公开(公告)号：US5532378A

公开(公告)日：1996-07-02

申请号：US356933

申请日：1994-12-15

申请人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen, hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, and R.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl,and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl , alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮，其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基的任选取代的基团， R 2代表氢，羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的系列中任意取代的基团，R 3表示任选被取代的基团， ，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US5405970A

公开(公告)日：1995-04-11

申请号：US31426

申请日：1993-03-15

申请人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen, hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, andR.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl,and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl, alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮，其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基，芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基 或R 2代表氢，羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的任选取代的基团，并且R 3代表包含烷基， 芳烷基，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US5057144A

公开(公告)日：1991-10-15

申请号：US556052

申请日：1990-07-20

申请人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04 ,  A01N43/653

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen, hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, andR.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl, and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl, alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮，其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基，芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基 或R 2代表氢，羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的任选取代的基团，并且R 3代表包含烷基， 芳烷基，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US5241074A

公开(公告)日：1993-08-31

申请号：US816365

申请日：1991-12-30

申请人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen, hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, andR.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl,and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl, alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮，其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基，芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基 或R 2代表氢，羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的任选取代的基团，并且R 3代表包含烷基， 芳烷基，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US5094683A

公开(公告)日：1992-03-10

申请号：US692439

申请日：1991-04-29

申请人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut Muller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, akinyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, andR.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl, and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl, alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基，芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基 R 2表示氢羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的任意取代的基团，并且R 3表示任选被取代的基团，该基团包括烷基， ，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US5625074A

公开(公告)日：1997-04-29

申请号：US632984

申请日：1996-04-16

申请人： Werner Daum ,  Klaus-Helmut M uller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Werner Daum ,  Klaus-Helmut M uller ,  Michael Schwamborn ,  Peter Babczinski ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

CPC分类号： C07D401/12 ,  A01N47/38 ,  A01N51/00 ,  C07D249/12 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D471/04 ,  C07D487/04

摘要： Herbicidal sulphonylaminocarbonyltriazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkylamino and dialkylamino,R.sup.2 represents hydrogen, hydroxyl, mercapto or amino, or represents an optionally substituted radical from the series comprising alkyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkylamino and dialkylamino, andR.sup.3 represents an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and heteroaryl,and salts thereof. Intermediates of the formula ##STR2## in which A.sup.1 represents in each case optionally substituted alkyl, alkenyl, cycloalkyl, alkoxy or dialkylamino andA.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, cycloalkyl, aralkyl, aryl or alkoxy,provided that both A.sup.1 and A.sup.2 do not simultaneously represent alkyl, are also new.

摘要翻译： 式（I）的除草磺酰基氨基羰基三唑啉酮，其中R 1表示氢，羟基或氨基，或代表包含烷基，烯基，炔基，环烷基，芳烷基，芳基，烷氧基，烯氧基，烷基氨基和二烷基氨基 或R 2代表氢，羟基，巯基或氨基，或代表包含烷基，环烷基，环烯基，芳烷基，芳基，烷氧基，烷基氨基和二烷基氨基的任选取代的基团，并且R 3代表包含烷基， 芳烷基，芳基和杂芳基，及其盐。 式（IIa）的中间体，其中A1表示在每种情况下为任选取代的烷基，烯基，环烷基，烷氧基或二烷基氨基，A 2表示氢，或在各种情况下表示任选取代的烷基，环烷基，芳烷基，芳基或烷氧基， 只要A1和A2不同时代表烷基，也是新的。

公开(公告)号：US4914123A

公开(公告)日：1990-04-03

申请号：US690930

申请日：1985-01-11

申请人： Werner Daum ,  Erich Klauke ,  Engelbert Kuhle ,  Wilhelm Brandes ,  Paul Reinecke

发明人： Werner Daum ,  Erich Klauke ,  Engelbert Kuhle ,  Wilhelm Brandes ,  Paul Reinecke

