公开(公告)号：US20070149400A1

公开(公告)日：2007-06-28

申请号：US10582934

申请日：2004-12-15

申请人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R1, R2 and/or R3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：L是氢，氯或溴; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或 含有一至四个由O，N和S杂原子组成的组的六元饱和，部分不饱和或芳族杂环，R 1和R 2连同氮 它们所连接的原子也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有作为环成员的O，N和S中的另外的杂原子和/或可被取代为 在说明书中定义; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，环烷基，卤代环烷基或苯基烷基; R 1，R 2和/或R 3可以如说明书中所定义的取代; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070117852A1

公开(公告)日：2007-05-24

申请号：US10582040

申请日：2004-12-22

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N43/56 ,  A01N43/40 ,  A01N43/78 ,  C07D213/24

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N47/48 ,  C07C251/38 ,  C07D207/34 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38

摘要： The present invention relates to (hetero)cyclylcarboxanilides of the formula I, in which n is 0, 1, 2, 3 or 4; and m is 1, 2 or 3, Y is oxygen or sulfur; A is unsubstituted or substituted phenyl or is an at least monounsaturated, unsubstituted or substituted 5- or 6-membered heterocycle, R1, R2, R3m, R4m, R5 and R6 are as defined in claim 1, and their agriculturally useful salts. Moreover, the present invention relates to the use of the (hetero)cyclylcarboxanilides of the formula I and their agriculturally useful salts as fungicides, and to crop protection compositions comprising these compounds.

摘要翻译： 本发明涉及式（I）的（杂）环己基甲酰苯胺，其中n为0,1,2,3或4; m为1,2或3，Y为氧或硫; A是未取代或取代的苯基，或至少是一个不饱和的，未取代的或取代的5元或6元杂环，R 1，R 2，R 3， R 4，R 5，R 5和R 6如权利要求1所定义，及其农业上有用的盐。 此外，本发明涉及式I的（杂）环己基甲酰苯胺及其农业上有用的盐作为杀真菌剂，以及包含这些化合物的作物保护组合物的用途。

公开(公告)号：US20070105873A1

公开(公告)日：2007-05-10

申请号：US10564013

申请日：2004-07-15

申请人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/54

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R3 and L are as defined in the description and R4 corresponds to one of the formulae in which Ra, X and Rb are as defined in the description; and also to processes for preparing these compounds, to pesticidal compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 3和L如说明书中所定义， SUP> 4 对应于其中R a，S，X和R b的定义之一如说明书中所定义; 以及制备这些化合物的方法，包括这些化合物的农药组合物及其作为农药的用途。

公开(公告)号：US20060229328A1

公开(公告)日：2006-10-12

申请号：US10549936

申请日：2004-03-30

申请人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D239/02

CPC分类号： A01N43/54 ,  C07D239/28 ,  C07D239/30

摘要： 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

公开(公告)号：US20050176736A1

公开(公告)日：2005-08-11

申请号：US10508409

申请日：2003-03-19

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C255/57

摘要： The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1-C8 alkoxy, C1-C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

摘要翻译： 本发明涉及式（I）的三唑并嘧啶，其中取代基定义如下：L 1表示氰基，S（-O）n A 1 或其中A 1代表氢，羟基，烷基，烷基氨基或二烷基氨基;或C（= O） A 2代表C 1 -C 8烷氧基，C 1 -C 6烷基，C 1 -C 6 - >卤代烷氧基或在A 中命名的基团之一; 而n代表0,1或2; L 2，L 3表示氢或卤素; L 4，L 5代表氢，卤素或烷基; X表示卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1表示烷基，卤代烷基，环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环 含有一个至四个来自含有O，N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环，其可被中断和/或被 来自O，N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物，含有后者的试剂和所述化合物用于防治有害真菌的用途。

公开(公告)号：US20050107401A1

公开(公告)日：2005-05-19

申请号：US10505146

申请日：2003-02-06

申请人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A61K31/506 ,  C07D43/04

CPC分类号： C07D401/04

摘要： The invention relates to 2-(2-pyridyl)-5-phenyl-6-amninopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

