Pesticidal compounds
    2.
    发明授权
    Pesticidal compounds 失效
    杀虫化合物

    公开(公告)号:US5091414A

    公开(公告)日:1992-02-25

    申请号:US619872

    申请日:1990-11-29

    IPC分类号: C07F9/24

    CPC分类号: C07F9/2487

    摘要: A compound of Formula (I):(I) R.sup.1 (CA.dbd.CA.sup.1).sub.x --C(.dbd.X)NR.sup.2 R.sup.3where R.sup.1 is alkyl optionally substituted by a group selected from alkoxy, alkenyl, alkynyl, alkenyloxy, alkynyloxy, aryl, aryloxy, arylalkoxy and cycloalkyl fused to an aryl ring; x=1 or 2; X=O or S; each A and A.sup.1 is independently hydrogen, alkyl or haloalkyl; R.sup.2 is alkyl, alkenyl or cycloalkyl any of which may be substituted by halo, alkenyl, alkyl, cycloalkyl, alkynyl, dioxalanylalkyl or alkoxy; and R.sup.3 is selected from groups (A) to (D):(A) --Y=X.sup.1 --(R.sup.4).sub.a where X.sup.1 is O or S, Y is phosphorus or carbon, R.sup.4 is hydrogen, alkyl, alkoxy, acyl or CO.sub.2 R.sup.5 where R.sup.5 is alkyl or aryl, and a is 1 or 2(B) --S(R.sup.6)(O).sub.bwhere R.sup.6 is alkyl, aryl, aryloxy, alkoxy, thioalkoxy, thioaryl, alkythio, alkoxythio or arylthio and b is 0, 1 or 2(C) --S(O).sub.c NR.sup.7 R.sup.8where c is 0, 1 or 2, R.sup.7 is --COR.sup.9 or --CO.sub.2 R.sup.9 where R.sup.9 is hydrogen, alkyl or a fluorine atom, a group (A) or (B) as defined above, or alkyl substituted by acyl, carboalkoxy or cyano, and R.sup.8 is alkyl(D) R.sup.1 --(CA.dbd.CA.sup.1).sub.n --C(.dbd.X)N(R.sup.2)--wherein the subtituents are independently selected as in Formula (I) above.

    摘要翻译: 式(I)化合物:(I)R1(CA = CA1)xC(= X)NR2R3其中R1是任选被选自烷氧基,烯基,炔基,烯氧基,炔氧基,芳基,芳氧基,芳基烷氧基和芳氧基的基团取代的烷基, 稠合到芳环的环烷基; x = 1或2; X = O或S; 每个A和A1独立地是氢,烷基或卤代烷基; R2是烷基,烯基或环烷基,其中任何一个可以被卤素,烯基,烷基,环烷基,炔基,二氧戊环基烷基或烷氧基取代; (A)-Y = X1-(R4)a其中X1为O或S,Y为磷或碳,R4为氢,烷基,烷氧基,酰基或CO2R5 其中R 5是烷基或芳基,且a是1或2(B)-S(R 6)(O)b,其中R 6是烷基,芳基,芳氧基,烷氧基,硫代烷氧基,硫代芳基,链炔基,烷硫基或芳硫基,b是0, 1或2(C)-S(O)cNR 7 R 8,其中c是0,1或2,R 7是-COR 9或-CO 2 R 9,其中R 9是氢,烷基或氟原子,定义的基团(A)或(B) 或者被酰基,烷氧羰基或氰基取代的烷基,R8是烷基(D)R1-(CA = CA1)nC(= X)N(R2) - ,其中取代基如上式(I)所示独立选择。

    Herbicide compositions of extended soil life
    3.
    发明授权
    Herbicide compositions of extended soil life 失效
    除草剂组合物延长土壤寿命

    公开(公告)号:US4662930A

    公开(公告)日:1987-05-05

    申请号:US649638

    申请日:1984-09-12

    摘要: The soil life of herbicidally active thiolcarbamates is extended by employing in combination therewith certain organophosphorus compounds having the formula 3 ##STR1## in which R.sup.4 is selected from the group consisting of C.sub.1 -C.sub.4 alkyl and C.sub.1 -C.sub.4 alkoxy; R.sup.5 is selected from the group consisting of C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.2 -C.sub.4 alkenylthio and C.sub.2 -C.sub.4 alkynylthio; R.sup.6 is selected from the group consisting of hydrogen , C.sub.1 -C.sub.10 alkyl, C.sub.5 -C.sub.7 cycloalkyl and phenyl; and R.sup.7 is selected from the group consisting of C.sub.2 -C.sub.4 alkenyl, C.sub.1 -C.sub.10 alkoxy, C.sub.1 -C.sub.10 alkylthio, C.sub.2 -C.sub.6 alkynoxy, C.sub.2 -C.sub.5 carbalkoxy, phenyl, phenoxy, (C.sub.1 -C.sub.3 alkoxy)phenyl, benzyl and benzyloxy, all optionally substituted with up to two halogen atoms.

