公开(公告)号：WO2012103041A2

公开(公告)日：2012-08-02

申请号：PCT/US2012022285

申请日：2012-01-24

Applicant: DOW AGROSCIENCES LLC ,  ARNDT KIM E ,  RENGA JAMES M ,  ZHU YUANMING ,  WHITEKER GREGORY T ,  LOWE CHRISTIAN T

Inventor： ARNDT KIM E ,  RENGA JAMES M ,  ZHU YUANMING ,  WHITEKER GREGORY T ,  LOWE CHRISTIAN T

IPC: C07D213/79 ,  C07D213/803 ,  C07D213/81 ,  C07D213/84

CPC classification number: C07D213/84 ,  C07D213/79 ,  C07D213/803 ,  C07D213/81

Abstract: 4-Amino-3-chloro-5-fluoro-6-(substituted)picolinates are conveniently prepared from 3,4,5,6-tetrachloropicolinonitrile by a series of steps involving fluorine exchange, amination, halogen exchange and hydrolysis, esterification and transition metal assisted coupling.

Abstract translation: 通过一系列涉及氟交换，胺化，卤素交换和水解，酯化和转化的步骤，方便地从3,4,5,6-四氯吡啶腈制备4-氨基-3-氯-5-氟-6-（取代的）吡啶甲酸盐 金属辅助联轴器。

公开(公告)号：WO2012061290A3

公开(公告)日：2012-05-10

申请号：PCT/US2011/058578

申请日：2011-10-31

Applicant: DOW AGROSCIENCES LLC ,  YAP, Maurice C. H. ,  BUYSSE, Ann M. ,  KNUEPPEL, Daniel ,  ZHANG, Yu ,  GARIZI, Negar ,  NIYAZ, Noormohamed M. ,  LOWE, Christian T. ,  HUNTER, Ricky ,  TRULLINGER, Tony K. ,  DEMETER, David A. ,  PERNICH, Dan ,  DEAMICIS, Carl ,  ROSS, Ronald ,  JOHNSON, Timothy C.

Inventor： YAP, Maurice C. H. ,  BUYSSE, Ann M. ,  KNUEPPEL, Daniel ,  ZHANG, Yu ,  GARIZI, Negar ,  NIYAZ, Noormohamed M. ,  LOWE, Christian T. ,  HUNTER, Ricky ,  TRULLINGER, Tony K. ,  DEMETER, David A. ,  PERNICH, Dan ,  DEAMICIS, Carl ,  ROSS, Ronald ,  JOHNSON, Timothy C.

IPC: A01N43/50 ,  A61K31/415

Abstract: This document discloses molecules having the following formula (I): and processes related thereto.

公开(公告)号：WO2012103041A3

公开(公告)日：2012-08-02

申请号：PCT/US2012/022285

申请日：2012-01-24

Applicant: DOW AGROSCIENCES LLC ,  ARNDT, Kim E. ,  RENGA, James M. ,  ZHU, Yuanming ,  WHITEKER, Gregory T. ,  LOWE, Christian T.

Inventor： ARNDT, Kim E. ,  RENGA, James M. ,  ZHU, Yuanming ,  WHITEKER, Gregory T. ,  LOWE, Christian T.

IPC: A01N43/40

Abstract: 4-Amino-3-chloro-5-fluoro-6-(substituted) picolinates are conveniently prepared from 3,4;5,6-tetrachloropicolinonitrile by a series of steps involving fluorine exchange, amination, halogen exchange and hydrolysis, esterification and transition metal assisted coupling. The present invention concerns a process for the preparation of 4-amino-3-chloro-5-fluoro-6-(substituted)picolinates. More particularly, the present invention concerns a process for the preparation of 4-amino-3-chloro-5-fluoro-6-(substituted)picolinates in which the 5-fluoro substituent is introduced by a halogen exchange early in the process scheme.

