1,3-Diacyl derivatives of imidazolidine
    3.
    发明授权
    1,3-Diacyl derivatives of imidazolidine 失效
    咪唑烷的1,3-二酰基衍生物

    公开(公告)号:US3917638A

    公开(公告)日:1975-11-04

    申请号:US44842774

    申请日:1974-03-04

    申请人: US AGRICULTURE

    IPC分类号: C07D233/02 C07D49/34

    CPC分类号: C07D233/02

    摘要: 1,3-Diacyl imidazolidines and hexahydropyrimidines were prepared by the reaction of formaldehyde and an N,N''-alkylenebisamide in the presence of a strong acid catalyst, the substituent acyl groups being acetyl, butyryl, pentanoyl, hexanoyl, heptanoyl, octanoyl, nonanoyl, decanoyl, palmitoyl, stearoyl, and oleoyl. These compounds exhibit antimycotic activity.

    摘要翻译: 1,3-二酰基咪唑烷和六氢嘧啶通过在强酸催化剂存在下甲醛与N,N'-亚烷基二甲酰胺的反应制备,取代基酰基为乙酰基,丁酰基,戊酰基,己酰基,庚酰基,辛酰基,壬酰基 癸酰基,棕榈酰基,硬脂酰基和油酰基。 这些化合物显示出抗真菌活性。

    Phosphonated N,N-disubstituted fatty amides as bactericidal and fungicidal agents
    4.
    发明授权
    Phosphonated N,N-disubstituted fatty amides as bactericidal and fungicidal agents 失效
    磷酸化的N,N-二取代的脂肪酰胺作为杀菌剂和杀真菌剂

    公开(公告)号:US3911120A

    公开(公告)日:1975-10-07

    申请号:US33586073

    申请日:1973-02-26

    申请人: US AGRICULTURE

    IPC分类号: A01N57/18 C07F9/40 A01N9/36

    CPC分类号: A01N57/18 C07F9/4006

    摘要: Phosphonated N,N-disubstituted fatty amides were prepared by the free radical addition of dialkyl phosphites to terminal and nonterminal double bonds of N,N-disubstituted amides. The free radical additions of the dialkyl phosphites to the unsaturated amides were initiated by irradiation with gamma radiation from cobalt-60. These new compounds exhibit antimicrobial activity.

    摘要翻译: 通过将亚磷酸二烷基酯自由基加成到N,N-二取代酰胺的末端和非末端双键来制备膦酸化的N,N-二取代的脂肪酰胺。 亚磷酸二烷基酯向不饱和酰胺的自由基添加通过用来自钴-60的γ辐射照射来引发。 这些新化合物表现出抗菌活性。

    Quaternary ammonium salts of n-substituted palmitamides
    8.
    发明授权
    Quaternary ammonium salts of n-substituted palmitamides 失效
    N-取代的棕榈酰胺的季铵盐

    公开(公告)号:US3869483A

    公开(公告)日:1975-03-04

    申请号:US26586972

    申请日:1972-06-23

    申请人: US AGRICULTURE

    IPC分类号: C07D295/185 C07C103/30

    CPC分类号: C07D295/185

    摘要: A number of new quaternary ammonium salts of n-substituted palmitamides have been prepared by conventional methods. These derivatives have been characterized by exhibiting antimycotic activity and three of the derivatives, 4-palmitoyl-1,1dimethylpiperazinium iodide, (2palmitoylaminoethyl)trimethylammonium iodide, and 4-palmitoyl-1methyl-1-(1,4,5,6,7,7-hexachlorobicyclo(2.2.1)-hepta-2,5-diene -2methylene)piperazinium bromide have been further characterized by exhibiting nematocidal activity.

    摘要翻译: 已经通过常规方法制备了许多新的N-取代的棕榈酰胺季铵盐。 这些衍生物的特征在于显示出抗真菌活性,并且三种衍生物,4-棕榈酰基-1,1-二甲基哌嗪鎓碘化物,(2-棕榈酰氨基乙基)三甲基碘化铵和4-棕榈酰-1-甲基-1-(1,4, 5,6,7,7-六氯双环[2.2.1] - 庚-2,5-二烯-2-亚甲基)哌嗪鎓溴化物的进一步特征在于具有杀线虫活性。