Hypertensive phenylalkylamines and salts thereof
    108.
    发明授权
    Hypertensive phenylalkylamines and salts thereof 失效
    高效苯丙氨酸及其盐

    公开(公告)号:US4146645A

    公开(公告)日:1979-03-27

    申请号:US761476

    申请日:1977-01-24

    CPC分类号: C07C275/40

    摘要: Compounds of the formula ##STR1## wherein R.sub.1 is hydrogen, --(CH.sub.2).sub.n --R.sub.4 or --CO--R.sub.5,where n is 1 or 2,R.sub.4 is hydrogen, cyano or benzoyl, andR.sub.5 is hydrogen, lower alkoxy, benzyloxy, --CH.sub.2 --NH.sub.2, --CH(CH.sub.3)--NH.sub.2, --CH.sub.2 --NH--CH.sub.2 --C.sub.6 H.sub.5 or --CH(CH.sub.3)--NH--CH.sub.2 --C.sub.6 H.sub.5,R.sub.2 is hydrogen or methyl, andR.sub.3 is amino, nitro, --NH--CO--R.sub.6 or --NH--A--R.sub.7,where R.sub.6 is hydrogen, methyl, methoxy, ethoxy, methylthio or ethylthio,R.sub.7 is amino, methylamino or dimethylamino, andA is --CO-- or --SO.sub.2 --,provided, however, that R.sub.1 and R.sub.4 are other than hydrogen and R.sub.2 is other than hydrogen or methyl when R.sub.6 is hydrogen or methyl, and non-toxic, pharmacologically acceptable acid addition salts thereof; the compounds as well as their salts are useful as hypertensives.

    Alkyl-4-alkyl-N-alkoxycarbonyl-1-thioallophanimidate
    109.
    发明授权
    Alkyl-4-alkyl-N-alkoxycarbonyl-1-thioallophanimidate 失效
    烷基-4-烷基-N-烷氧羰基-1-硫代乙酰亚氨酸酯

    公开(公告)号:US4014924A

    公开(公告)日:1977-03-29

    申请号:US662002

    申请日:1976-02-27

    CPC分类号: C07C335/38

    摘要: Allophanimidates and carbamates of the formulas ##STR1## where R.sub.1 is hydrogen or alkyl;R.sub.2 is alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, benzyl or phenyl optionally substituted;R.sub.3 is SR.sub.4 or OR.sub.4 ;R.sub.4 is alkyl, cycloalkyl, alkenyl, alkynyl, phenyl, or benzyl;R.sub.5 is alkyl, alkenyl, cycloalkyl, benzyl or phenyl optionally substituted; andR.sub.6 is hydrogen or alkylX.sub.1, x.sub.2 and X.sub.3 are oxygen or sulfur, are useful as herbicides.Exemplary of the compounds is methyl 4-tert-butyl-N-methoxycarbonyl-1-thioallophanimidate.

    摘要翻译: 其中R 1是氢或烷基的式(I)的化合物: R2是烷基,环烷基,环烷基烷基,烯基,炔基,苄基或任选取代的苯基; R3是SR4或OR4; R4是烷基,环烷基,烯基,炔基,苯基或苄基; R5是烷基,烯基,环烷基,苄基或任选取代的苯基; R 6为氢或烷基X1,X 2和X 3为氧或硫,可用作除草剂。