公开(公告)号：US20090131462A1

公开(公告)日：2009-05-21

申请号：US11988471

申请日：2006-07-21

Applicant: Markus Gewehr ,  Reinhard Stierl ,  Horst Dieter Brix ,  Thomas Grote ,  Siegfried Strathmann ,  Maria Scherer ,  Frank Werner

Inventor： Markus Gewehr ,  Reinhard Stierl ,  Horst Dieter Brix ,  Thomas Grote ,  Siegfried Strathmann ,  Maria Scherer ,  Frank Werner

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  A01N43/50 ,  A01P3/00 ,  A01N43/76 ,  A01N43/653 ,  A01N43/40

CPC classification number: A01N43/56 ,  A01N47/14 ,  A01N61/00 ,  A01N2300/00

Abstract: The invention relates to a fungicidally active agent containing at least one other defined fungicide in addition to the fungicide N-[2-(1,3-dimethylbutyl)-3-thienyl]-1-methyl-3-(trifluormethyl)-1H-pyrazol-4-carboxamide (penthiopyrad). The invention also relates to a method for controlling pathogenic fungi using one such agent, and to the use of said agent for controlling pathogenic fungi.

Abstract translation: 本发明涉及除了杀真菌剂N- [2-（1,3-二甲基丁基）-3-噻吩基] -1-甲基-3-（三氟甲基）-1H-咪唑类除外，还含有至少一种其它限定的杀真菌剂的杀真菌活性剂 吡唑-4-甲酰胺（五氯吡啶）。 本发明还涉及使用一种这样的试剂控制致病真菌的方法，以及所述药物用于控制致病真菌的用途。

公开(公告)号：US07501530B2

公开(公告)日：2009-03-10

申请号：US10548840

申请日：2004-03-20

Applicant: Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Tormo i Blasco ,  Anja Schwögler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

Inventor： Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Tormo i Blasco ,  Anja Schwögler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

IPC: C07D333/22 ,  C07C333/32 ,  A01N25/00 ,  C07C335/00 ,  A01N25/32

CPC classification number: C07D333/38

Abstract: The invention relates to novel biphenyl carboxamides of formula (I), wherein A, R, Z, X, Y, m and n have the meanings given in the description, to multiple methods for producing these substances, to their use for combating unwanted micro-organisms and to novel intermediate products and the production thereof.

Abstract translation: 本发明涉及式（I）的新型联苯甲酰胺，其中A，R，Z，X，Y，m和n具有与本说明书中给出的含义相同的多种生产这些物质的方法，用于防治不想要的微生物 和新颖的中间产品及其生产。

公开(公告)号：US07449471B2

公开(公告)日：2008-11-11

申请号：US11677862

申请日：2007-02-22

Applicant: Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

Inventor： Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC: C07D239/42 ,  C07D239/30 ,  A61K31/505 ,  A61K31/506 ,  A01N43/54

CPC classification number: C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

Abstract: 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5 ; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：US20080269171A1

公开(公告)日：2008-10-30

申请号：US11778784

申请日：2007-07-17

Applicant: Eberhard Ammermann ,  Reinhard Stierl ,  Gisela Lorenz ,  Siegfried Strathmann ,  Klaus Schelberger ,  V. James Spadafora ,  Thomas Christen

Inventor： Eberhard Ammermann ,  Reinhard Stierl ,  Gisela Lorenz ,  Siegfried Strathmann ,  Klaus Schelberger ,  V. James Spadafora ,  Thomas Christen

IPC: A01N57/16 ,  A01N43/653 ,  A01N43/88 ,  A01P3/00

CPC classification number: A01N43/653 ,  A01N57/16 ,  A01N51/00 ,  A01N47/02 ,  A01N2300/00

Abstract: A fungicidal mixture, comprising (1) 2-[2-(1-chlorocyclopropyl)-3-(2-chlorophenyl)-2-hydroxypropyl]-2,4-dihydro-[1,2,4]-triazole-3-thione (prothioconazole) of the formula I or its salts or adducts and at least one insecticide selected from the group consisting of (2) fipronil of the formula II (3) chlorpyrifos of the formula III (4) thiamethoxam of the formula IV in a synergistically effective amount is described.

Abstract translation: 一种杀真菌混合物，其包含（1）2- [2-（1-氯环丙基）-3-（2-氯苯基）-2-羟丙基] -2,4-二氢 - [1,2,4] 式（I）的硫酮（丙硫菌唑）或其盐或加合物和至少一种杀虫剂，其选自（2）式II（3）的氟虫腈式（Ⅳ）式Ⅳ的毒死蜱将式Ⅳ的噻虫嗪 描述协同有效量。

公开(公告)号：US20080176831A1

公开(公告)日：2008-07-24

申请号：US11596891

申请日：2005-05-17

Applicant: Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

Inventor： Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC: A01N43/46 ,  C07D403/04 ,  A01N43/54 ,  A01P7/00 ,  A01P3/00 ,  A01N43/58

CPC classification number: C07D401/04 ,  C07D403/04

Abstract: The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N— or —S—; R1 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

Abstract translation: 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R 1至R 3如在说明书中所定义，X是 基团-CH-R a，N - 或-S-; R 1可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 3 > 6个 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a， p是1至4的整数; Y是基团-CH-R a - 或-N-R b是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6 烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物及其作为农药的用途。

公开(公告)号：US20080153700A1

公开(公告)日：2008-06-26

申请号：US10589877

申请日：2005-03-14

Applicant: Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

Inventor： Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC: A01N43/90 ,  A01N25/26 ,  A01P3/00

CPC classification number: A01N43/90 ,  A01N47/04 ,  A01N2300/00

Abstract: Fungicidal mixtures comprising, as active components, 1 ) the triazolopyrimidine derivative of the formula I 2) tolylfluanid of the formula II, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures, and also compositions comprising these mixtures.

