中科微点-全球专利检索

  1. Login
  2. Sign Up

Search Results

8 records (took 0.012 seconds)

    PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    1.
    发明申请
    PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
    作为杀菌剂有用的吡咯烷酮酸酰胺衍生物

    公开(公告)号：WO2003048128A1

    公开(公告)日：2003-06-12

    申请号：PCT/GB2002/005303

    申请日：2002-11-25

    Applicant: SYNGENTA LIMITED ,  SYNGENTA PARTICIPATIONS AG ,  WHITTINGHAM, William, Guy ,  LAWSON, Kevin, Robert ,  WORTHINGTON, Paul, Anthony ,  RUSSELL, Charles, Adam ,  SALMON, Roger ,  MAY, Leslie, Francis ,  JORG, Mario ,  PACHLATKO, Johannes, Paul

    Inventor： WHITTINGHAM, William, Guy ,  LAWSON, Kevin, Robert ,  WORTHINGTON, Paul, Anthony ,  RUSSELL, Charles, Adam ,  SALMON, Roger ,  MAY, Leslie, Francis ,  JORG, Mario ,  PACHLATKO, Johannes, Paul

    IPC: C07D213/65

    CPC classification number: C07D213/70 ,  A01N43/40 ,  C07D213/65 ,  C07D213/68 ,  C07D213/80 ,  C07D213/82 ,  C07D213/85

    Abstract: Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.

    Abstract translation: 通式（I）的杀真菌化合物：其中X和Y独立地为H，卤素，C 1-8烷基，C 3-6环烷基，C 2-8链烯基，C 2-8 炔基，C> 1-8 <烷氧基，C 1-8烷基硫基，硝基，氨基，单 - 或二 - （C 1-6）烷基氨基，单 - 或二 - （C 2-6） 链烯基氨基，单 - 或二 - （C 2-6）炔基氨基，甲酰氨基，C 1-4烷基（甲酰基）氨基，C 1-4烷基羰基氨基，C 1-4烷基（C 1 -4 <烷基羰基）氨基，氰基，甲酰基，C 1-4烷基羰基，C 1-4烷氧基羰基，氨基羰基，一或二 - （C 1-4）烷基氨基羰基，羧基， 4 <烷基羰基氧基，芳基（C 1-4）烷基羰基氧基，C 1-4烷基亚磺酰基，C 1-4烷基磺酰基，C 1-4烷基磺酰氧基，芳基，杂芳基，芳氧基，芳硫基，杂芳氧基或杂芳硫基 其中任何前述烷基，环烷基，烯基，炔基，芳基，杂芳基，基团或部分任选被取代; R 1是苯基，氰基，C 1-4烷基，C 2-4链烯基或C 2-4炔基，其中烷基，烯基和炔基在其末端碳原子上任选被一个，两个或三个卤素原子取代， 具有C 1-4烷基羰基，C 1-4烷氧基羰基或羟基的氰基，或者R 1是烷基烷基或烷基磺酰基烷基，其中总碳原子数为2或3的烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基或烷基磺酰基烷基 ; R 2是H，C 1-4烷基，C 1-4烷氧基甲基或苄氧基甲基，其中苄基部分的苯环任选被C 1-4烷氧基取代; R 3和R 4独立地是H，C 1-3烷基，C 2-3烯基或C 2-3炔基，条件是两者都不是H，当两者都不是H时，它们的总碳原子数不超过 4或R 3和R 4与它们所连接的碳原子一起形成任选含有一个O，S或N原子并任选被卤素或C 1-4烷基取代的3或4元碳环 ; 羟基，C 1-6烷氧基，C 1-6烷硫基，氰基，C 1-4烷基羰基氧基，氨基羰基氧基，C 1-4烷氧基，C 1-4烷氧基， ，单或二（C 1-4）烷基氨基羰基氧基或三（C 1-4）烷基甲硅烷氧基。 含有它们的化合物和组合物特别可用于防治植物的真菌感染。

    FUNGICIDES
    2.
    发明申请
    FUNGICIDES 审中-公开
    杀菌剂

    公开(公告)号：WO1997011951A1

    公开(公告)日：1997-04-03

    申请号：PCT/GB1996002228

    申请日：1996-09-10

    Applicant: ZENECA LIMITED ,  LAWSON, Kevin, Robert ,  MOUND, William, Roderick ,  WHITTINGHAM, William, Guy

