公开(公告)号：WO2011101867A3

公开(公告)日：2012-04-26

申请号：PCT/IN2011000100

申请日：2011-02-18

Applicant: CADILA HEALTHCARE LTD ,  DWIVEDI SHRIPRAKASH DHAR ,  PRASAD ASHOK ,  ROY RUSHIKESH UDAYKUMAR ,  PATEL MAYUR RAMNIKBHAI

Inventor： DWIVEDI SHRIPRAKASH DHAR ,  PRASAD ASHOK ,  ROY RUSHIKESH UDAYKUMAR ,  PATEL MAYUR RAMNIKBHAI

IPC: C07D277/56 ,  A61K31/426 ,  A61P19/06

CPC classification number: C07D277/56

Abstract: Substantially pure salts of febuxostat of Formula (IA): wherein Y is Na+, K+, Li+, Mg2+, Ca2+, Zn2+, Ba2+, Sr2+, choline, epolamine and N+(R)4 and processes for preparation thereof are disclosed.

Abstract translation: 公开了式（IA）的Febostostat的基本纯盐：其中Y是Na +，K +，Li +，Mg 2+，Ca 2+，Zn 2+，Ba 2+，Sr 2+，胆碱，亚胺胺和N +（R）4及其制备方法。

公开(公告)号：WO2012025940A1

公开(公告)日：2012-03-01

申请号：PCT/IN2011/000572

申请日：2011-08-24

Applicant: CADILA HEALTHCARE LIMITED ,  DWIVEDI, Shriprakash, Dhar ,  PRASAD, Ashok ,  PATEL, Mahesh, Shankarbhai ,  SHARMA, Piyush, Rajendra

Inventor： DWIVEDI, Shriprakash, Dhar ,  PRASAD, Ashok ,  PATEL, Mahesh, Shankarbhai ,  SHARMA, Piyush, Rajendra

IPC: C07D223/16 ,  A61K31/55

CPC classification number: C07D223/16 ,  A61K31/55

Abstract: The present invention discloses Crystalline Form Zeta "ζ" of ivabradine hydrochloride and process for its preparation..

Abstract translation: 本发明公开了晶型Zeta“α” 伊伐布雷定盐酸盐及其制备方法

公开(公告)号：WO2011101867A2

公开(公告)日：2011-08-25

申请号：PCT/IN2011/000100

申请日：2011-02-18

Applicant: CADILA HEALTHCARE LIMITED ,  DWIVEDI, Shriprakash, Dhar ,  PRASAD, Ashok ,  ROY, Rushikesh, Udaykumar ,  PATEL, Mayur, Ramnikbhai

Inventor： DWIVEDI, Shriprakash, Dhar ,  PRASAD, Ashok ,  ROY, Rushikesh, Udaykumar ,  PATEL, Mayur, Ramnikbhai

CPC classification number: C07D277/56

Abstract: Substantially pure salts of febuxostat of Formula (IA): wherein Y is Na + , K + , Li + , Mg 2+ , Ca 2+ , Zn 2+ , Ba 2+ , Sr 2+ , choline, epolamine and N + (R) 4 and processes for preparation thereof are disclosed.

Abstract translation: 公开了具有式（IA）的Febostost的基本纯盐：其中Y是Na +，K +，Li +，Mg 2+，Ca 2+，Zn 2+，Ba 2+，Sr 2+，胆碱，亚胺胺和N +（R）4及其制备方法。

公开(公告)号：WO2010013157A3

公开(公告)日：2011-04-28

申请号：PCT/IB2009053043

申请日：2009-07-14

Applicant: ALEMBIC LTD ,  DEO KESHAV ,  PRASAD ASHOK ,  ARORA SUNIL

Inventor： DEO KESHAV ,  PRASAD ASHOK ,  ARORA SUNIL

IPC: C07H5/02

CPC classification number: C07H15/18 ,  A23L27/37 ,  C07H5/02 ,  C07H13/04 ,  Y02P20/582

Abstract: The present invention relates to cost efficient process for preparation of sucralose. The present invention relates to recovery of the reagents from feed mixture obtained in various steps of sucralose. Particularly, the present invention relates to recovery of trityl chloride, ß-picoline, triphenylphosphine oxide (TPPO) and methyl acetate.

Abstract translation: 本发明涉及用于制备三氯半乳蔗糖的成本有效的方法。 本发明涉及从三氯蔗糖各步骤中获得的饲料混合物中回收试剂。 特别地，本发明涉及三苯甲基氯，β-甲基吡啶，三苯基氧化膦（TPPO）和乙酸甲酯的回收。

公开(公告)号：WO2010070511A2

公开(公告)日：2010-06-24

申请号：PCT/IB2009/055414

申请日：2009-11-30

Applicant: ALEMBIC LIMITED ,  PONNAIAH, Ravi ,  PRASAD, Ashok ,  PANCHASARA, Dineshkumar Ramabhai ,  CHAVAN, Gajanan Jijaba ,  PRAJAPATI, Bhavesh Hareshbhai ,  PATEL, Ilesh Mahendrabhai

Inventor： PONNAIAH, Ravi ,  PRASAD, Ashok ,  PANCHASARA, Dineshkumar Ramabhai ,  CHAVAN, Gajanan Jijaba ,  PRAJAPATI, Bhavesh Hareshbhai ,  PATEL, Ilesh Mahendrabhai

IPC: C07D211/02

CPC classification number: C07D211/02 ,  C07D211/32 ,  C07D211/70

Abstract: The present invention relates to novel process for preparing Donepezil hydrochloride of formula (I)

