公开(公告)号：US20070167463A1

公开(公告)日：2007-07-19

申请号：US10589876

申请日：2005-03-08

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04

摘要： 5,6-Dialkyl-7-aminotriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, alkoxymethylene or alkoxyethylene, where the aliphatic groups may be substituted as defined in the description; R2 is n-propyl or n-butyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的5,6-二烷基-7-氨基三唑并嘧啶：R 1是烷基，烷氧基亚甲基或烷氧基亚乙基，其中脂族基团可以如说明书中所定义的取代 ; R 2是正丙基或正丁基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070149588A1

公开(公告)日：2007-06-28

申请号：US10582984

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/64

CPC分类号： C07D487/04

摘要： The invention relates to 6-(2,3,6-trifluorophenyl)-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R2 represents hydrogen or one of the groups cited for R1; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N and can contain one to three additional heteroatoms from the groups O, N and S as a ring member; R1 and/or R2 can be substituted in accordance with the description; X represents cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy. The invention also relates to methods for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.

摘要翻译： 本发明涉及式（I）的6-（2,3,6-三氟苯基） - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基，卤代烷基，环烷基，卤代环烷基， 烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或含有一至四个O，N或S基的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R 2表示氢或R 1所引用的基团之一; R 1和R 2与它们所键合的氮原子一起也可以形成五或六元杂环基或杂芳基，其通过 并且可以含有一个至三个作为环成员的来自基团O，N和S的另外的杂原子; R 1和/或R 2可以根据描述代替; X表示氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基。 本发明还涉及生产所述化合物的方法，含有后者的试剂和用于对抗植物致病性真菌的用途。

公开(公告)号：US20070149515A1

公开(公告)日：2007-06-28

申请号：US10579144

申请日：2004-11-18

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04

摘要： 6-(2,4,6-Trifluorophenyl)triazolopyrimidines of the formula I in which the substituents have the following meanings: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, cycloalkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned in R1, R1 and R2 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered ring which is interrupted by an atom from the group consisting of O, N and S, and/or R1 and/or R2 can be substituted according to the description; X is cyano, C1-C4-alkoxy, C3-C4-alkenyloxy, C1-C2-haloalkoxy or C3-C4-halo-alkenyloxy; process for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

摘要翻译： 其中取代基具有以下含义的式I的6-（2,4,6-三氟苯基）三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基 ，卤代炔基，环炔基，苯基，萘基或五或六元饱和，部分不饱和或芳族杂环，其包含一至四个由O，N和S组成的组的杂原子，R 2是氢 或者R 1，R 1和R 2中提到的基团之一也可以与它们所键合的氮原子一起， 形成五元或六元环，其被来自由O，N和S组成的组的原子和/或R 1和/或R 2 可以根据描述进行替代; X是氰基，C 1 -C 4 - 烷氧基，C 3 -C 4 - 炔基氧基，C 1 -C 4 - C 1 -C 2 - 卤代烷氧基或C 3 -C 4 - 卤代 - 链烯氧基; 制备这些化合物的方法，包含它们的制剂及其在控制有害植物病原真菌中的用途。

公开(公告)号：US20070129380A1

公开(公告)日：2007-06-07

申请号：US10565656

申请日：2004-07-03

申请人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/505 ,  C07D239/42

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R1, R2 and R3 are as defined in the description and R4 is as defined below: R4 corresponds to one of the formulae where Ra is hydrogen, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C3-C6-cycloalkyl or C1-C4-alkoxy and R5 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C4-alkyloxy-C1-C2-alkyl, phenyl-C1-C2-alkyl or phenyloxy-C1-C2-alkyl, to processes for preparing these compounds, to compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和这些取代基R 1，R 2和R 3是 如在说明书中所定义的，R 4是如下定义的：R 4对应于下式之一其中R a a是氢，C 1〜 C 1 -C 6烷基，C 2 -C 8 - 烯基，C 2 - 亚烷基，C 2 -C 6 - C 1 -C 8 - 炔基，C 3 -C 6 - 环烷基或C 1 -C 6 - 4 - 烷氧基和R 5是氢，C 1 -C 6 - 烷基，C 2〜 C 1 -C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 6 - 4 - 烷氧基-C 1 -C 2 - 烷基，苯基-C 1 -C 2 - 亚烷基 烷基或苯氧基-C 1 -C 2 - 烷基，用于制备这些化合物的方法，包含这些化合物的组合物及其作为农药的用途。