IPC分类号： A01N43/08 ,  A01N43/10 ,  A01N47/02 ,  A01N47/04 ,  C07D333/38 ,  C07F7/18

CPC分类号： C07D333/38 ,  A01N43/10 ,  A01N47/02 ,  A01N47/04

摘要： Acyloxythiophenes of the formula ##STR1## in which R.sup.1 represents alkyl, alkoxyalkyl, alkylthioalkyl, halogenoalkyl, cyanoalkyl, trialkylsilylmethyl, alkenyl or alkinyl,R.sup.2 represents alkyl,n represents 0 or 1 andR.sup.3 to R.sup.5 are identical or different and represent hydrogen, alkyl, alkoxy, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, halogenoalkylsulphinyl, halogenoalkylsulphonyl, N-halogenoalkyl-N-halogenoalkylthioamino, chlorine or fluorine andR.sup.6 and R.sup.7 represent hydrogen, fluorine, chlorine, nitro or trifluoromethyl, with the proviso that one of the radicals R.sup.3 to R.sup.7 is a fluorine-containing radical or at least 3 of the radicals R.sup.3 to R.sup.7 represent fluorine and/or chlorine,which possess fungicidal activity.

摘要翻译： 式中，R 1表示烷基，烷氧基烷基，烷硫基烷基，卤代烷基，氰基烷基，三烷基甲硅烷基甲基，烯基或炔基，R 2表示烷基，n表示0或1，R 3至R 5相同或不同，表示氢，烷基， 烷氧基，卤代烷基，卤代烷氧基，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基，N-卤代烷基-N-卤代烷硫基氨基，氯或氟，R6和R7表示氢，氟，氯，硝基或三氟甲基，条件是基团R3至R7中的一个为 含氟基团或至少3个基团R 3至R 7表示具有杀真菌活性的氟和/或氯。

公开(公告)号：US4960768A

公开(公告)日：1990-10-02

申请号：US348931

申请日：1989-05-08

申请人： Werner Daum ,  Gerd Hanssler

发明人： Werner Daum ,  Gerd Hanssler

IPC分类号： A01N43/08 ,  A01N43/10 ,  C07D333/38

CPC分类号： C07D333/38 ,  A01N43/10

摘要： Novel fungicidally active acyloxythiophene-carboxamides of the formula ##STR1## in which R.sup.1 represents alkyl, alkoxyalkyl, alkylthioalkyl, fluoroalkyl, cyanoalkyl, alkenyl, alkinyl or cycloalkyl,R.sup.2 represents alkyl or optionally substituted phenyl,R.sup.3 represents alkylsulphonyl, halogenoalkylsulphonyl, optionally substituted phenylsulphonyl or the --OC--Q radical, in whichQ represents alkyl which is optionally identically or differently substituted by halogen, alkoxy, alkylthio, alkylsulphonyl, alkylthioalkoxy, alkoxycarbonyl, phenyl, phenoxy or halogenophenoxy; alkenyl which is optionally identically or differently substituted by halogen, phenyl, halogenophenyl or halogenoalkylphenyl; alkinyl; cycloalkyl; alkoxy which is optionally substituted by halogen or cyano; phenyl which is optionally identically or differently substituted by halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, alkylsulphinyl, halogenoalkylsulphinyl, alkylsulphonyl or halogenoalkylsulphonyl; pyridyl; monoalkylamino, the alkyl part being optionally substituted by halogen, cyano, alkoxycarbonyl, dialkylaminocarbonyl, alkanyleneaminocarbonyl or oxaalkanyleneaminocarbonyl; 1-cyanocycloalkylamino; dialkylamino; alkanyleneamino; oxaalkanyleneamino; N-alkyl-N-phenylamino or phenylamino, in which the phenyl radical in each is optionally identically or differently substituted by halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, alkylsulphonyl, halogenoalkylsulphonyl, alkanylenedioxy, halogenoalkanylenedioxy or by --O--CHal.sub.2 --O--CHal.sub.2 --, orR.sup.4 represents alkyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, fluoroalkyl, alkenyl, alkinyl, cycloalkyl or alkoxy,R.sup.5 represents hydrogen, alkyl, alkoxyalkyl, alkylthioalkyl, fluoroalkyl, cyanoalkyl, alkenyl, alkinyl or cycloalkyl,R.sup.4 and R.sup.5, together with the adjacent nitrogen atom represent an optionally substituted heterocycle which can be substituted, in the alkylene chain, by further heteroatoms.

