Substituted imidazolinylpyrimidines
    91.
    发明授权
    Substituted imidazolinylpyrimidines 失效
    取代的咪唑啉基嘧啶

    公开(公告)号:US5244865A

    公开(公告)日:1993-09-14

    申请号:US891493

    申请日:1992-05-29

    摘要: Herbicidal new substituted imidazolinylpyrimidines of the general formula (I) ##STR1## in which R.sup.1 represents hydrogen, halogen, cyano, nitro or thiocyanato, or represents a hydroxyl, mercapto, amino, carbonyl, sulphinyl, sulphonyl, alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aryl or heterocyclyl radical, each of which is optionally substituted,R.sup.2 represents hydrogen, hydroxyl, halogen, alkyl or halogenoalkyl,R.sup.3 represents hydrogen, or represents alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aryl or heterocyclyl, each of which is optionally substituted, or represents an equivalent of an inorganic or organic cation,R.sup.4 and R.sup.5 independently of each other in each case represent hydrogen, alkyl, halogenoalkyl or cycloalkyl andX represents oxygen or sulphur.

    摘要翻译: 通式(I)的除草新的取代的咪唑啉基嘧啶其中R 1表示氢,卤素,氰基,硝基或氰硫基,或表示羟基,巯基,氨基,羰基,亚磺酰基,磺酰基,烷基,烯基, 炔基,环烷基,环烯基,芳基或杂环基,其各自任选被取代,R 2表示氢,羟基,卤素,烷基或卤代烷基,R 3表示氢,或表示烷基,烯基,炔基,环烷基,环烯基,芳基或杂环基, 各自任选被取代,或表示无机或有机阳离子的当量,R 4和R 5彼此独立地表示氢,烷基,卤代烷基或环烷基,X表示氧或硫。

    Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives
    93.
    发明授权
    Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives 失效
    除草剂4-烷氧基 - 和4-(取代的)氨基 - 吡咯烷酮衍生物

    公开(公告)号:US5191089A

    公开(公告)日:1993-03-02

    申请号:US565536

    申请日:1990-08-09

    CPC分类号: A01N43/36 C07D207/38

    摘要: Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives of the formula ##STR1## in which X and Y independently of one another represent hydrogen, halogen, alkyl, alkoxy, halogenoalkyl or in each case unsubstituted or substituted aryloxy or arylthio,Z represents halogen, alkyl or alkoxy,n represents the number 0, 1, 2 or 3,A represents in each case unsubstituted or in each case halogen-substituted alkyl, alkenyl, alkynyl, alkoxyalkyl, polyalkoxyalkyl or alkylthioalkyl, cycloalkyl which is optionally interrupted by hetero atoms, arylalkyl which is unsubstituted or substituted by halogen, alkyl, halogenoalkyl, alkoxy and/or nitro, unsubstituted aryl or aryl substituted by a member selected from the group consisting of halogen, alkyl, alkoxy, halogenoalkyl, halogenoalkoxy and phenoxy or phenylthio which are in each case unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl and/or halogenoalkoxy,B represents hydroxyl, alkoxy, halogenoalkoxy or cycloalkoxy, the cycloalkyl radical being unsubstituted or substituted by halogen and/or alkyl, orB represents the group ##STR2## wherein C and D independently of one another represent hydrogen, alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl or polyalkoxyalkyl, cycloalkyl which is optionally interrupted by hetero atoms or in each case unsubstituted or substituted phenyl, phenylalkyl, phenoxyalkyl, hetaryl or hetarylalkyl, orC and D together with the nitrogen atom to which they are bonded, form a 3- to 9-membered, optionally substituted ring which is optionally interrupted by the further hetero atoms,with the proviso that at least one radical X, Y or Z does not represent chlorine or methyl if B represents hydroxyl and A has a meaning other than optionally substituted aryl.

    摘要翻译: 式(I)的除草4-烷氧基 - 和4-(取代的)氨基 - 芳基吡咯烷酮衍生物,其中X和Y彼此独立地代表氢,卤素,烷基,烷氧基,卤代烷基或在各种情况下是未取代或取代的 芳氧基或芳硫基,Z表示卤素,烷基或烷氧基,n表示数0,1,2或3,A表示各自为未取代的或在各种情况下为卤素取代的烷基,烯基,炔基,烷氧基烷基,聚烷氧基烷基或烷硫基烷基,环烷基 烷基,卤代烷基,烷氧基和/或硝基,未经取代的芳基或被选自卤素,烷基,烷氧基,卤代烷基,卤代烷氧基的成员所取代的芳基, 苯氧基或苯硫基,其各自为未被取代或被卤素,烷基,烷氧基,卤代烷基和/或卤代烷氧基取代,B代表羟基,烷氧基,卤代烷氧基或环 烷氧基,环烷基是未取代的或被卤素和/或烷基取代,或B表示基团,其中C和D彼此独立地表示氢,烷基,烯基,烷氧基烷基,烷硫基烷基或聚烷氧基烷基,任选地中断的环烷基 通过杂原子或在每种情况下未取代或取代的苯基,苯基烷基,苯氧基烷基,杂芳基或杂芳基烷基,或C和D与它们所键合的氮原子一起形成3至9元任选取代的环,其任选地 被另外的杂原子中断,条件是至少一个基团X,Y或Z不表示氯或甲基,如果B表示羟基,并且A具有除任选取代的芳基以外的含义。