Abstract translation: 作为活性成分的杀真菌混合物包括：1）式II的三唑并嘧啶衍生物2）式II的甲苯基流质，协同有效量，使用化合物I与化合物II的混合物来控制有害真菌的方法，以及使用 具有用于制备这种混合物的化合物II的化合物I，以及包含这些混合物的组合物。

公开(公告)号：US20080132522A1

公开(公告)日：2008-06-05

申请号：US11631006

申请日：2005-07-12

Applicant: Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/54 ,  C07D401/04 ,  A01P3/00 ,  A01P13/00 ,  A01P15/00

CPC classification number: C07D239/34 ,  C07D401/04 ,  C07D403/12

Abstract: The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R4, B and L are as defined in the description and Y is a group —O— or —S—, and to processes for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

Abstract translation: 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 4，B和L如说明书中所定义，以及 Y是基团-O-或-S-，并且使用本发明的化合物进行制备，杀虫组合物和控制有害真菌和动物害虫的方法。

公开(公告)号：US20080108686A1

公开(公告)日：2008-05-08

申请号：US11628325

申请日：2005-06-16

Applicant: Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

Inventor： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC: A01N43/56 ,  A01P3/00 ,  C07D231/12

CPC classification number: A01N43/56 ,  C07D231/14

Abstract: The present invention relates to N-(ortho-phenyl)-1-methyl-3-difluoromethylpyrazole-4-carboxanilides of the formula I in which the substituents are as defined below:R1 and R2 independently of one another are halogen, C1-C6-alkyl, C1-C6-haloalkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy.

Abstract translation: 本发明涉及式I的N-（邻苯基）-1-甲基-3-二氟甲基吡唑-4-甲酰苯胺，其中取代基如下：R 1和R 2 > 2个彼此独立地是卤素，C 1 -C 6 - 烷基，C 1 -C 6 氰基，硝基，甲氧基，三氟甲氧基或二氟甲氧基。

公开(公告)号：US20080064756A1

公开(公告)日：2008-03-13

申请号：US10566297

申请日：2004-08-13

Applicant: Rainer Berghaus ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann

Inventor： Rainer Berghaus ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann

IPC: A01N37/52

CPC classification number: A01N43/10 ,  A01N37/52 ,  A01N43/56 ,  A01N43/653 ,  A01N2300/00

Abstract: The present invention relates to the use of alkoxylated alcohols (alcohol alkoxylates) as adjuvant for improving the fungicidal action of benzamide oxime derivatives of the formula (I) such as, for example, N-phenylacetyl-2-difluoromethoxy-5,6-difluorobenzamide (O-cyclopropylmethyl)oxime or N-phenylacetyl-2-trifluoromethoxy-5,6-difluorobenzamide (O-cyclopropylmethyl)oxime. The present invention also relates to corresponding compositions and kits.

Abstract translation: 本发明涉及烷氧基化醇（醇烷氧基化物）作为佐剂用于改善式（I）的苯甲酰胺肟衍生物的杀真菌作用的用途，例如N-苯基乙酰基-2-二氟甲氧基-5,6-二氟苯甲酰胺 （O-环丙基甲基）肟或N-苯基乙酰基-2-三氟甲氧基-5,6-二氟苯甲酰胺（O-环丙基甲基）肟。 本发明还涉及相应的组合物和试剂盒。

公开(公告)号：US20080058208A1

公开(公告)日：2008-03-06

申请号：US11547185

申请日：2005-03-26

Applicant: Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: C07D487/04 ,  A01N25/34 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-cycloalkyl-7-aminotriazolopyrimidines of formula (I), where X=alkylene or alkenylene, whereby the carbon chain can be interrupted by one or two heteroatoms selected from S, O or NR1, R1═H, alkyl or C(═O)alkyl, L=halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, alkinyl or NR2R3; R2,R3=each one of the groups given for R1 and m=a whole number from 0 to 5, whereby the aliphatic groups can be substituted by one to three of the following groups: halogen, cyano, nitro, hydroxy, alkoxy, alkylthio, or NRaRb, where Ra, Rb═H or alkyl in which the carbon chains can be halogenated. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the prevention of fungal pests harmful to plants.

Abstract translation: 本发明涉及式（I）的5,6-环烷基-7-氨基三唑并嘧啶，其中X =亚烷基或亚烯基，其中碳链可被一个或两个选自S，O或NR 1的杂原子中断， 卤素，氰基，硝基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，炔基或NR 2（O） 3 3 R 2，R 3 =每个给定R 1的基团，m = 0至5的整数，由此脂族基 基团可以被一至三个以下基团取代：卤素，氰基，硝基，羟基，烷氧基，烷硫基或NR a R b，其中R 0， 或其中碳链可以被卤化的烷基。 本发明还涉及生产所述化合物的方法，包含该化合物的试剂及其用于预防对植物有害的真菌害虫的用途。