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公开(公告)号:WO2009129370A1
公开(公告)日:2009-10-22
申请号:PCT/US2009/040771
申请日:2009-04-16
Applicant: GLAXO GROUP LIMITED , DENG, Jianghe , LAINE, Dramane, Ibrahim , MCCLELAND, Brent, W. , PALOVICH, Michael, R. , PETITJEAN, Emile, Veronique
Inventor: DENG, Jianghe , LAINE, Dramane, Ibrahim , MCCLELAND, Brent, W. , PALOVICH, Michael, R. , PETITJEAN, Emile, Veronique
CPC classification number: C07D207/14 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14
Abstract: What is disclosed herein are compounds of the following formula (I); or a salt thereof wherein Ar is a monocyclic heteroaromatic ring, a bicyclic heteroaromatic ring or a bicyclic heterocycloalkylaromatic ring.
Abstract translation: 本文公开的是下式(I)的化合物; 或其盐,其中Ar是单环杂芳环,双环杂芳环或双环杂环烷基芳族环。
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公开(公告)号:WO2006062931A3
公开(公告)日:2007-04-19
申请号:PCT/US2005044033
申请日:2005-12-05
Applicant: SMITHKLINE BEECHAM CORP , LAINE DRAMANE IBRAHIM , PALOVICH MICHAEL R
Inventor: LAINE DRAMANE IBRAHIM , PALOVICH MICHAEL R
IPC: A61K31/56 , A61K9/72 , A61K31/439 , A61K31/46
CPC classification number: A61K31/7072
Abstract: Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
Abstract translation: 毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2006055503A3
公开(公告)日:2006-08-03
申请号:PCT/US2005041230
申请日:2005-11-15
Applicant: GLAXO GROUP LTD , BUDZIK BRIAN W , JIN JIAN , LAINE DRAMANE I , PALOVICH MICHAEL R , RIVERO RALPH A , WANG YONGHUI , XIE HAIBO
Inventor: BUDZIK BRIAN W , JIN JIAN , LAINE DRAMANE I , PALOVICH MICHAEL R , RIVERO RALPH A , WANG YONGHUI , XIE HAIBO
IPC: A61K31/496 , C07D401/12 , C07D403/12
CPC classification number: C07D487/08 , C07D295/155 , C07D295/185 , C07D401/12 , C07D403/12 , C07D471/10 , C07D487/10
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
Abstract translation: 提供了毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2006062931A2
公开(公告)日:2006-06-15
申请号:PCT/US2005/044033
申请日:2005-12-05
Inventor: LAINE, Dramane, Ibrahim , PALOVICH, Michael, R.
IPC: A61K31/7072
CPC classification number: A61K31/7072
Abstract: Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
Abstract translation: 提供了毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。 p>
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公开(公告)号:WO2006043950A1
公开(公告)日:2006-04-27
申请号:PCT/US2004/034536
申请日:2004-10-20
Applicant: SMITHKLINE BEECHAM CORPORATION , BUSCH-PETERSEN, Jakob , PALOVICH, Michael, R. , WIDDOWSON, Katherine, L.
IPC: A61K31/54
CPC classification number: C07D295/26 , C07C311/47 , C07C317/28 , C07C323/49 , C07C2601/02 , C07D211/28 , C07D307/14
Abstract: This invention relates to novel compounds of Formula (I) to (VII), and compositions thereof, useful in the treatment of disease states mediated by the chemokine, Interleukin-8 (IL-8).
Abstract translation: 本发明涉及式(I)至(VII)的新化合物及其组合物,其可用于治疗由趋化因子介导的疾病状态,白细胞介素-8(IL-8)。
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公开(公告)号:WO2006017768A2
公开(公告)日:2006-02-16
申请号:PCT/US2005027958
申请日:2005-08-05
Applicant: GLAXO GROUP LTD , BUSCH-PETERSEN JAKOB , DAVIS RODERICK S , LAINE DRAMANE IBRAHIM , NEIPP CHRISTOPHER E , PALOVICH MICHAEL R
Inventor: BUSCH-PETERSEN JAKOB , DAVIS RODERICK S , LAINE DRAMANE IBRAHIM , NEIPP CHRISTOPHER E , PALOVICH MICHAEL R
IPC: A61K31/4745
CPC classification number: C07D451/14
Abstract: Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
Abstract translation: 毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2005046586A8
公开(公告)日:2005-09-01
申请号:PCT/US2004036663
申请日:2004-11-04
Applicant: GLAXO GROUP LTD , WAN ZEHONG , YAN HONGXING , PALOVICH MICHAEL R , LAINE DRAMANE I
Inventor: WAN ZEHONG , YAN HONGXING , PALOVICH MICHAEL R , LAINE DRAMANE I
IPC: A61K20060101 , A61K31/46 , C07D451/02
CPC classification number: C07D451/02
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
Abstract translation: 提供毒蕈碱性乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2005046586A3
公开(公告)日:2005-05-26
申请号:PCT/US2004/036663
申请日:2004-11-04
Applicant: GLAXO GROUP LIMITED , WAN, Zehong , YAN, Hongxing , PALOVICH, Michael, R. , LAINE, Dramane, I. , LEE, Dennis , STAVENGER, Robert, A. , GOODMAN, Krista, B. , HILFIKER, Mark, A. , CUI, Haifeng , VIET, Andrew, W. , MARINO, Joseph, P.
Inventor: WAN, Zehong , YAN, Hongxing , PALOVICH, Michael, R. , LAINE, Dramane, I. , LEE, Dennis , STAVENGER, Robert, A. , GOODMAN, Krista, B. , HILFIKER, Mark, A. , CUI, Haifeng , VIET, Andrew, W. , MARINO, Joseph, P.
IPC: A61K31/46
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
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公开(公告)号:WO2002079122A2
公开(公告)日:2002-10-10
申请号:PCT/US2002/010038
申请日:2002-03-27
Inventor: PALOVICH, Michael, R. , WIDDOWSON, Katherine, L.
IPC: C07C
CPC classification number: C07C311/47 , C07C311/43 , C07C319/02 , C07C2601/04 , C07C323/20
Abstract: Methods of synthesizing phenol-containing compounds are disclosed.
Abstract translation: 公开了合成含酚化合物的方法。 p>
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公开(公告)号:WO2007016639A3
公开(公告)日:2007-07-05
申请号:PCT/US2006030153
申请日:2006-08-02
Applicant: GLAXO GROUP LTD , BUSCH-PETERSEN JAKOB , LAINE DRAMANE IBRAHIM , PALOVICH MICHAEL R , DAVIS RODERICK S , FU WEI , XIE HAIBO
Inventor: BUSCH-PETERSEN JAKOB , LAINE DRAMANE IBRAHIM , PALOVICH MICHAEL R , DAVIS RODERICK S , FU WEI , XIE HAIBO
IPC: A61K31/46 , C07D451/02
CPC classification number: C07D451/02
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
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