    摘要翻译: 除草活性硫代氨基​​甲酸酯的土壤寿命通过结合使用具有式3“IMAGE”的某些有机磷化合物延长,其中R 4选自C 1 -C 4烷基和C 1 -C 4烷氧基; R5选自C1-C4烷基,C1-C4烷氧基,C1-C4烷硫基,C2-C4烯硫基和C2-C4炔硫基; R 6选自氢,C 1 -C 10烷基,C 5 -C 7环烷基和苯基; 并且R 7选自C 2 -C 4烯基,C 1 -C 10烷氧基,C 1 -C 10烷硫基,C 2 -C 6炔氧基,C 2 -C 5烷氧羰基,苯基,苯氧基,(C 1 -C 3烷氧基)苯基,苄基和苄氧基, 全部任选被至多两个卤素原子取代。

    Phosphonylureidobenzene derivatives and their medicinal use
    5.
    发明授权
    Phosphonylureidobenzene derivatives and their medicinal use 失效
    膦酰基脲衍生物及其药用

    公开(公告)号:US4247546A

    公开(公告)日:1981-01-27

    申请号:US967035

    申请日:1978-12-06

    摘要: The invention includes phosphonylureidobenzene compounds of the general formula ##STR1## or pharmaceutically acceptable salts in whichR.sup.1 and R.sup.2 are identical or different and represent an alkyl group, orR.sup.1 and R.sup.2 together represent a dimethylene group, a trimethylene group or a tetramethylene group,X and Y are identical or different and represent an oxygen atom or a sulphur atom andR.sup.3 and R.sup.4 are identical or different and represent an alkyl group, orR.sup.3 and R.sup.4 together represent a trimethylene group or a tetramethylene group, orR.sup.3 and R.sup.4, together with the carbon atom and nitrogen atom between them, form a thiazolidine ring system, which are used medicinally as parasiticides.The compounds are particularly effective in combatting helminths in carnivores.Also included in the invention are pharmaceutical compositions containing said phosphonylureidobenzene compounds and methods for the treatment of warm-blooded animals by administering said compounds or compositions.

    摘要翻译: 本发明包括通式为(I)的膦酰基脲基化合物或其中R 1和R 2相同或不同并且表示烷基的药学上可接受的盐,或者R 1和R 2一起表示二亚甲基,三亚甲基或四亚甲基 基,X和Y相同或不同,表示氧原子或硫原子,R3和R4相同或不同,表示烷基,或R3和R4一起表示三亚甲基或四亚甲基,或R 3和R 4 与它们之间的碳原子和氮原子一起形成噻唑烷环体系,它们在医药上用作杀寄生虫剂。 这些化合物特别有效地对抗食肉动物的蠕虫。 本发明还包括含有所述膦酰基脲基化合物的药物组合物和通过施用所述化合物或组合物治疗温血动物的方法。

    Method for the control of cattle grubs employing a phenylene
bis[imino(thio]carbonyl)diphosphor(thio)-amidic acid ester
    6.
    发明授权
    Method for the control of cattle grubs employing a phenylene bis[imino(thio]carbonyl)diphosphor(thio)-amidic acid ester 失效
    使用亚苯基双{8亚氨基(硫代{9羰基)二磷(硫代) - 酰胺酸酯)控制tle的方法

    公开(公告)号:US4137310A

    公开(公告)日:1979-01-30

    申请号:US912812

    申请日:1978-06-05

    申请人: Guang T. Wang

    发明人: Guang T. Wang

    IPC分类号: A01N57/30 C07F9/24 A61K31/66

    CPC分类号: C07F9/2487 A01N57/30

    摘要: There is provided a method for controlling the larvae of heel flies which parasitize ruminants and other warm-blooded animals by administering to said animals an effective amount of an unsubstituted or substituted phenylene bis[imino(thio)carbonyl]diphosphor(thio)amidic acid ester.

    摘要翻译: 提供了一种通过向所述动物施用有效量的未取代或取代的亚苯基双[亚氨基(硫代)羰基]二磷酸(硫代)酰胺酸酯的方法来控制寄生反刍动物和其它温血动物的脚跟蝇幼虫的方法 。

    Alkylation of N-acyl-O-hydrocarbylphosphoroamidothioate salts
    9.
    发明授权
    Alkylation of N-acyl-O-hydrocarbylphosphoroamidothioate salts 失效
    N-酰基-O-烃基磷酰胺硫代磷酸盐的烷基化

    公开(公告)号:US3925520A

    公开(公告)日:1975-12-09

    申请号:US47997274

    申请日:1974-06-17

    申请人: CHEVRON RES

    发明人: FRANKE HANS G

    IPC分类号: C07F9/24

    CPC分类号: C07F9/2487

    摘要: S-ammonium (or metal) salts of N-acyl-Ohydrocarbylphosphoroamidothioates horoamidothioates are prepared by reacting an N-acyl-O,O-dihydrocarbylphosphoroamidothioate with an ammonium (or metal) sulfide or polysulfide. The S-ammonium (or metal) salts can be alkylated to produce an O-hydrocarbyl-Shydrocarbyl-N-acylphosphoroamidothioate.

    摘要翻译: 通过使N-酰基-O,O-二烃基磷酰氨基硫代磷酸酯与铵(或金属)硫化物或多硫化物反应来制备N-酰基-O-烃基磷酰氨基硫代磷酸酯horoamidothioates的S-铵(或金属)盐。 可以将S-铵(或金属)盐烷基化以制备O-烃基-S-烃基-N-酰基磷酰氨基硫代磷酸酯。

    N-acyl-o-hydrocarbylphosphoro-amidothioate salts
    10.
    发明授权
    N-acyl-o-hydrocarbylphosphoro-amidothioate salts 失效
    N-ACYL-O-氢氯化磷酰胺盐

    公开(公告)号:US3833623A

    公开(公告)日:1974-09-03

    申请号:US31747772

    申请日:1972-12-21

    申请人: CHEVRON RES

    发明人: MAGEE P

    IPC分类号: C07F9/24 C08H3/00 C08H9/02

    CPC分类号: C07F9/2487

    摘要: S-ALKALI METAL S-AMMONIUM SALTS OF N-ACYL-O-HYDROCARBYLPHOSPHOROAMIDOTHIOATES ARE PREPARED BY REACTING AN N-ACYL-O,O-DIHYDROCARBYLPHOSPHOROAMIDOTHIOATE WITH AN ALKALI METAL MERCAPTIDE OR AMMONIUM MERCAPTIDE.