公开(公告)号：US20060211711A1

公开(公告)日：2006-09-21

申请号：US10550571

申请日：2004-03-30

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-烷基氨基 - 三唑并嘧啶类，其中取代基具有以下含义：L =卤素，烷基，卤代烷基，烷氧基，氨基，NHR，NR 2，氰基，S（O） 或者C（O）A 2 O 2。 R =烷基或烷基羰基，A 1〜H 2，羟基，烷基，烷基氨基或亚烷基氨基; n = 0,1或2; 链烯基，烷氧基，卤代烷氧基或A 1中引用的基团之一; m = 1,2,3,4或5，其中至少一个基团L存在于与三唑并嘧啶骨架的键的邻位; X =卤素，氰基，烷基，卤代烷基或烷氧基; R 1 =氢或烷基; R 2 =炔基，其可以是未取代的或根据描述取代的。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂及其用于对抗有害植物病原真菌的用途。

公开(公告)号：US20060135538A1

公开(公告)日：2006-06-22

申请号：US11340977

申请日：2006-01-30

申请人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-(R)-Aminotriazolopyrimidines of the formula I where the substituents and the index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C1o-alkyl, C1-C4-alkoxymethyl, C3-C1o-cycloalkyl; R4 is halogen, Cl-C4-alkyl, C1-C4-haloalkyl or Cl-C4-alkoxy; n is a number from 1 to 5; Y is halogen, cyano, Cl-C4-alkyl or Cl-C4-alkoxy; where * is a center of chirality in the R configuration, processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 7-（R） - 取代基和指数如下所定义的式I的氨基三唑并嘧啶：R 1是氢或甲基; R 2是甲基; R 3是C 1 -C 2烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷基， 亚烷基氧基甲基，C 3 -C 30环烷基; R 4是卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基或C 1 -C 4 - C 4 - 烷氧基; n是从1到5的数字; Y是卤素，氰基，C 1 -C 4 - 烷基或C 1 -C 4 - 烷氧基; 其中*是R构型的手性中心，描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20050272748A1

公开(公告)日：2005-12-08

申请号：US10531980

申请日：2003-11-14

申请人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or —C(═O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R1 and/or R2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 2-巯基取代的式Ⅰ的三唑并嘧啶，其中取代基如下：L是卤素，氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基或-C ）-一个; A是氢，羟基，烷基，烯基，烷氧基，卤代烷氧基，烷基氨基或二烷基氨基; m为0,1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 至10元饱和，部分不饱和或芳族杂环，其含有一个至四个由O，N和S组成的组的杂原子; R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元环，其可被来自基团的原子中断 由O，N和S组成; 其中R 1和/或R 2可以如描述中所述被取代; 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US06956034B2

公开(公告)日：2005-10-18

申请号：US10477355

申请日：2002-05-17

申请人： Joachim Rheinheimer ,  Andreas Gypser ,  Ingo Rose ,  Thomas Grote ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Joachim Rheinheimer ,  Andreas Gypser ,  Ingo Rose ,  Thomas Grote ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  John-Bryan Speakman ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04 ,  C07D413/04 ,  A61K31/536 ,  A61K31/5365

CPC分类号： C07D513/04 ,  A01N43/86 ,  A01N43/90 ,  C07D265/24

摘要： Oxazin(ethi)one compounds of the formula I: in which the variables Z, R1, R2, R3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.