    Herbicidal pyrazolin-5-one derivatives, compositions and use
    94.
    发明授权
    Herbicidal pyrazolin-5-one derivatives, compositions and use 失效
    除草剂吡唑啉-5-酮衍生物,组合物和用途

    公开(公告)号:US5174808A

    公开(公告)日:1992-12-29

    申请号:US610597

    申请日:1990-11-08

    摘要: Herbicidal pyrazolin-5-one derivatives of the formula ##STR1## in which R.sup.1 represents alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkynyl, alkenyl or alkynyl substituted by optionally substituted phenyl, halogenoalkenyl, alkoxy, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsulphinylalkyl, alkoxycarbonylalkyl, in each case optionally substituted aryl, aralkyl, aryloxyalkyl or arylthioalkyl, an optionally substituted heterocycle, heterocyclylalkyl or the --NH--CO--R.sup.3 or --CO--O--R.sup.4 groups, in which R.sup.3 and R.sup.4 in each case independently of one another represent alkyl or aryl,R.sup.2 represents hydrogen, alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkinyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsuslphinylalkyl or alkoxycarbonylalkyl andAr represents optionally substituted aryl or a heterocycle which is optionally substituted and optionally fused,excluding the compounds 1-(3-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazoline-5-one, 1-(4-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one, 1-(4-trifluoronethylphenyl-3-methylthiomethyl-4-(N-hydroxyaminomethylidene))-pyrazolin-5-one and 1-(4-n-nitrophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one.

    摘要翻译: 式(Ⅰ)的除草吡唑啉-5-酮衍生物,其中R 1表示被任选取代的苯基,卤代烯基,烷氧基,烷氧基烷基,烷基硫代烷基,烷基磺酰基烷基,烷基亚磺酰基烷基,烷基磺酰基烷基, 烷氧基羰基烷基,在各种情况下均为任选取代的芳基,芳烷基,芳氧基烷基或芳硫基烷基,任选取代的杂环,杂环基烷基或-NH-CO-R 3或-CO-O-R 4基团,其中R 3和R 4各自独立地为 另一个代表烷基或芳基,R 2表示氢,烷基,环烷基,卤代烷基,烯基,炔基,卤代烯基,烷氧基烷基,烷基硫代烷基,烷基磺酰基烷基,烷基磺酰基烷基或烷氧基羰基烷基,Ar表示任选取代的芳基或任选被取代和任选稠合的杂环, 化合物1-(3-氯苯基)-3-甲硫基甲基-4-(N-羟基氨基亚甲基) - 吡唑并-5-酮, 1-(4-氯苯基)-3-甲基硫代甲基-4-(N-羟基氨基亚甲基) - 吡唑啉-5-酮,1-(4-三氟甲基苯基-3-甲硫基甲基-4-(N-羟基氨基甲基二烯) 5-(1-硝基苯基)-3-甲基硫代甲基-4-(N-羟基氨基亚甲基) - 对]吡唑-5-酮。

    Herbicidal sulphonylaminocarbonyltriazolinones having substituents
bonded via oxygen of the formula
    98.
    发明授权
    Herbicidal sulphonylaminocarbonyltriazolinones having substituents bonded via oxygen of the formula 失效
    具有通过下式的氧连接的取代基的除草磺酰基氨基羰基三唑啉酮

    公开(公告)号:US5869681A

    公开(公告)日:1999-02-09

    申请号:US881269

    申请日:1997-06-24

    摘要: Herbicidal sulphonylaminocarbonyltriazolinones having substituents bonded via oxygen of the formula ##STR1## in which R.sup.1 represents hydrogen, amino, or an optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl, aryl, alkylamino, cycloalkylamino or dialkylamino radical,R.sup.2 represents an optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aralkyl or aryl radical, andR.sup.3 represents an optionally substituted alkyl, aralkyl, aryl or heteroaryl radical,and salts thereof, with the exception of the compounds:2-(2-methoxycarbonyl-phenylsulphonylaminocarbonyl)-4-methyl-5-methoxy-2,4-dihydro-3H-1,2,4-triazol-3-one,2-(2-trifluoromethoxy-phenylsulphonylaminocarbonyl)-4-cyclopropyl-5-methoxy-2,4-dihydro-3H-1,2,4-triazol-3-one,2-(2-difluoromethoxy-phenylsulphonylaminocarbonyl)-4-cyclobutyl-5-ethoxy-2,4-dihydro-3H-1,2,4-triazol-3-one, and2-(2-methoxycarbonyl-phenylsulphonylaminocarbonyl)-4-ethyl-5-ethoxy-2,4-dihydro-3H-1,2,4-triazol-3-one.