摘要翻译： 本发明涉及式I的2-（2-吡啶基）-5-苯基-6-脒嘧啶，其中取代基和指数具有以下含义：R 1表示卤素，羟基，杂环基， 烷氧基，烷氧基羰基，氨基甲酰基，烷基氨基羰基，二烷基氨基羰基，吗啉代羰基，吡咯烷基羰基，烷基羰基氨基，烷基氨基。 二烷基氨基，烷硫基，烷基亚磺酰基，烷基磺酰基，羟基磺酰基，氨基磺酰基，烷基氨基磺酰基，二烷基氨基磺酰基; m = 0或1-4; R 2表示氢，卤素，氰基，烷基，卤代烷基或烷氧基; R 3，R 4表示氢，烷基，卤代烷基，环烷基，卤代烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R 3 O 和R 4与它们连接的氮原子一起形成5或6元环，其被来自基团O，N或S的原子和/或可被取代 根据说明; R 5表示卤素，烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7，R 8表示氢，卤素，烷基或卤代烷基; R 9表示氢，卤素，羟基，氰基，烷基，烷氧基，环烷氧基，卤代烷氧基，烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物，除了其用于对抗不期望的植物之外。

公开(公告)号：US20100222219A1

公开(公告)日：2010-09-02

申请号：US12438169

申请日：2007-08-13

申请人： Jan Klaas Lohmann ,  Wassilios Grammenos ,  Michael Puhl ,  Jochen Dietz ,  Bernd Müller ,  Joachim Rheinheimer ,  Jens Renner

发明人： Jan Klaas Lohmann ,  Wassilios Grammenos ,  Michael Puhl ,  Jochen Dietz ,  Bernd Müller ,  Joachim Rheinheimer ,  Jens Renner

IPC分类号： A01C1/06 ,  C07D409/12 ,  A01N43/40 ,  A01P7/00 ,  A01P7/04

CPC分类号： A01N43/40 ,  C07D409/12

摘要： The present invention relates to thiophene-sulfonic acid picolyl amides of the Formula (I), where RI to R7 and n are as defined in the claims and to the N-oxides, the agriculturally acceptable salts and the veterinarily acceptable salts of the compounds (I), with the proviso that if the thiophene ring is bonded to the sulfonyl group via position 2, R6 cannot be at position 5. The invention also relates to a process for preparing these compounds. Furthermore, the invention relates to the use of the compounds I and the N-oxides and the agriculturally acceptable salts thereof for combating phytopathogenic fungi (hereinafter referred to as harmful fungi). Additionally, the compounds (I), their N-oxides and salts can be used for controlling arthropodal pests. Furthermore, the invention relates to seed comprising a compound (I) or an N-oxide or agriculturally acceptable salt thereof.

摘要翻译： 本发明涉及式（I）的噻吩 - 磺酸吡啶甲酰胺，其中R 1至R 7和n如权利要求中所定义，和N-氧化物，农业上可接受的盐和化合物的兽医学上可接受的盐 I），条件是如果噻吩环通过位置2与磺酰基键合，则R6不能在5位。本发明还涉及制备这些化合物的方法。 此外，本发明涉及化合物I和N-氧化物及其农业上可接受的盐对抗植物病原性真菌（以下称为有害真菌）的用途。 此外，化合物（I），其N-氧化物和盐可用于控制节肢动物害虫。 此外，本发明涉及包含化合物（I）或其N-氧化物或农业上可接受的盐的种子。

公开(公告)号：US20090099019A1

公开(公告)日：2009-04-16

申请号：US11920417

申请日：2006-05-16

申请人： Jochen Dietz ,  Markus Gewehr ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schafer

发明人： Jochen Dietz ,  Markus Gewehr ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schafer

IPC分类号： A01N43/78 ,  C07D277/56

CPC分类号： C07D277/56 ,  C07D277/587

摘要： Thiazolecarboxanilides of the formula I in which the variables are as defined below: A is X is halogen; Y is cyano, nitro, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is 0, 1; R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-haloalkyl; R2 is hydrogen, methyl, halogen; R3 is hydrogen, methyl, ethyl; W is O, S; and processes for preparing these compounds, compositions and seed comprising them and methods for controlling harmful fungi.

