Substituted imidazolinylpyrimidines
    1.
    发明授权
    Substituted imidazolinylpyrimidines 失效
    取代的咪唑啉基嘧啶

    公开(公告)号:US5244865A

    公开(公告)日:1993-09-14

    申请号:US891493

    申请日:1992-05-29

    摘要: Herbicidal new substituted imidazolinylpyrimidines of the general formula (I) ##STR1## in which R.sup.1 represents hydrogen, halogen, cyano, nitro or thiocyanato, or represents a hydroxyl, mercapto, amino, carbonyl, sulphinyl, sulphonyl, alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aryl or heterocyclyl radical, each of which is optionally substituted,R.sup.2 represents hydrogen, hydroxyl, halogen, alkyl or halogenoalkyl,R.sup.3 represents hydrogen, or represents alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aryl or heterocyclyl, each of which is optionally substituted, or represents an equivalent of an inorganic or organic cation,R.sup.4 and R.sup.5 independently of each other in each case represent hydrogen, alkyl, halogenoalkyl or cycloalkyl andX represents oxygen or sulphur.

    摘要翻译: 通式(I)的除草新的取代的咪唑啉基嘧啶其中R 1表示氢,卤素,氰基,硝基或氰硫基,或表示羟基,巯基,氨基,羰基,亚磺酰基,磺酰基,烷基,烯基, 炔基,环烷基,环烯基,芳基或杂环基,其各自任选被取代,R 2表示氢,羟基,卤素,烷基或卤代烷基,R 3表示氢,或表示烷基,烯基,炔基,环烷基,环烯基,芳基或杂环基, 各自任选被取代,或表示无机或有机阳离子的当量,R 4和R 5彼此独立地表示氢,烷基,卤代烷基或环烷基,X表示氧或硫。

    Substituted triazolinone herbicides and plant growth regulators
    3.
    发明授权
    Substituted triazolinone herbicides and plant growth regulators 失效
    取代的三唑啉酮除草剂和植物生长调节剂

    公开(公告)号:US5523409A

    公开(公告)日:1996-06-04

    申请号:US125975

    申请日:1993-09-23

    摘要: Novel herbicides and plant growth regulants of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkylalkyl or cycloalkyl, or represents in each case optionally substituted aralkyl or aryl,R.sup.2 represents a radical ##STR2## or represents a radical --S(O).sub.n --R.sup.7, R.sup.3 and R.sup.4 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylaminoalkyl, alkoxycarbonylalkyl or alkoxycarbonylalkenyl, or represent in each case optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkenyl or cycloalkenylalkyl, or represent optionally substituted heterocyclylalkyl, or represent in each case optionally substituted aralkyl, aroyl or aryl, or represent alkoxy, alkenyloxy, alkinyloxy, aralkyloxy or aryloxy, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,X represents oxygen or sulphur andY represents oxygen or sulphur,whereinR.sup.5 and R.sup.6 independently of one another each represent alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkyl or cycloalkylalkyl, or represent in each case optionally substituted aryl, aralkyl or heteroaryl, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,R.sup.7 represents alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkylalkyl, or represents in each case optionally substituted aralkyl or aryl andn represents the number 0, 1 or 2,but wherein R.sup.2 only represents a radical --S(O).sub.n --R.sup.7 if R.sup.3 and R.sup.4 do not simultaneously represent methyl.Intermediates therefor where NR.sup.3 R.sup.4 is replaced by Cl are also new.

    摘要翻译: 式(I)的新型除草剂和植物生长调节剂,其中R 1表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基烷基或环烷基,或在每种情况下表示任选取代的芳烷基或 芳基,R 2表示基团,或表示基团-S(O)n -R 7,R 3和R 4彼此独立地表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,氰基烷基,羟基烷基,烷氧基烷基 或烷基氨基烷基,烷氧基羰基烷基或烷氧基羰基烯基,或在每种情况下表示任选取代的环烷基,环烷基烷基,环烯基或环烯基烷基,或代表任选取代的杂环基烷基,或在每种情况下表示任选取代的芳烷基,芳酰基或芳基,或代表烷氧基,烯氧基,烷氧基,芳烷氧基 或芳氧基,或者与它们所键合的氮原子一起代表任选的 取代的杂环基,X表示氧或硫,Y表示氧或硫,其中R5和R6彼此独立地表示烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基或环烷基烷基,或各自表示 任选取代的芳基,芳烷基或杂芳基,或与它们所键合的氮原子一起表示任选取代的杂环基,R 7表示烷基,烯基,炔基,环烷基或环烷基烷基,或在每种情况下表示任选取代的芳烷基或 芳基,n表示数字0,1或2,但如果R3和R4不同时表示甲基,则其中R2仅表示基团-S(O)n-R7。 NR3R4被Cl取代的中间体也是新的。

