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公开(公告)号:WO2005104745A3
公开(公告)日:2006-08-03
申请号:PCT/US2005014386
申请日:2005-04-27
Applicant: GLAXO GROUP LTD , LAINE DRAMANE I , PALOVICH MICHAEL R , MCCLELAND BRENT W , NEIPP CHRISTOPHER E , THOMAS SONIA M
Inventor: LAINE DRAMANE I , PALOVICH MICHAEL R , MCCLELAND BRENT W , NEIPP CHRISTOPHER E , THOMAS SONIA M
IPC: A61K31/44 , C07D453/02
CPC classification number: C07D453/02 , A61K31/439
Abstract: Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
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2.
公开(公告)号:WO2006065788A2
公开(公告)日:2006-06-22
申请号:PCT/US2005/045012
申请日:2005-12-13
Applicant: GLAXO GROUP LIMITED , BUSCH-PETERSEN, Jakob , DAVIS, Roderick, S. , FU, Wei , JIN, Jian , LAINE, Dramane, I. , PALOVICH, Michael, R.
Inventor: BUSCH-PETERSEN, Jakob , DAVIS, Roderick, S. , FU, Wei , JIN, Jian , LAINE, Dramane, I. , PALOVICH, Michael, R.
IPC: A61K31/44
CPC classification number: C07D513/04
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
Abstract translation: 提供毒蕈碱性乙酰胆碱受体拮抗剂及其使用方法。
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3.QUATERNARY AMMONIUM SALTS OF FUSED HETEAROMATIC AMINES AS NOVEL MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS 审中-公开
Title translation: 作为新型麦芽糖乙酰胆碱受体拮抗剂的融合的蜂窝状氨基酸的季铵盐公开(公告)号:WO2006065755A2
公开(公告)日:2006-06-22
申请号:PCT/US2005/044951
申请日:2005-12-13
Applicant: GLAXO GROUP LIMITED , BUSCH-PETERSEN, Jakob , DAVIS, Roderick, S. , FU, Wei , JIN, Jian , LAINE, Dramane, I. , PALOVICH, Michael, R.
Inventor: BUSCH-PETERSEN, Jakob , DAVIS, Roderick, S. , FU, Wei , JIN, Jian , LAINE, Dramane, I. , PALOVICH, Michael, R.
IPC: A61K31/4747 , A61K31/47
CPC classification number: C07D471/04 , C07D513/04
Abstract: Novel derivatives of cyclic amines, pharmaceutical compositions, processes for their preparation, and use thereof in treating muscarinic acetylcholine receptor mediated diseases are provided.
Abstract translation: 提供环胺的新型衍生物,药物组合物,其制备方法及其在治疗毒蕈碱性乙酰胆碱受体介导的疾病中的用途。
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4.MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS FIELD OF THE INVENTION 审中-公开
Title translation: 麦角胺乙酰胆碱受体拮抗剂技术领域本发明涉及麦角胺乙酰胆碱受体拮抗剂公开(公告)号:WO2005112644A2
公开(公告)日:2005-12-01
申请号:PCT/US2005016148
申请日:2005-05-10
Applicant: GLAXO GROUP LTD , LAINE DRAMANE I , MCCLELAND BRENT W , NEIPP CHRISTOPHER E , PALOVICH MICHAEL R
Inventor: LAINE DRAMANE I , MCCLELAND BRENT W , NEIPP CHRISTOPHER E , PALOVICH MICHAEL R
IPC: A01N43/90 , C07D453/02
CPC classification number: C07D453/02
Abstract: Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
Abstract translation: 毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2005094835A1
公开(公告)日:2005-10-13
申请号:PCT/US2004/008032
申请日:2004-03-17
Applicant: GLAXO GROUP LIMITED , BUSCH-PETERSEN, Jakob , LAINE, Dramane, I. , PALOVICH, Michael, R.
Inventor: BUSCH-PETERSEN, Jakob , LAINE, Dramane, I. , PALOVICH, Michael, R.
IPC: A61K31/55
CPC classification number: C07D409/12 , C07D223/16 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/04 , C07D413/12 , C07D413/14 , C07D471/04
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
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6.