    摘要翻译: 具有通过式氨基氧的取代基键合的除草磺酰基氨基羰基三唑啉酮或任选取代的烷基,烯基,炔基,环烷基,芳烷基,芳基,烷基氨基,环烷基氨基或二烷基氨基,R2表示任选取代的烷基,烯基,炔基,环烷基,环烯基, 芳基或芳基,R 3表示任选取代的烷基,芳烷基,芳基或杂芳基及其盐,除了化合物:2-(2-甲氧基羰基 - 苯基磺酰基氨基羰基)-4-甲基-5-甲氧基-2 ,4-二氢-3H-1,2,4-三唑-3-酮,2-(2-三氟甲氧基 - 苯基磺酰氨基羰基)-4-环丙基-5-甲氧基-2,4-二氢-3H-1,2,4 - 三唑-3-酮,2-(2-二氟甲氧基 - 苯基磺酰基氨基羰基)-4-环丁基-5-乙氧基-2,4-二氢-3H-1,2,4-三唑-3-酮和2-(2 - 甲氧基羰基 - 苯基磺酰基氨基羰基)-4-乙基-5-乙氧基-2,4-二氢-3H-1,2,4-三唑-3-酮。

    Substituted 1-H-3-aryl-pyrrolidine-2,4-dione derivatives
    100.
    发明授权
    Substituted 1-H-3-aryl-pyrrolidine-2,4-dione derivatives 失效
    取代的1-H-3-芳基 - 吡咯烷-2,4-二酮衍生物

    公开(公告)号:US5462913A

    公开(公告)日:1995-10-31

    申请号:US140635

    申请日:1993-10-21

    摘要: The invention relates to new 1-H-3-aryl-pyrrolidine-2,4-dione derivatives of the formula (I) ##STR1## in which A and B together with the carbon atom to which they are bonded represent a substituted cycle,X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents 0, 1, 2 or 3,G represents hydrogen (a) or the groups ##STR2## represents a metal ion equivalent or an ammonium ion, L and M represents oxygen and/or sulphur,R.sup.1 represents in each case optionally halogen-substituted alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl, which can be interrupted by hetero atoms, optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl,R.sup.2 represents in each case optionally halogen-substituted alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or in each case optionally substituted phenyl or benzyl,R.sup.3, R.sup.4 and R.sup.5 independently of one another represent in each case optionally halogen-substituted alkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkenylthio, cycloalkylthio and in each case optionally substituted phenyl, phenoxy or phenylthio,R.sup.6 and R.sup.7 independently of one another represent hydrogen, in each case optionally halogen-substituted alkyl, alkenyl, alkoxy, alkoxyalkyl, or represent optionally substituted phenyl, optionally substituted benzyl, or, together with the adjacent N-atom, represent a cycle which is optionally interrupted by oxygen or sulphur,to processes for their preparation, and to their use as pesticides.

    摘要翻译: 本发明涉及式(I)的新的1-H-3-芳基 - 吡咯烷-2,4-二酮衍生物,其中A和B与它们所键合的碳原子一起代表 取代的环,X表示烷基,卤素或烷氧基,Y表示氢,烷基,卤素,烷氧基或卤代烷基,Z表示烷基,卤素或烷氧基,n表示0,1,2或3,G表示氢(a) 表示金属离子当量或铵离子,L和M表示氧和/或硫,R1各自表示卤素取代的烷基,烯基,烷氧基烷基,烷硫基烷基,聚烷氧基烷基或环烷基,其可以是 被杂原子任选取代的苯基,任选取代的苯基烷基,取代的杂芳基,取代的苯氧基烷基或取代的羟基烷氧基烷基,R 2在每种情况下任选为卤素取代的烷基,烯基,烷氧基烷基,聚烷氧基烷基或在每种情况下任选取代的苯基o R 3,R 4和R 5彼此独立地表示在每种情况下任选为卤素取代的烷基,烷氧基,烷基氨基,二烷基氨基,烷硫基,烯硫基,环烷基硫基,并且在每种情况下均为任选取代的苯基,苯氧基或苯硫基,R6和R7独立地为 彼此表示氢,在各种情况下均为卤素取代的烷基,烯基,烷氧基,烷氧基烷基,或代表任选取代的苯基,任选取代的苄基,或与相邻的N-原子一起代表任选地被氧或 硫磺,其制备方法和作为农药的用途。