    Isoxazolecarboxylic acid derivatives
    5.
    发明授权
    Isoxazolecarboxylic acid derivatives 失效
    异恶唑羧酸衍生物

    公开(公告)号:US5374605A

    公开(公告)日:1994-12-20

    申请号:US2307

    申请日:1993-01-08

    摘要: The invention relates to isoxazolecarboxylic acid derivatives of the general formula (I) ##STR1## in which A represents alkanediyl,Q represents oxygen, sulphur, imino (NH) or alkylimino (N-alkyl),R.sup.1 represents an in each case optionally substituted radical from the series comprising alkyl, cycloalkyl or phenyl,R.sup.2 represents hydrogen, halogen or optionally substituted alkyl, andR.sup.3 represents in each case optionally substituted cyclohexyl or phenyl,with the exception of the compounds: N-benzyl-5-cyclopropyl-isoxazole-3-carboxamide N-(2-phenyl-ethyl)-5-methyl-isoxazole-3-carboxamide and N-benzyl-5-methyl-isoxazole-3-carboxamide, a process for their preparation, and their use as herbicides.

    摘要翻译: 本发明涉及通式(I)的化合物(I)的异恶唑羧酸衍生物,其中A代表烷二基,Q代表氧,硫,亚氨基(NH)或烷基亚氨基(N-烷基),R1代表每种情况 任选取代的烷基,环烷基或苯基系列的取代基,R 2表示氢,卤素或任选取代的烷基,R 3表示在任何情况下均为任选取代的环己基或苯基,但化合物除外:N-苄基-5-环丙基 - 异恶唑-3-甲酰胺N-(2-苯基 - 乙基)-5-甲基 - 异恶唑-3-甲酰胺和N-苄基-5-甲基 - 异恶唑-3-甲酰胺,其制备方法及其作为除草剂的用途 。

    Herbicidal substituted sulphonylamidinohydrazones
    9.
    发明授权
    Herbicidal substituted sulphonylamidinohydrazones 失效
    除草取代磺酰脒腙

    公开(公告)号:US5213608A

    公开(公告)日:1993-05-25

    申请号:US916330

    申请日:1992-07-16

    IPC分类号: A01N47/44 C07D521/00

    CPC分类号: C07D521/00 A01N47/44

    摘要: Herbicidal substituted sulphonylamidinohydrazones of the formula ##STR1## in which R.sup.1 represents in each case optionally substituted aryl, aralkyl or heteroaryl,R.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, aryl or aralkyl,R.sup.3 represents hydrogen, or represents in each case optionally substituted alkyl, alkenyl, alkadienyl, alkinyl, (hetero)aryl, aralkyl, aralkenyl, alkoxy, alkoxycarbonyl or dialkylamino, or together with R.sup.2 represents optionally substituted alkanediyl,R.sup.4 represents hydrogen, halogen, hydroxyl, alkyl, halogenoalkyl, alkoxyalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, amino, alkylamino or dialkylamino,X represents nitrogen or a --CH group,Y represents nitrogen or a --CR.sup.5 group whereR.sup.5 represents hydrogen, halogen, cyano, alkyl, formyl, alkyl-carbonyl or alkoxy-carbonyl, andZ represents nitrogen or a --CR.sup.6 group whereR.sup.6 represents hydrogen, halogen, hydroxyl, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, alkylamino or dialkylamino.

    摘要翻译: 式(I)的除草取代的磺酰基脒基腙,其中R 1在每种情况下表示任选取代的芳基,芳烷基或杂芳基,R 2表示氢,或在各种情况下表示任选取代的烷基,芳基或芳烷基,R 3表示氢或表示 在任何情况下,任选取代的烷基,烯基,链二烯基,炔基,(杂)芳基,芳烷基,芳烯基,烷氧基,烷氧基羰基或二烷基氨基,或与R 2表示任选取代的烷二基,R 4表示氢,卤素,羟基,烷基,卤代烷基, 烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,氨基,烷基氨基或二烷基氨基,X表示氮或-CH基,Y表示氮或-CR5基,其中R5表示氢,卤素,氰基,烷基,甲酰基, - 羰基,Z表示氮或-CR 6基团,其中R 6表示氢,卤素,羟基,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基, 烷基氨基或二烷基氨基。