Abstract translation: 本发明涉及制备式（I）的盐酸多奈哌齐的新方法，

公开(公告)号：WO2010067252A1

公开(公告)日：2010-06-17

申请号：PCT/IB2009/055407

申请日：2009-11-30

Applicant: ALEMBIC LIMITED ,  PONNAIAH, Ravi ,  PRASAD, Ashok ,  RANA, Piyush Maheshbhai ,  KANZARIYA, Kamlesh Shankarlal ,  DOLIA, Mitulkumar Bharatkumar

Inventor： PONNAIAH, Ravi ,  PRASAD, Ashok ,  RANA, Piyush Maheshbhai ,  KANZARIYA, Kamlesh Shankarlal ,  DOLIA, Mitulkumar Bharatkumar

IPC: C07C17/10 ,  C07C231/06 ,  C07C209/62

CPC classification number: C07C211/38 ,  C07C17/10 ,  C07C209/62 ,  C07C231/06 ,  C07C231/14 ,  C07C233/06 ,  C07C2603/74

Abstract: The present invention relates to an improved process for the preparation of 1-bromo-3,5-dimethyl adamantane of formula (III), which is an useful intermediate for synthesis of 1-amino-3,5-dimethyl adamantane of formula (I) or pharmaceutically acceptable salt thereof.

Abstract translation: 本发明涉及制备式（III）的1-溴-3,5-二甲基金刚烷的改进方法，其是用于合成式（I）的1-氨基-3,5-二甲基金刚烷的有用中间体 ）或其药学上可接受的盐。

公开(公告)号：WO2005016936A3

公开(公告)日：2005-08-11

申请号：PCT/IB2004002648

申请日：2004-08-13

Applicant: RANBAXY LAB LTD ,  KUMAR YATENDRA ,  PRASAD MOHAN ,  SINGH KAPTAN ,  PRASAD ASHOK ,  RICHHARIYA SANTOSH

Inventor： KUMAR YATENDRA ,  PRASAD MOHAN ,  SINGH KAPTAN ,  PRASAD ASHOK ,  RICHHARIYA SANTOSH

IPC: C07D501/00 ,  A61K31/545

CPC classification number: C07D501/00

Abstract: The present invention relates to a selective process for preparation of Z-isomer of cefditoren of Formula I and pharmaceutically acceptable salts and esters thereof. cefditoren possesses a wide spectrum of antibacterial activity against Gram-positive and Gram-negative bacteria.

Abstract translation: 本发明涉及制备式I的头孢托仑的Z-异构体的选择性方法及其药学上可接受的盐和酯。 头孢托仑具有抗革兰氏阳性和革兰氏阴性菌的广谱抗菌活性。

公开(公告)号：WO2002060866A3

公开(公告)日：2002-08-08

申请号：PCT/IB2002/000264

申请日：2002-01-29

Applicant: RANBAXY LABORATORIES LIMITED ,  KUMAR, Yatendra ,  PRASAD, Mohan ,  PRASAD, Ashok

Inventor： KUMAR, Yatendra ,  PRASAD, Mohan ,  PRASAD, Ashok

IPC: C07D501/26

Abstract: The present invention relates to an improved and industrially advantageous process for the preparation of pure 7-amino-3-alkoxymethyl-3-cephem-4-carboxylic acids, and salts thereof. In particular, the present invention relates to a process for the preparation of pure 7-amino-3-methoxymethyl-3-cephem-4-carboxylic acid (7-AMCA) and salts thereof.

公开(公告)号：WO2002060866A2

公开(公告)日：2002-08-08

申请号：PCT/IB2002/000264

申请日：2002-01-29

Applicant: RANBAXY LABORATORIES LIMITED ,  KUMAR, Yatendra ,  PRASAD, Mohan ,  PRASAD, Ashok

Inventor： KUMAR, Yatendra ,  PRASAD, Mohan ,  PRASAD, Ashok

IPC: C07D

CPC classification number: C07D501/00

Abstract: The present invention relates to an improved and industrially advantageous process for the preparation of pure 7-amino-3-alkoxymethyl-3-cephem-4-carboxylic acids, and salts thereof. In particular, the present invention relates to a process for the preparation of pure 7-amino-3-methoxymethyl-3-cephem-4-carboxylic acid (7-AMCA) and salts thereof.

Abstract translation: 本发明涉及用于制备纯的7-氨基-3-烷氧基甲基-3-头孢烯-4-羧酸的改进和工业上有利的方法及其盐。 特别地，本发明涉及制备纯的7-氨基-3-甲氧基甲基-3-头孢烯-4-羧酸（7-AMCA）及其盐的方法。

公开(公告)号：WO2013098833A3

公开(公告)日：2013-10-10

申请号：PCT/IN2012000599

申请日：2012-09-10

Applicant: CADILA HEALTHCARE LTD ,  DWIVEDI SHRIPRAKASH DHAR ,  PRASAD ASHOK ,  PAL DAYA RAM ,  SHARMA MUKUL HARI PRASAD ,  JAIN KULDEEP NATWARLAL ,  PATEL NAITIK BHARATBHAI

Inventor： DWIVEDI SHRIPRAKASH DHAR ,  PRASAD ASHOK ,  PAL DAYA RAM ,  SHARMA MUKUL HARI PRASAD ,  JAIN KULDEEP NATWARLAL ,  PATEL NAITIK BHARATBHAI

IPC: C07D413/14 ,  C07D413/10

CPC classification number: C07D413/14 ,  C07D265/32 ,  C07D413/10

Abstract: The invention discloses processes for the preparation of rivaroxaban and its pharmaceutically acceptable salts, solvates, and hydrates thereof. The invention also relates to novel intermediates for the preparation of rivaroxaban.

Abstract translation: 本发明公开了制备利伐沙班及其药学上可接受的盐，溶剂化物和水合物的方法。 本发明还涉及用于制备利伐沙班的新型中间体。