Fungicidal pyrazoles
    6.
    发明授权
    Fungicidal pyrazoles 有权
    杀真菌吡唑

    公开(公告)号:US09062005B2

    公开(公告)日:2015-06-23

    申请号:US13254205

    申请日:2010-03-03

    摘要: Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein Q1 is a phenyl ring, naphthalenyl ring system, a 5- to 6-membered fully unsaturated heterocyclic ring or an 8- to 10-membered heteroaromatic bicyclic ring system, each as described with optional substituents as defined in the disclosure; Q2 is a phenyl ring, a naphthalenyl ring system, a 5- to 6-membered saturated, partially unsaturated or fully unsaturated heterocyclic ring, or an 8- to 10-membered heteroaromatic bicyclic ring system, each as described with optional substituents as defined in the disclosure; X is O, S(O)m, NR4, CR15R16, C(═O) or C(═S); and R1, R1a, R2, R4, R15, R16 and m are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention. Also disclosed are compounds of Formula 2, including all geometric and stereoisomers, and salts thereof, wherein X is NH; and Q1, Q2 and R2 are as defined for Formula 1; which are useful as intermediates for preparing compounds of Formula 1.

    摘要翻译: 公开了式1的化合物,包括所有几何和立体异构体,N-氧化物及其盐,其中Q1是苯环,萘环体系,5-至6-元完全不饱和杂环或8-至10- 每个如本公开中所定义的任选的取代基所述; Q2是苯环,萘环体系,5至6元饱和,部分不饱和或完全不饱和的杂环或8至10元杂芳族双环系统,每个如在如 披露; X是O,S(O)m,NR 4,CR 15 R 16,C(= O)或C(= S))。 并且R1,R1a,R2,R4,R15,R16和m如本公开所定义。 还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法,包括施用有效量的本发明化合物或组合物。 还公开了式2的化合物,包括所有几何和立体异构体及其盐,其中X是NH; 且Q1,Q2和R2如式1所定义; 其可用作制备式1化合物的中间体。

    FUNGICIDAL PYRAZOLES
    7.
    发明申请
    FUNGICIDAL PYRAZOLES 有权
    真菌PYRAZOLES

    公开(公告)号:US20110319430A1

    公开(公告)日:2011-12-29

    申请号:US13254205

    申请日:2010-03-03

    摘要: Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein Q1 is a phenyl ring, naphthalenyl ring system, a 5- to 6-membered fully unsaturated heterocyclic ring or an 8- to 10-membered heteroaromatic bicyclic ring system, each as described with optional substituents as defined in the disclosure; Q2 is a phenyl ring, a naphthalenyl ring system, a 5- to 6-membered saturated, partially unsaturated or fully unsaturated heterocyclic ring, or an 8- to 10-membered heteroaromatic bicyclic ring system, each as described with optional substituents as defined in the disclosure; X is O, S(O)m, NR4, CR15R16, C(═O) or C(═S); and R1, R1a, R2, R4, R15, R16 and m are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention. Also disclosed are compounds of Formula 2, including all geometric and stereoisomers, and salts thereof, wherein X is NH; and Q1, Q2 and R2 are as defined for Formula 1; which are useful as intermediates for preparing compounds of Formula 1.

    摘要翻译: 公开了式1的化合物,包括所有几何和立体异构体,N-氧化物及其盐,其中Q1是苯环,萘环体系,5-至6-元完全不饱和杂环或8-至10- 每个如本公开中所定义的任选的取代基所述; Q2是苯环,萘环体系,5至6元饱和,部分不饱和或完全不饱和的杂环或8至10元杂芳族双环系统,每个如在如 披露; X是O,S(O)m,NR 4,CR 15 R 16,C(= O)或C(= S))。 并且R1,R1a,R2,R4,R15,R16和m如本公开所定义。 还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法,包括施用有效量的本发明化合物或组合物。 还公开了式2的化合物,包括所有几何和立体异构体及其盐,其中X是NH; 且Q1,Q2和R2如式1所定义; 其可用作制备式1化合物的中间体。

    Fungicidal pyrazoles
    9.
    发明授权
    Fungicidal pyrazoles 有权
    杀真菌吡唑

    公开(公告)号:US08754115B2

    公开(公告)日:2014-06-17

    申请号:US13816847

    申请日:2011-08-31

    IPC分类号: A61K31/415 C07D231/10

    摘要: Disclosed are compounds of Formula 1 and Formula 1A including all stereoisomers, N-oxides, and salts thereof, wherein Q1, Q2, R1, R2, R4, R5 and X are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 or Formula 1A and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.

    摘要翻译: 公开了式1和式1A的化合物,其包括所有立体异构体,N-氧化物及其盐,其中Q1,Q2,R1,R2,R4,R5和X如本公开所定义。 还公开了含有式1或式1A化合物的组合物和用于控制由真菌病原体引起的植物病害的方法,包括施用有效量的本发明化合物或组合物。