公开(公告)号：WO2013003740A1

公开(公告)日：2013-01-03

申请号：PCT/US2012/044970

申请日：2012-06-29

Applicant: DOW AGROSCIENCES LLC ,  EPP, Jeffrey, B. ,  LOWE, Christian, T. ,  RENGA, James, M. ,  SCHMITZER, Paul, R. ,  ECKELBARGER, Joseph, D. ,  GUENTHENSPBERGER, Katherine, A. ,  SIDDALL, Thomas, L. ,  YERKES, Carla, N. ,  FISCHER, Lindsey, Gayle ,  GIAMPIETRO, Natalie, Christine ,  KISTER, Jeremy ,  ROTH, Joshua

Inventor： EPP, Jeffrey, B. ,  LOWE, Christian, T. ,  RENGA, James, M. ,  SCHMITZER, Paul, R. ,  ECKELBARGER, Joseph, D. ,  GUENTHENSPBERGER, Katherine, A. ,  SIDDALL, Thomas, L. ,  YERKES, Carla, N. ,  FISCHER, Lindsey, Gayle ,  GIAMPIETRO, Natalie, Christine ,  KISTER, Jeremy ,  ROTH, Joshua

IPC: A01N43/40

CPC classification number: C07D213/79 ,  A01N43/40 ,  A01N55/00 ,  C07D213/65 ,  C07D213/73 ,  C07D405/04 ,  C07F7/0812 ,  C07F7/082

Abstract: 3-alkoxy, thioalkyl and amino-4-amino-6-(substituted)picolinic acids having a halogen, alkyl or mono-, di- tri- and tetra-substituted aryl substituents in the 6-position, and their acid derivatives, are herbicides demonstrating a broad spectrum of weed control.

Abstract translation: 在6-位具有卤素，烷基或一取代，二取代和四取代的芳基取代基的3-烷氧基，硫代烷基和氨基-4-氨基-6-（取代的）吡啶甲酸及其酸衍生物是 表现出广泛杂草控制的除草剂。

公开(公告)号：WO2012103042A1

公开(公告)日：2012-08-02

申请号：PCT/US2012/022286

申请日：2012-01-24

Applicant: DOW AGROSCIENCES LLC ,  YERKES, Carla N. ,  LOWE, Christian T. ,  ECKELBARGER, Joseph D. ,  EPP, Jeffrey B. ,  GUENTHENSPBERGER, Katherine A. ,  SIDDALL, Thomas L. ,  SCHMITZER, Paul R.

Inventor： YERKES, Carla N. ,  LOWE, Christian T. ,  ECKELBARGER, Joseph D. ,  EPP, Jeffrey B. ,  GUENTHENSPBERGER, Katherine A. ,  SIDDALL, Thomas L. ,  SCHMITZER, Paul R.

IPC: A01N43/90 ,  A61K31/519

CPC classification number: C07D239/42 ,  A01N43/40 ,  A01N43/54 ,  C07D213/73 ,  C07D213/79 ,  C07D239/34 ,  C07D239/47 ,  C07D405/12

Abstract: Arylalkyl esters of 4-aminopicolinic acids and 6-amino-4-pyrimidinecarboxylates are herbicides for control of weeds especially those species common to rice and wheat cropping systems and in pasture management programs.

Abstract translation: 4-氨基吡啶甲酸和6-氨基-4-嘧啶羧酸盐的芳基烷基酯是用于防治杂草的除草剂，特别是用于水稻和小麦作物系统以及牧场管理程序中常见的杂草。

公开(公告)号：WO2012061290A2

公开(公告)日：2012-05-10

申请号：PCT/US2011058578

申请日：2011-10-31

Applicant: DOW AGROSCIENCES LLC ,  YAP MAURICE C H ,  BUYSSE ANN M ,  KNUEPPEL DANIEL ,  ZHANG YU ,  GARIZI NEGAR ,  NIYAZ NOORMOHAMED M ,  LOWE CHRISTIAN T ,  HUNTER RICKY ,  TRULLINGER TONY K ,  DEMETER DAVID A ,  PERNICH DAN ,  DEAMICIS CARL ,  ROSS RONALD ,  JOHNSON TIMOTHY C

Inventor： YAP MAURICE C H ,  BUYSSE ANN M ,  KNUEPPEL DANIEL ,  ZHANG YU ,  GARIZI NEGAR ,  NIYAZ NOORMOHAMED M ,  LOWE CHRISTIAN T ,  HUNTER RICKY ,  TRULLINGER TONY K ,  DEMETER DAVID A ,  PERNICH DAN ,  DEAMICIS CARL ,  ROSS RONALD ,  JOHNSON TIMOTHY C