公开(公告)号：US4518605A

公开(公告)日：1985-05-21

申请号：US500732

申请日：1983-06-03

申请人： Wilhelm Brandes ,  Werner Daum

发明人： Wilhelm Brandes ,  Werner Daum

IPC分类号： A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00 ,  A01N43/64 ,  C07D233/61

CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： Fungicidally active novel azole-substituted oximino-cyano-acetamide derivatives of the formula ##STR1## in which R.sup.1 and R.sup.3 each independently is hydrogen or alkyl having up to 3 carbon atoms,R.sup.2 is hydrogen, alkyl having up to 6 carbon atoms, or halogenoalkyl having up to 2 carbon atoms and up to 5 halogen atoms,R.sup.4 is hydrogen or CO--NH--R.sup.5,R.sup.5 is hydrogen, cycloalkyl having 3 to 7 carbon carbon atoms, or alkyl having up to 8 carbon atoms and optionally substituted by cyano, hydrocarbonyl, aminocarbonyl, alkoxy and/or alkoxycarbonyl, each having up to 4 carbon atoms in the alkyl part,A is N or CH, andn is 0 or 1.

摘要翻译： 其中R1和R3各自独立地为氢或具有至多3个碳原子的烷基，R2为氢，具有至多6个碳原子的烷基或卤代烷基的杀真菌活性新型唑类取代的肟基 - 氰基 - 乙酰胺衍生物 具有至多2个碳原子和至多5个卤素原子，R 4是氢或CO-NH-R 5，R 5是氢，具有3至7个碳原子的环烷基或具有至多8个碳原子并且任选被氰基取代的烷基， 烷基部分中具有至多4个碳原子的烃基，氨基羰基，烷氧基和/或烷氧基羰基，A为N或CH，n为0或1。

公开(公告)号：US4863954A

公开(公告)日：1989-09-05

申请号：US194742

申请日：1988-05-17

申请人： Werner Daum ,  Gerd Hanssler

发明人： Werner Daum ,  Gerd Hanssler

IPC分类号： A01N43/08 ,  A01N43/10 ,  C07D333/38

CPC分类号： C07D333/38 ,  A01N43/10

摘要： Novel fungicidally active acyloxythiophene-carboxamides of the formula ##STR1## in which R.sup.1 represents alkyl, alkoxyalkyl, alkylthioalky, fluoroalkyl, cyanoalkyl, alkenyl, alkinyl or cycloalkyl,R.sup.2 represents alkyl or optionally substituted phenyl,R.sup.3 represents alkylsulphonyl, halogenoalkylsulphonyl, optionally substituted phenylsulphonyl or the --OC--Q radical, in whichQ represents alkyl which is optionally identically or differently substituted by halogen, alkoxy, alkylthio, alkylsulphonyl, alkylthioalkoxy, alkoxycarbonyl, phenyl, phenoxy or halogenophenoxy; alkenyl which is optionally identically or differently substituted by halogen, phenyl, halogenophenyl or halogenoalkylphenyl; alkinyl; cycloalkyl; alkoxy which is optionally substituted by halogen or cyano; phenyl which is optionally identically or differently substituted by halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, alkylsulphinyl, halogenoalkylsulphinyl, alkylsulphonyl or halogenoalkylsulphonyl; pyridyl; monoalkylamino, the alkyl part being optionally substituted by halogen, cyano, alkoxycarbonyl, dialkylaminocarbonyl, alkanyleneaminocarbonyl or oxaalkanyleneaminocarbonyl; 1-cyanocycloalkylamino; dialkylamino; alkanyleneamino; oxaalkanyleneamino; N-alkyl-N-phenylamino or phenylamino, in which the phenyl radical in each is optionally identically or differently substituted by halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, alkylsulphonyl, halogenoalkylsulphonyl, alkanylenedioxy, halogenoalkanylenedioxy or by --O--CHal.sub.2 --O--CHal.sub.2 -, orR.sup.4 represents alkyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, fluoroalkyl, alkenyl, alkinyl, cycloalkyl or alkoxy,R.sup.5 represents hydrogen, alkyl, alkoxyalkyl, alkylthioalkyl, fluoroalkyl, cyanoalkyl, alkenyl, alkinyl or cycloalkyl,R.sup.4 and R.sup.5, together with the adjacent nitrogen atom represent an optionally substituted heterocycle which can be substituted, in the alkylene chain, by further heteroatoms.