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    PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    1.
    发明申请
    PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
    作为杀菌剂有用的吡咯烷酮酸酰胺衍生物

    公开(公告)号：WO2003048128A1

    公开(公告)日：2003-06-12

    申请号：PCT/GB2002/005303

    申请日：2002-11-25

    Applicant: SYNGENTA LIMITED ,  SYNGENTA PARTICIPATIONS AG ,  WHITTINGHAM, William, Guy ,  LAWSON, Kevin, Robert ,  WORTHINGTON, Paul, Anthony ,  RUSSELL, Charles, Adam ,  SALMON, Roger ,  MAY, Leslie, Francis ,  JORG, Mario ,  PACHLATKO, Johannes, Paul

    Inventor： WHITTINGHAM, William, Guy ,  LAWSON, Kevin, Robert ,  WORTHINGTON, Paul, Anthony ,  RUSSELL, Charles, Adam ,  SALMON, Roger ,  MAY, Leslie, Francis ,  JORG, Mario ,  PACHLATKO, Johannes, Paul

    IPC: C07D213/65

    CPC classification number: C07D213/70 ,  A01N43/40 ,  C07D213/65 ,  C07D213/68 ,  C07D213/80 ,  C07D213/82 ,  C07D213/85

    Abstract: Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.

    Abstract translation: 通式（I）的杀真菌化合物：其中X和Y独立地为H，卤素，C 1-8烷基，C 3-6环烷基，C 2-8链烯基，C 2-8 炔基，C> 1-8 <烷氧基，C 1-8烷基硫基，硝基，氨基，单 - 或二 - （C 1-6）烷基氨基，单 - 或二 - （C 2-6） 链烯基氨基，单 - 或二 - （C 2-6）炔基氨基，甲酰氨基，C 1-4烷基（甲酰基）氨基，C 1-4烷基羰基氨基，C 1-4烷基（C 1 -4 <烷基羰基）氨基，氰基，甲酰基，C 1-4烷基羰基，C 1-4烷氧基羰基，氨基羰基，一或二 - （C 1-4）烷基氨基羰基，羧基， 4 <烷基羰基氧基，芳基（C 1-4）烷基羰基氧基，C 1-4烷基亚磺酰基，C 1-4烷基磺酰基，C 1-4烷基磺酰氧基，芳基，杂芳基，芳氧基，芳硫基，杂芳氧基或杂芳硫基 其中任何前述烷基，环烷基，烯基，炔基，芳基，杂芳基，基团或部分任选被取代; R 1是苯基，氰基，C 1-4烷基，C 2-4链烯基或C 2-4炔基，其中烷基，烯基和炔基在其末端碳原子上任选被一个，两个或三个卤素原子取代， 具有C 1-4烷基羰基，C 1-4烷氧基羰基或羟基的氰基，或者R 1是烷基烷基或烷基磺酰基烷基，其中总碳原子数为2或3的烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基或烷基磺酰基烷基 ; R 2是H，C 1-4烷基，C 1-4烷氧基甲基或苄氧基甲基，其中苄基部分的苯环任选被C 1-4烷氧基取代; R 3和R 4独立地是H，C 1-3烷基，C 2-3烯基或C 2-3炔基，条件是两者都不是H，当两者都不是H时，它们的总碳原子数不超过 4或R 3和R 4与它们所连接的碳原子一起形成任选含有一个O，S或N原子并任选被卤素或C 1-4烷基取代的3或4元碳环 ; 羟基，C 1-6烷氧基，C 1-6烷硫基，氰基，C 1-4烷基羰基氧基，氨基羰基氧基，C 1-4烷氧基，C 1-4烷氧基， ，单或二（C 1-4）烷基氨基羰基氧基或三（C 1-4）烷基甲硅烷氧基。 含有它们的化合物和组合物特别可用于防治植物的真菌感染。

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