摘要翻译： 恶嗪（ethi）一种式I化合物，其中变量Z，R 1，R 2，R 3和n分别为 权利要求1中限定，A是5或6元碳环或具有1,2或3个选自N，O和S的杂原子的5或6元杂环，其中每个杂环通过 描述了两个碳原子与恶嗪（ethi）一个环，并且描述了恶嗪（ethi）一种化合物I的农业上有用的盐。 此外，本发明描述了化合物I及其盐用于控制植物病原真菌的用途，其包含化合物I和/或其盐的杀真菌有效量的组合物和控制植物病原真菌的方法，其包括处理真菌或物质， 用杀真菌有效量的至少一种如权利要求1所述的式I化合物和/或其盐的植物，种子或受真菌侵袭威胁的土壤。

公开(公告)号：US06559151B2

公开(公告)日：2003-05-06

申请号：US09735126

申请日：2000-12-12

申请人： Klaus Jüergen Pees ,  Frank Schieweck ,  Jordi Tormo I Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

发明人： Klaus Jüergen Pees ,  Frank Schieweck ,  Jordi Tormo I Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

IPC分类号： A01N4390

CPC分类号： C07D487/04

摘要： 6-(2-Trifluoromethyl-phenyl)-triazolopyrimidines of formula I in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or substituted as defined in the specification; or R1 and R2 together with the interjacent nitrogen atom represents a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted as defined in the specification; R3 is hydrogen, halogen, alkyl, alkoxy and haloalkyl; and X is halogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic fungi are described.

摘要翻译： 具有式Iin的6-（2-三氟甲基 - 苯基） - 三唑并嘧啶，其中R1和R2独立地表示氢或烷基，烯基，炔基，链二烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或5-或6-元杂环基， 至四个氮原子或一至三个氮原子和一个硫或氧原子，或5-或6-元杂芳基，其含有1-4个氮原子或1-3个氮原子和一个硫或氧原子，或其中R1和R2基团可以 如说明书中所定义; 或R 1和R 2与中间的氮原子一起表示含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5或6元杂环，其可以如说明书中所定义而被取代; R3 是氢，卤素，烷基，烷氧基和卤代烷基; 和X是卤素;描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原真菌的用途。

公开(公告)号：US06262273B1

公开(公告)日：2001-07-17

申请号：US09254569

申请日：1999-03-10

申请人： Gerhard Hamprecht ,  Joachim Gebhardt ,  Heinz Isak ,  Michael Rack ,  Joachim Rheinheimer ,  Peter Schäfer

发明人： Gerhard Hamprecht ,  Joachim Gebhardt ,  Heinz Isak ,  Michael Rack ,  Joachim Rheinheimer ,  Peter Schäfer

IPC分类号： C07D21371

CPC分类号： C07D213/71

摘要： Substituted thiopyridines of the general formula I where n is 1 or 2; R1 is chlorine, C1-C3-fluoroalkyl, nitro or methylsulfonyl; R2 is a C1-C10-alkyl, C2-C10-alkenyl or C2-C10-alkynyl radical, in each case unsubstituted or substituted by halogen, C1-C4-alkoxy, C1-C4-alkoxycarbonyl, di-(C1-C4-alkylamino) carbonyl, cyano or nitro, a C3-C8-cycloalkyl radical, or a C1-C4-alkylenephenyl, phenyl or naphthyl radical which is unsubstituted or substituted in the phenyl moiety by halogen, C1-C3-alkyl, C1-C3-alkoxy, trifluoromethyl, cyano or nitro.

摘要翻译： 通式Iwheren的取代的硫代吡啶为1或2; R 1为氯，C 1 -C 3 - 氟代烷基，硝基或甲基磺酰基; R 2为C 1 -C 10 - 烷基，C 2 -C 10 - 烯基或C 2 -C 10 - 炔基 C 1 -C 4 - 烷氧基羰基，C 1 -C 4 - 烷基氨基羰基，氰基或硝基，C 3 -C 8环烷基或C 1 -C 4亚烷基苯基， 苯基或萘基，其在苯基部分被卤素，C 1 -C 3 - 烷基，C 1 -C 3 - 烷氧基，三氟甲基，氰基或硝基取代。