Process for the preparation of 1,3-dialkanoyl hexahydropyrimidine
    2.
    发明授权
    Process for the preparation of 1,3-dialkanoyl hexahydropyrimidine 失效
    1,3-二烷酰基六氢嘧啶的制备方法

    公开(公告)号:US3872120A

    公开(公告)日:1975-03-18

    申请号:US44842674

    申请日:1974-03-04

    申请人: US AGRICULTURE

    CPC分类号: C07D239/04 C07D233/02

    摘要: 1,3-Diacyl imidazolidines and hexahydropyrimidines were prepared by the reaction of formaldehyde and an N,N''-alkylenebisamide in the presence of a strong acid catalyst, the substituent acyl groups being acetyl, butyryl, pentanoyl, hexanoyl, heptanoyl, octanoyl, nonanoyl, decanoyl, palmitoyl, stearoyl, and oleoyl. These compounds exhibit antimycotic activity.

    摘要翻译: 1,3-二酰基咪唑烷和六氢嘧啶通过在强酸催化剂存在下甲醛与N,N'-亚烷基二甲酰胺的反应制备,取代基酰基为乙酰基,丁酰基,戊酰基,己酰基,庚酰基,辛酰基,壬酰基 癸酰基,棕榈酰基,硬脂酰基和油酰基。 这些化合物显示出抗真菌活性。

    1,3-Diacyl derivatives of imidazolidine
    3.
    发明授权
    1,3-Diacyl derivatives of imidazolidine 失效
    咪唑烷的1,3-二酰基衍生物

    公开(公告)号:US3917638A

    公开(公告)日:1975-11-04

    申请号:US44842774

    申请日:1974-03-04

    申请人: US AGRICULTURE

    IPC分类号: C07D233/02 C07D49/34

    CPC分类号: C07D233/02

    摘要: 1,3-Diacyl imidazolidines and hexahydropyrimidines were prepared by the reaction of formaldehyde and an N,N''-alkylenebisamide in the presence of a strong acid catalyst, the substituent acyl groups being acetyl, butyryl, pentanoyl, hexanoyl, heptanoyl, octanoyl, nonanoyl, decanoyl, palmitoyl, stearoyl, and oleoyl. These compounds exhibit antimycotic activity.

    摘要翻译: 1,3-二酰基咪唑烷和六氢嘧啶通过在强酸催化剂存在下甲醛与N,N'-亚烷基二甲酰胺的反应制备,取代基酰基为乙酰基,丁酰基,戊酰基,己酰基,庚酰基,辛酰基,壬酰基 癸酰基,棕榈酰基,硬脂酰基和油酰基。 这些化合物显示出抗真菌活性。

    Phosphonated N,N-disubstituted fatty amides as bactericidal and fungicidal agents
    4.
    发明授权
    Phosphonated N,N-disubstituted fatty amides as bactericidal and fungicidal agents 失效
    磷酸化的N,N-二取代的脂肪酰胺作为杀菌剂和杀真菌剂

    公开(公告)号:US3911120A

    公开(公告)日:1975-10-07

    申请号:US33586073

    申请日:1973-02-26

    申请人: US AGRICULTURE

    IPC分类号: A01N57/18 C07F9/40 A01N9/36

    CPC分类号: A01N57/18 C07F9/4006

    摘要: Phosphonated N,N-disubstituted fatty amides were prepared by the free radical addition of dialkyl phosphites to terminal and nonterminal double bonds of N,N-disubstituted amides. The free radical additions of the dialkyl phosphites to the unsaturated amides were initiated by irradiation with gamma radiation from cobalt-60. These new compounds exhibit antimicrobial activity.

    摘要翻译: 通过将亚磷酸二烷基酯自由基加成到N,N-二取代酰胺的末端和非末端双键来制备膦酸化的N,N-二取代的脂肪酰胺。 亚磷酸二烷基酯向不饱和酰胺的自由基添加通过用来自钴-60的γ辐射照射来引发。 这些新化合物表现出抗菌活性。