摘要:
Compounds I ##STR1## where A equals t-butyl or a large number of (substituted) aromatics; Y equals azolyl; or Y equals --X--R.sup.1 where X=oxygen or sulfur and R.sup.1 equals (cyclo)alkyl or (heterocyclic) aryl; or Y equals ##STR2## where R.sup.2 equals (cyclo)alkyl, acetyl or aryl; or Y equals --NR.sup.3 R.sup.4 where R.sup.3 /R.sup.4 is alkyl; or Y equals several nitrogen-containing heterocyclic rings; Z equals OH, alkylcarbonyloxy, hal, alkoxy or benzyloxy; and the salts thereof are effective antimycotics or fungicides.They are obtained by reaction of II ##STR3## with (CH.sub.3).sub.2 ##STR4## and further reaction of the compound IV ##STR5## obtained from this with a nucleophile YM (M=hydrogen or a metal equivalent).The compounds I (where Z=OH) resulting from this can be acylated or alkylated, or converted into I where Z=hal.
摘要:
Compounds I ##STR1## where A equals t-butyl, phenyl, biphenylyl, phenoxyphenyl, benzylphenyl, benzyloxyphenyl, phenylthiophenyl, phenylsulfinylphenyl, phenylsulfonylphenyl, naphthyl, 1,2,3,4-tetrahydronaphthyl, indanyl, fluorenyl, thienyl, furyl, pyridyl, isoxazolyl, pyrazolyl, benzofuryl or benzothienyl,Z equals CO, CH.sub.2 or radicals of ketone derivatives;Y equals azole or equals --X--R.sup.8 (R.sup.8 =(cyclo)alkyl or an aromatic) or equals a number of amine derivatives or equal acyl,are antimycotics. The preparation and use as medicaments are described.
摘要:
1-(1,3-Dioxolan-2-ylmethyl)-azoles of the general formula ##STR1## and their stereoisomers and their salts with physiologically acceptable acids, the preparation of these compounds, pharmaceutical formulations containing the latter and their use against mycoses, protozoa and Gram-positive and Gram-negative bacteria are described.
摘要:
New 1-(1,3-dioxolan-2-ylmethyl)azoles, their stereoisomers and their salts are described, as are processes for their preparation. The new compounds are chemotherapeutic agents. They are active against skin fungi, mold fungi and yeasts and against bacteria.
摘要:
The system for holding a number of in-line two wheeled vehicles has a vertical support column. A lifting bracket has an end that engages a vertical channel of the vertical support. A counter balance system in the vertical support column is connected to the lifting bracket. A horizontal track runs perpendicular to a face of the vertical support column with the vertical channel. A horizontal bracket engages the horizontal track. A bike or other two wheel vehicle is held by the lifting bracket. Because the lifting bracket has a counter balance system a person can easily lift the bike up in the air. The horizontal bracket can also hold a bike. A bike on the horizontal bracket can be slid so that it is under the lifting bracket, which may be holding a second bike.
摘要:
The preparation of (optionally substituted) 2-mercaptobenzothiazole by reaction of corresponding 2-halogenoanilines with an alkali metal xanthate or alkaline earth metal xanthate or with CS.sub.2 in the presence of bases.
摘要:
The system for holding a number of in-line two wheeled vehicles has a vertical support column. A lifting bracket has an end that engages a vertical channel of the vertical support. A counter balance system in the vertical support column is connected to the lifting bracket. A horizontal track runs perpendicular to a face of the vertical support column with the vertical channel. A horizontal bracket engages the horizontal track. A bike or other two wheel vehicle is held by the lifting bracket. Because the lifting bracket has a counter balance system a person can easily lift the bike up in the air. The horizontal bracket can also hold a bike. A bike on the horizontal bracket can be slid so that it is under the lifting bracket, which may be holding a second bike.
摘要:
A multiple-level bicycle storing system includes a framework with a vertical support and a mounting frame defining upper and lower storing spaces. Each storing space includes a receiver to hold a bicycle. The upper receiver has a distal end, a proximal end and a U-shaped channel along the top surface. The upper receiver is pivotally attached to the mounting frame, enabling the upper receiver to tilt from horizontal to a loading and unloading position. The proximal end of the upper receiver is located near the floor when pivoted into the loading and unloading position. The upper receiver pivots up from the loading and unloading position into the horizontal storage position. The bicycles and the storing spaces are enclosed, and a floor separates the lower storing space from the upper storing space. Each storing space includes a lockable door and conceals the pivot point, upper receiver and bicycles inside the enclosure.
摘要:
A multiple-level bicycle storing system includes a framework having a vertical support and a horizontal mounting frame. The framework defines a lower storing space with a lower receiver, a middle storing space with an upper receiver attached to the mounting frame with a pivot mechanism, and an upper storing space. The upper storing space includes an upper track having a horizontal rail, a shuttle movably engaging the rail, an electric shuttle motor attached to the rail and the shuttle and a power source, a cable winch incorporated into the shuttle, an electric winch motor attached to the cable winch and the power source, a control box attached between the winch motor, the shuttle motor and the power source, and a bicycle support attached to the cable winch. The pivot mechanism includes a pluraility of rollers, rails, a lever and a gas spring to enable extension of the upper receiver.
摘要:
A multiple-level bicycle storing system includes a framework having a vertical support and a horizontal mounting frame. The framework defines a lower storing space with a lower receiver, a middle storing space with an upper receiver attached to the mounting frame with a pivot mechanism, and an upper storing space. The upper storing space includes an upper track having a horizontal rail, a shuttle movably engaging the rail, an electric shuttle motor attached to the rail and the shuttle and a power source, a cable winch incorporated into the shuttle, an electric winch motor attached to the cable winch and the power source, a control box attached between the winch motor, the shuttle motor and the power source, and a bicycle support attached to the cable winch. The pivot mechanism includes a plurality of rollers, rails, a lever and a gas spring to enable extension of the upper receiver.