    Inventor： ZENECA LIMITED

    IPC: C07F05/02

    CPC classification number: C07F5/027 ,  A01N55/08

    Abstract: A compound of formula (I), wherein A and A are, independently, phenyl, furyl or thienyl each optionally substituted by halogen, C1-4alkyl, C1-4alkoxy, C1-4alkylthio, C1-4haloalkyl, C1-4haloalkoxy or C1-4haloalkylthio; R is C1-4alkyl, C1-4haloalkyl, C2-4alkenyl, C2-4haloalkenyl, C3-7cycloalkyl, C3-7cycloalkyl(C1-4)alkyl, benzyl or phenyl, wherein benzyl and phenyl are optionally substituted by halogen, C1-4alkyl, C1-4haloalkyl, C1-4alkoxy or C1-4haloalkoxy; and R and R are, independently, hydrogen, C1-8alkyl, C1-8haloalkyl, C1-8alkoxy, C1-8haloalkoxy, halogen, nitro, COR , NR R or phenyl (optionally substituted by halogen, C1-4alkyl, C1-4haloalkyl, C1-4alkoxy, C1-4haloalkoxy or NR R ); or R and R join together to form a ring, the ring being optionally substituted by halogen, C1-4alkyl, C1-4haloalkyl, C1-4alkoxy, C1-4haloalkoxy or nitro; and R , R and R are independently hydrogen or C1-4alkyl.

    Abstract translation: 式（I）的化合物，其中A 1和A 2独立地是苯基，呋喃基或噻吩基，其各自任选被卤素，C 1-4烷基，C 1-4烷氧基，C 1-4烷硫基，C 1-4卤代烷基，C 1 -4卤代烷氧基或C1-4卤代烷硫基; R为C 1-4烷基，C 1-4卤代烷基，C 2-4烯基，C 2-4卤代烯基，C 3-7环烷基，C 3-7环烷基（C 1-4）烷基，苄基或苯基，其中苄基和苯基任选被卤素，C 1-4烷基， C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基; R 1和R 2独立地是氢，C 1-8烷基，C 1-8卤代烷基，C 1-8烷氧基，C 1-8卤代烷氧基，卤素，硝基，COR 7，NR 5 R 6或 苯基（任选被卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基或NR 5 R 6取代）; 或R 1和R 2连接在一起形成环，该环任选被卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基或硝基取代; 和R 5，R 6和R 7独立地是氢或C 1-4烷基。

    FUNGICIDES
    3.
    发明申请
    FUNGICIDES 审中-公开
    杀菌剂

    公开(公告)号：WO1995007022A1

    公开(公告)日：1995-03-16

    申请号：PCT/GB1994001751

    申请日：1994-08-11

    Applicant: ZENECA LIMITED ,  CROWLEY, Patrick, Jelf ,  HEANEY, Stephen, Paul ,  LAWSON, Kevin, Robert ,  YOULE, David

    Inventor： ZENECA LIMITED

    IPC: A01N37/44

    CPC classification number: A01N43/36 ,  A01N37/44 ,  A01N37/46 ,  A01N43/08 ,  A01N43/10 ,  A01N47/18 ,  C07C229/48 ,  C07C235/54 ,  C07C237/20 ,  C07C271/24 ,  C07C2601/08 ,  C07D207/16 ,  C07D307/24 ,  Y02P20/55

    Abstract: A method of combating fungi which comprises applying to a plant, to a seed of a plant or to the locus of a seed or plant a compound of formula (I), wherein X is O, S, SO, SO2, NR or CLM; A, B, D, E, L and M are, independently, hydrogen, halogen, alkyl, mono- or di-haloalkyl, benzyl (optionally substituted by halogen or haloalkyl) or hydroxy; A and B or D and E or L and M may together form a =S, =O or =CR R group; B and L or D and L may together form a bond; V is O or NR ; R and R are, independently, hydrogen or an amine protecting group; R , R and R are, independently, hydrogen, alkyl or benzyl; R and R are, independently, hydrogen, halogen, alkyl, phenyl, benzyl, alkoxy or acyloxy; or a salt thereof; provided that when X is CLM, R , R , R , A, M, D and E are all hydrogen, L and B are either both hydrogen or together form a bond, and V is O then the compound of formula (I) is in the form of a salt, but not a hydrochloride salt.