公开(公告)号:WO2004091482A3
公开(公告)日:2004-12-23
申请号:PCT/US2004010641
申请日:2004-04-07
Applicant: GLAXO GROUP LTD , BUSCH-PETERSEN JAKOB , LAINE DRAMANE I , PALOVICH MICHAEL R , MCCLELAND BRENT W
Inventor: BUSCH-PETERSEN JAKOB , LAINE DRAMANE I , PALOVICH MICHAEL R , MCCLELAND BRENT W
IPC: A61K20060101 , A61K31/403 , C07D209/58 , C07D519/00
CPC classification number: C07D519/00 , C07D487/08
Abstract: Novel thiazole aniline compounds, pharmaceutical compositions, methods of making them and used therof in treating M3 muscarinic acetylcholine receptor mediated diseases are disclosed
Abstract translation: 公开了新的噻唑苯胺化合物,药物组合物及其制备方法并用于治疗M3毒蕈碱乙酰胆碱受体介导的疾病
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7.M3MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS 审中-公开
Title translation: M3MUSCARINIC ACETYLCHOLINE受体拮抗剂公开(公告)号:WO2004012684A2
公开(公告)日:2004-02-12
申请号:PCT/US2003/024569
申请日:2003-08-06
Applicant: GLAXO GROUP LIMITED , LAINE, Dramane, I. , BELL, Ricahrd , BUSCH-PETERSEN, Jakob , PALOVICH, Michael
Inventor: LAINE, Dramane, I. , BELL, Ricahrd , BUSCH-PETERSEN, Jakob , PALOVICH, Michael
IPC: A61K
CPC classification number: C07D513/04 , C07D417/12
Abstract: M 3 Muscarinic Acetylcholine Receptor Antagonists and methods of using them are provided.
Abstract translation: 提供了M 3蕈毒碱乙酰胆碱受体拮抗剂及其使用方法。 p>
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8.
公开(公告)号:WO2006055503A3
公开(公告)日:2006-08-03
申请号:PCT/US2005041230
申请日:2005-11-15
Applicant: GLAXO GROUP LTD , BUDZIK BRIAN W , JIN JIAN , LAINE DRAMANE I , PALOVICH MICHAEL R , RIVERO RALPH A , WANG YONGHUI , XIE HAIBO
Inventor: BUDZIK BRIAN W , JIN JIAN , LAINE DRAMANE I , PALOVICH MICHAEL R , RIVERO RALPH A , WANG YONGHUI , XIE HAIBO
IPC: A61K31/496 , C07D401/12 , C07D403/12
CPC classification number: C07D487/08 , C07D295/155 , C07D295/185 , C07D401/12 , C07D403/12 , C07D471/10 , C07D487/10
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
Abstract translation: 提供了毒蕈碱乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2005046586A8
公开(公告)日:2005-09-01
申请号:PCT/US2004036663
申请日:2004-11-04
Applicant: GLAXO GROUP LTD , WAN ZEHONG , YAN HONGXING , PALOVICH MICHAEL R , LAINE DRAMANE I
Inventor: WAN ZEHONG , YAN HONGXING , PALOVICH MICHAEL R , LAINE DRAMANE I
IPC: A61K20060101 , A61K31/46 , C07D451/02
CPC classification number: C07D451/02
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
Abstract translation: 提供毒蕈碱性乙酰胆碱受体拮抗剂及其使用方法。
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公开(公告)号:WO2005046586A3
公开(公告)日:2005-05-26
申请号:PCT/US2004/036663
申请日:2004-11-04
Applicant: GLAXO GROUP LIMITED , WAN, Zehong , YAN, Hongxing , PALOVICH, Michael, R. , LAINE, Dramane, I. , LEE, Dennis , STAVENGER, Robert, A. , GOODMAN, Krista, B. , HILFIKER, Mark, A. , CUI, Haifeng , VIET, Andrew, W. , MARINO, Joseph, P.
Inventor: WAN, Zehong , YAN, Hongxing , PALOVICH, Michael, R. , LAINE, Dramane, I. , LEE, Dennis , STAVENGER, Robert, A. , GOODMAN, Krista, B. , HILFIKER, Mark, A. , CUI, Haifeng , VIET, Andrew, W. , MARINO, Joseph, P.
IPC: A61K31/46
Abstract: Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
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