IPC: A61K31/4439 ,  A01H5/10 ,  A01N25/34 ,  A01P1/00 ,  A01P3/00 ,  A01P5/00 ,  A01P7/02 ,  A01P7/04 ,  A01P9/00 ,  A01P11/00 ,  A01P13/00 ,  A01P15/00 ,  A01P17/00 ,  A01P19/00 ,  A01P21/00 ,  A01P23/00 ,  A61K31/444 ,  C07D401/04 ,  C07D401/14 ,  C07D417/14

CPC classification number: C07D417/14 ,  A01N25/00 ,  A01N43/12 ,  A01N43/56 ,  A01N43/653 ,  A01N43/74 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N47/18 ,  A01N47/36 ,  A01N47/40 ,  A01N51/00 ,  A61K31/4439 ,  A61K31/506 ,  A61K45/06 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14

Abstract: This document discloses molecules having the following formula (I): and processes related thereto.

Abstract translation: 该文献公开了具有下式（I）的分子及其相关的方法。

公开(公告)号：WO2012116246A3

公开(公告)日：2014-04-24

申请号：PCT/US2012026418

申请日：2012-02-24

Applicant: DOW AGROSCIENCES LLC ,  LOWE CHRISTIAN T ,  TRULLINGER TONY K ,  HUNTER RICKY

Inventor： LOWE CHRISTIAN T ,  TRULLINGER TONY K ,  HUNTER RICKY

IPC: A01H5/00 ,  A01N43/40 ,  C07D401/00

CPC classification number: A01N43/56 ,  C07D401/04 ,  C07D401/14

Abstract: This document discloses pesticidal molecules having the following formula ("Formula One"): and processes related thereto.

Abstract translation: 该文献公开了具有下式（“一级方程式”）的杀虫剂分子及其相关的方法。

公开(公告)号：WO2012116246A2

公开(公告)日：2012-08-30

申请号：PCT/US2012/026418

申请日：2012-02-24

Applicant: DOW AGROSCIENCES LLC ,  LOWE, Christian, T. ,  TRULLINGER, Tony, K. ,  HUNTER, Ricky

Inventor： LOWE, Christian, T. ,  TRULLINGER, Tony, K. ,  HUNTER, Ricky

IPC: A01N43/56 ,  C07D401/14 ,  A01C1/06 ,  A61K31/444 ,  C07D401/04 ,  A61K31/4439 ,  A61P33/14 ,  A01P7/02 ,  A01P7/04 ,  A01P5/00

CPC classification number: A01N43/56 ,  C07D401/04 ,  C07D401/14

Abstract: This document discloses pesticidal molecules having the following formula ("Formula One"): and processes related thereto.

Abstract translation: 该文献公开了具有下式（“一级方程式”）的杀虫剂分子及其相关的方法。

公开(公告)号：WO2012103047A1

公开(公告)日：2012-08-02

申请号：PCT/US2012/022291

申请日：2012-01-24

Applicant: DOW AGROSCIENCES LLC ,  WHITEKER, Gregory, T. ,  ARNDT, Kim, E. ,  RENGA, James, M. ,  ZHU, Yuanming ,  LOWE, Christian, T. ,  SIDDALL, Thomas, L. ,  PODHOREZ, David, E. ,  ROTH, Gary, Alan ,  WEST, Scott, P.

Inventor： WHITEKER, Gregory, T. ,  ARNDT, Kim, E. ,  RENGA, James, M. ,  ZHU, Yuanming ,  LOWE, Christian, T. ,  SIDDALL, Thomas, L. ,  PODHOREZ, David, E. ,  ROTH, Gary, Alan ,  WEST, Scott, P.

IPC: A01N43/40 ,  C07D213/04

CPC classification number: C07D213/803 ,  C07D213/79

Abstract: 4-Amino-5-fluoro-3-halo-6-(substituted)picolinates are conveniently prepared from 4,5,6-trichloropicolinates by a series of steps involving fluorine exchange, amination, halogen exchange, halogenation and transition metal assisted coupling.

Abstract translation: 通过涉及氟交换，胺化，卤素交换，卤化和过渡金属辅助偶联的一系列步骤，方便地由4,5,6-三氯吡啶酸盐制备4-氨基-5-氟-3-卤代-6-（取代的）吡啶甲酸盐。