    Abstract translation: 一种防治真菌的方法，其包括向植物，植物种子或种子或植物的场所施用式（I）化合物，其中X为O，S，SO，SO 2，NR 8， 或CLM; A，B，D，E，L和M独立地为氢，卤素，烷基，单 - 或二 - 卤代烷基，苄基（任选被卤素或卤代烷基）或羟基取代; A和B或D和E或L和M可以一起形成= S，= O或= CR 6 R 7组; B和L或D和L可以一起形成键; V是O或NR 4; R 1和R 2独立地是氢或胺保护基; R 3，R 4和R 8独立地是氢，烷基或苄基; R 6和R 7独立地是氢，卤素，烷基，苯基，苄基，烷氧基或酰氧基; 或其盐; 条件是当X为CLM时，R 1，R 2，R 3，A，M，D和E均为氢，L和B均为氢或一起形成键，V为O 那么式（I）的化合物是盐的形式，而不是盐酸盐。

    HERBICIDAL COMPOUNDS
    5.
    发明申请
    HERBICIDAL COMPOUNDS 审中-公开
    除草化合物

    公开(公告)号：WO2012045721A2

    公开(公告)日：2012-04-12

    申请号：PCT/EP2011/067278

    申请日：2011-10-04

    Applicant: SYNGENTA LIMITED ,  MORRIS, James Alan ,  MITCHELL, Glynn ,  LAWSON, Kevin Robert ,  HUNT, James Charle Atlee

    Inventor： MORRIS, James Alan ,  MITCHELL, Glynn ,  LAWSON, Kevin Robert ,  HUNT, James Charle Atlee

    IPC: A01N43/42

    CPC classification number: H04H40/45 ,  A01N43/90 ,  C07D471/04

    Abstract: The present invention relates to novel herbicidal oxopyridine and thionopyridine derivatives of Formula (I), or an agronomically acceptable salt of said compound wherein R 1 , X 1 , X 2 , X 3 , X 4 , A 1 , R a , R b , R c and R d are as defined herein. The invention further relates to processes and intermediates for the preparation of the oxopyridine derivatives, to compositions which comprise the herbicidal compounds, and to their use for controlling weeds, in particular in crops of useful plants.

    Abstract translation: 本发明涉及式（I）的新型除草氧代吡啶和硫代吡啶衍生物，或其中R1，X1，X2，X3，X4，A1，Ra，Rb，Rc和Rd如本文所定义的所述化合物的农艺学上可接受的盐。 本发明还涉及用于制备氧代吡啶衍生物的方法和中间体，包含除草化合物的组合物及其用于控制​​杂草的用途，特别是在有用植物的作物中。

    4-ACYLAMINOBENZAMIDES AND THEIR USE AS FUNGICIDES
    6.
    发明申请
    4-ACYLAMINOBENZAMIDES AND THEIR USE AS FUNGICIDES 审中-公开
    4-ACYLAMINOBENZAMIDES及其作为防腐剂使用

    公开(公告)号：WO1994000422A2

    公开(公告)日：1994-01-06

    申请号：PCT/GB1993001115

    申请日：1993-05-28

    Applicant: ZENECA LIMITED ,  CROWLEY, Jelf, Patrick ,  LAWSON, Kevin, Robert

    Inventor： ZENECA LIMITED

    IPC: C07C237/42

    CPC classification number: C07C237/42 ,  A01N37/46 ,  A01N37/52 ,  C07C259/10

    Abstract: A fungicidal compound having formula (I), wherein either: A and B are both fluoro; W is oxygen; Z is NR'R''; R' is C1-4 alkyl; R'' is C1-4 alkyl, C1-4 alkoxy or C1-4 haloalkyl; and R3 is C(CH3)2F; provided that when R' is methyl then R'' is not ethyl; oŸ rŸ A and B are, independently, hydrogen, halogen, C1-4 alkyl, C1-4 alkoxy or C1-4 haloalkyl; W is N-X-R2; Z is YR1; X is oxygen, sulphur or a bond; Y is oxygen or sulphur; R1 and R2 are, independently, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, heterocyclyl, heterocyclylalkyl, heterocyclyloxyalkyl, alkoxyalkyl or alkylthioalkyl, or R1 and R2 join to form a ring; R3 is optionally substituted alkyl, optionally substituted alkoxy, optionally substituted cycloalkyl, optionally substituted alkenyl, optionally substituted alkynyl or R4R5N; R4 and R5 are, independently, alkyl, alkylcarbonyl, formyl or hydrogen; and metal complexes thereof.