摘要翻译： 式I的噻唑甲酰苯胺，其中变量如下定义：A是X是卤素; Y是氰基，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，甲氧基或甲硫基; p为0，1; R1是氢，卤素，C1-C4-烷基，C1-C4卤代烷基; R2是氢，甲基，卤素; R3是氢，甲基，乙基; W是O，S; 以及制备这些化合物，组合物和包含它们的种子的方法以及用于控制有害真菌的方法。

公开(公告)号：US06730680B2

公开(公告)日：2004-05-04

申请号：US10314595

申请日：2002-12-10

申请人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

发明人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

IPC分类号： A01N4354

CPC分类号： C07D487/04

摘要： 6-Phenyl-Pyrazolopyrimidines of formula I wherein R1 is alkyl, alkenyl, alkynyl, alkadienyl or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom,  where these radicals may be unsubstituted or substituted as defined in the specification, Y is oxygen, sulfur, NR2 or a single bond; wherein R2 is defined in the specification; and R1 and R2 together with the interjacent nitrogen atom may represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted by one or more Rc radicals; m is 0 or an integer from 1 to 4; L each independently is halogen, nitro, alkyl, alkoxy, and X is halogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic fungi are described.

摘要翻译： 式I的6-苯基 - 吡唑并嘧啶，其中R 1是含有1-4个氮原子或一至三个氮的烷基，烯基，炔基，链二烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或5-或6-元杂环基 原子和一个硫或氧原子，或含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元杂芳基，其中这些基团可以未被取代或如说明书中所定义的取代， Y是氧，硫，NR 2或单键; 其中R 2在说明书中定义; 和R 1和R 2与中间的氮原子一起可以表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5或6元杂环，其可被取代 由一个或多个R c基团取代; m为0或1至4的整数; L各自独立地为卤素，硝基，烷基，烷氧基和X为卤素;制备这些化合物的方法和中间体， 描述了用于控制植物病原真菌的用途。

公开(公告)号：US06552026B2

公开(公告)日：2003-04-22

申请号：US09735033

申请日：2000-12-12

申请人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

发明人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

IPC分类号： C07D48704

CPC分类号： C07D487/04

摘要： 6-Phenyl-Pyrazolopyrimidines of formula I wherein R1 is alkyl, alkenyl, alkynyl, alkadienyl or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom,  where these radicals may be unsubstituted or substituted as defined in the specification, Y is oxygen, sulfur, NR2 or a single bond; wherein R2is defined in the specification; and R1 and R 2 together with the interjacent nitrogen atom may represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted by one or more Rc radicals; m is 0 or an integer from 1 to 4; L each independently is halogen, nitro, alkyl, alkoxy, and X is halogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic fungi are described.

摘要翻译： 式I的6-苯基 - 吡唑并嘧啶，其中R1是具有1-4个氮原子或1-3个氮原子的烷基，烯基，炔基，链二烯基或卤代烷基，环烷基，双环烷基，苯基，萘基或5-或6-元杂环基， 硫或氧原子，或含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元杂芳基，其中这些基团可以未被取代或如说明书中所定义取代，Y是氧 ，硫，NR 2或单键; 其中R2在说明书中定义; 并且R 1和R 2与中间的氮原子一起可以表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5或6元杂环，其可被一个或多个R c 基团; m为0或1至4的整数; L各自独立地为卤素，硝基，烷基，烷氧基和X为卤素;制备这些化合物的方法和中间体，包含它们的组合物及其用于防治植物病原真菌的用途。