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36 条记录 (耗时 0.009 秒)

    Diaminocycloalkanes
    1.
    发明授权
    Diaminocycloalkanes 失效
    DIAMINOCYCLOALKANES

    公开(公告)号：US3652559A

    公开(公告)日：1972-03-28

    申请号：US3652559D

    申请日：1968-05-13

    申请人： UPJOHN CO

    发明人： SZMUSZKOVICZ JACOB

    IPC分类号： C07D295/02 ,  C07D87/38

    CPC分类号： C07D295/02 ,  Y10S514/866 ,  Y10S514/869 ,  Y10S514/91

    摘要： CIS- AND TRANS-DIAMINOCYCLOALKANES ACID ADDITION AND QUATERNARY AMMONIUM SALTS THEREOF. THE NOVEL COMPOUNDS ARE USEFUL AS TERTIARY AMINES AND CATALYSTS. IN ADDITION, MANY OF THE 1,2- AND 1,3-DIAMINOCYCLOALKANES EXHIBIT ACTIVITY AS CENTRAL NERVOUS SYSTEM STIMULANTS, DIURETICS, ANOREXIGENIC AND ANTIDIABETIC AGENTS.

    3 5-disubstituted 1 2 4-oxadiazoles
    2.
    发明授权
    3 5-disubstituted 1 2 4-oxadiazoles 失效
    3 5 - 发现1 2 4-氧化氮

    公开(公告)号：US3651054A

    公开(公告)日：1972-03-21

    申请号：US3651054D

    申请日：1967-01-31

    申请人： ABBOTT LAB

    发明人： CROVETTI ALDO JOSEPH ,  ESCH ANNE MARY VON

    IPC分类号： C07D413/04 ,  C07D417/14 ,  C07D487/18 ,  C07D85/52 ,  C07D87/38

    CPC分类号： C07D413/04 ,  C07D417/14

    摘要： COMPOUNDS COMPRISING 3,5-DISUBSTITUTED-1,2,4-OXADIAZOLES WITH ONE OF THE SUBSTITUENTS BEING 5-NITRO-2-FURYL. THE COMPOUNDS ARE USEFUL AS ANTIBACTERIAL, ANTHELMINTIC, AND ANTI-TRICHOMONAS AGENTS.

    摘要翻译： 新的抗微生物剂，其中R1包括卤代苯基，低级烷基，苯基，硝基苯基，二硝基苯基，硝基呋喃基和硝基噻吩基; R2包括氢和低级烷基; Nhet包括通过其氮键合的杂环部分，该杂环部分足够碱性以形成季铵盐。

    Substituted n aminoalkyl arylamino imidazolines-(2)
    6.
    发明授权
    Substituted n aminoalkyl arylamino imidazolines-(2) 失效
    取代的氨基亚氨基亚氨基咪唑啉酮（2）

    公开(公告)号：US3752810A

    公开(公告)日：1973-08-14

    申请号：US3752810D

    申请日：1970-11-16

    申请人： BOEHRINGER SOHN INGELHEIM

    发明人： STAEHLE H ,  KOEPPE H ,  KUMMER W ,  SAMTLEBEN H

    IPC分类号： C07D233/50 ,  C07D295/13 ,  C07D87/38 ,  C07D87/40

    CPC分类号： C07D295/13 ,  C07D233/50

    摘要： NOVEL COMPOUNDS SELECTED FROM THE GROUP CONSISTING OF N-AMINOALKYL-ARYLAMINO-IMIDAZOLINES-(2) OF THE FORMULA

    1-R5,2-((R1,R2,R3-PHENYL)-N(-R4)-)-2-IMIDAZOLINE

    WHEREIN R1, R2 AND R3 MAY BE THE SAME OR DIFFERENT AND ARE SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, FLUORINE, CHLORINE, BROMINE, TRIFLUOROMETHYL, CYANO AND LOWER ALKYL AND LOWER ALKOXY OF 1 TO 7 CARBON ATOMS AND ONE OF 54 AND R5 BEING HYDROGEN WITH THE OTHER BEING -(CH2)N-A, N IS 2 OR 3 AND A IS SELECTED FROM THE GROUP CONSISTING OF DIALKYLAMINO WITH 1 TO 4 CARBON ATOMS IN EACH ALKYL, MORPHOLINO, PYRROLIDINO AND PIPERIDINO AND THEIR NON-TOXIC, PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS HAVING HYPOTENSIVE ACTIVITY, THEIR PREPARATION AND THEIR USE.

    2,4,6-trisubstituted derivatives of pyrimidine
    7.
    发明授权
    2,4,6-trisubstituted derivatives of pyrimidine 失效
    吡啶的2,4,6-取代衍生物

    公开(公告)号：US3624084A

    公开(公告)日：1971-11-30

    申请号：US3624084D

    申请日：1968-01-22

    申请人： UCB SA

    发明人： MATHIEU JACQUES

    IPC分类号： A61K31/505 ,  C07D239/28 ,  C07D239/42 ,  C07D239/48 ,  C07D51/42 ,  C07D87/38

    CPC分类号： C07D239/48 ,  A61K31/505 ,  C07D239/28 ,  C07D239/42 ,  Y10S514/869 ,  Y10S514/929

    摘要： IN WHICH R1 is hydrogen, lower alkyl, aralkyl, R2 is hydrogen, halogen, lower alkyl, hydroxyalkylamino, omegaaryl-omega-hydroxyalkylamino, morpholino, R3 is hydrogen, lower alkyl eventually hydroxyl-substituted, aralkyl, R4 is lower alkyl substituted by at least one hydroxyl group separated from N by at least two carbon atoms, or R3 and R4 together with the extranuclear N are morpholino, as well as their salts with inorganic or organic acids. These compounds are hypotensives, peripheral and coronary vasodilators, diuretics, bronchodilators, spasmolytics and circulatory and respiratory analeptics.

    New 2,4,6-trisubstituted pyrimidine derivatives of the general formula

    Formamidine compounds of diphenyl-sulfone
    8.
    发明授权
    Formamidine compounds of diphenyl-sulfone 失效
    二苯基砜的甲醛化合物

    公开(公告)号：US3621013A

    公开(公告)日：1971-11-16

    申请号：US3621013D

    申请日：1969-03-28

    申请人： HOECHST AG

    发明人： WINKELMANN ERHARDT ,  RAETHER WOLFGANG

    IPC分类号： C07D295/195 ,  C07D87/38

    CPC分类号： C07D295/195

    摘要： Formamidine derivatives of diphenyl-sulfone which are effective medicaments against malaria are prepared by reacting 4,4'' diamino-diphenyl-sulfone of the formula

    WITH N-formyl compounds of the formula

    IN WHICH -N Z is a pyrrolidino, piperidino or morpholino radical, in the presence of acid halides and, if desired, converting the salts thus obtained into the free bases.