    Abstract translation: 具有式（I）的杀真菌化合物，其中：A和B均为氟; W是氧; Z是NR'R“; R'是C 1-4烷基; R“是C 1-4烷基，C 1-4烷氧基或C 1-4卤代烷基; 并且R 3是C（CH 3）2 F; 条件是当R'是甲基时，R“不是乙基; A，B分别独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基或C 1-4卤代烷基; W是N-X-R2; Z是YR1; X是氧，硫或键; Y是氧或硫; R1和R2独立地是烷基，卤代烷基，烯基，炔基，环烷基，环烷基烷基，杂环基，杂环基烷基，杂环基烷氧基，烷氧基烷基或烷硫基烷基，或R1和R2连接形成环; R 3是任选取代的烷基，任选取代的烷氧基，任选取代的环烷基，任选取代的烯基，任选取代的炔基或R 4 R 5 N; R4和R5独立地是烷基，烷基羰基，甲酰基或氢; 及其金属络合物。

    FUNGICIDES
    8.
    发明申请
    FUNGICIDES 审中-公开
    杀菌剂

    公开(公告)号：WO1997011952A1

    公开(公告)日：1997-04-03

    申请号：PCT/GB1996002230

    申请日：1996-09-10

    Applicant: ZENECA LIMITED ,  LAWSON, Kevin, Robert ,  MOUND, William, Roderick ,  WHITTINGHAM, William, Guy

    Inventor： ZENECA LIMITED

    IPC: C07F05/02

    CPC classification number: A01N55/08 ,  C07F5/027

    Abstract: A compound of formula (I) wherein A and A are, independently, phenyl, furyl or thienyl each optionally substituted by halogen, C1-4 alkyl, C1-4 alkoxy, C1-4 alkylthio, C1-4 haloalkyl, C1-4 haloalkoxy or C1-4 haloalkylthio; R is C1-4 alkyl, C1-4 haloakyl, C2-4 alkenyl, C2-4 haloalkenyl, C3-7 cycloalkyl, C3-7 cycloalkyl(C1-4)alkyl, benzyl or phenyl, wherein benzyl and phenyl are optionally substituted by halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy; and R , R , R and R are, independently, hydrogen, C1-8 alkyl, C1-8 haloalkyl, C1-8 alkoxy, C1-8 haloalkoxy, halogen, nitro, COR , NR R , benzyl or phenyl (wherein benzyl and phenyl are optionally substituted by halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 haloalkoxy or NR R ); R and R or R and R may join together to form a ring, the ring being optionally substituted by halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 haloalkoxy or nitro; and R , R and R are independently hydrogen or C1-4 alkyl; provided that at least one of R and R is hydrogen.

    Abstract translation: 式（I）的化合物，其中A 1和A 2独立地是苯基，呋喃基或噻吩基，其各自任选被卤素，C 1-4烷基，C 1-4烷氧基，C 1-4烷硫基，C 1-4 卤代烷基，C 1-4卤代烷氧基或C 1-4卤代烷硫基; R为C1-4烷基，C1-4卤代烷基，C2-4烯基，C2-4卤代烯基，C3-7环烷基，C3-7环烷基（C1-4）烷基，苄基或苯基，其中苄基和苯基任选被 卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基; 且R 1，R 2，R 3和R 4分别独立地为氢，C 1-8烷基，C 1-8卤代烷基，C 1-8烷氧基，C 1-8卤代烷氧基，卤素，硝基， COR 7，NR 5 R 6，苄基或苯基（其中苄基和苯基任选被卤素取代，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基或NR 5> - [R <6>）; R 1和R 2或R 2和R 3可以连接在一起形成环，该环任选被卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基， C 1-4卤代烷氧基或硝基; 和R 5，R 6和R 7独立地是氢或C 1-4烷基; 条件是R 1和R 4中的至少一个是氢。

Patent Agency Ranking