6烷氧基，C1-6烷氧基C1- 6烷氧基等，R 1表示C 1-2烷氧基羰基，乙酰基等，Z表示卤素原子，氰基等，X表示卤素原子，n表示0〜3的整数） 以及用于生产2-取代的氨基-6-卤甲基吡啶衍生物和四唑基肟衍生物的工业上有利的制备方法。
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公开(公告)号：US20090171539A1
公开(公告)日：2009-07-02
申请号：US12314818
申请日：2008-12-17
CPC分类号： F16H61/0213 , F16H59/66 , F16H2059/0252 , F16H2059/183
摘要： A control apparatus for an automatic transmission capable of operating in an automatic shift mode in which a speed ratio is automatically selected based on driving conditions of a vehicle, and a manual shift mode in which the speed ratio is changed based on an upshift command and a downshift command by manual operation of a manual operation unit, the control apparatus includes a controller that operates in a jumping shift mode that is included in the manual shift mode and that is composed of a smaller number of shift speeds than a number of shift speeds of the automatic shift mode; wherein the controller performs a downshift from a shift speed of the jumping shift mode at a time when the downshift command is issued by an operation of the manual operation unit based on the shift speed of the jumping shift mode.
摘要翻译： 一种自动变速器的控制装置，能够根据车辆的行驶状况自动选择速比的自动变速模式进行动作，根据升挡指令和 通过手动操作单元的手动操作来进行降档命令，控制装置包括控制器，该控制器以包括在手动换档模式中的跳跃换档模式操作，并且该换档模式由少于多个换档速度 自动换档模式; 其中，所述控制器根据所述跳跃换档模式的换档速度，通过所述手动操作单元的操作发出所述降档指令时，从所述跳跃换档模式的换档速度进行降档。
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10.发明授权2, 3-dihalogeno-6-trifluoromethylbenzene derivatives and process for producing the same 有权2,3-二卤代-6-三氟甲苯衍生物及其制备方法
公开(公告)号：US6054605A
公开(公告)日：2000-04-25
申请号：US249076
申请日：1999-02-12
申请人： Isamu Kasahara , Tadashi Sugiura , Tsutomu Inoue
发明人： Isamu Kasahara , Tadashi Sugiura , Tsutomu Inoue
IPC分类号： C07C45/44 , C07C47/55 , C07C63/70 , C07C69/76 , C07C233/65 , C07C251/48 , C07C255/50
CPC分类号： C07C255/50 , C07C233/65 , C07C251/48 , C07C45/44 , C07C47/55 , C07C63/70 , C07C69/76
摘要： The present invention is to provide 2,3-dihalogeno-6-trifluoromethylbenzene derivatives represented by a general formula [I]; ##STR1## wherein X.sub.1 and X.sub.2 are the same or different and each independently represents fluoro or chloro; Y represents COOH, CONH.sub.2, CN, CHO, CH.dbd.NOH or COOR', wherein R' is C.sub.1 -C.sub.4 alkyl, except the case that X.sub.1 and X.sub.2 are each chloro and Y is COOH, which are useful as the starting materials for producing pesticides, drugs and the like, and a process for producing such derivatives.
摘要翻译： 本发明提供由通式[I]表示的2,3-二卤代-6-三氟甲基苯衍生物。 其中X1和X2相同或不同并且各自独立地表示氟或氯; Y表示COOH，CONH 2，CN，CHO，CH = NOH或COOR'，其中R'为C 1 -C 4烷基，除了X1和X2各自为氯，Y为COOH，可用作生产原料 杀虫剂，药物等，以及这些衍生物的制造方法。
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