公开(公告)号：US20090036509A1

公开(公告)日：2009-02-05

申请号：US11628324

申请日：2005-06-11

Applicant: Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

Inventor： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC: A01N43/56 ,  C07D231/14 ,  A01P3/00

CPC classification number: C07D231/14

Abstract: The present invention relates to N-(ortho-phenyl)-1-methyl-3-trifluoromethylpyrazole-4-carboxanilides of the formula I in which the substituents are as defined below: R1 and R2 independently of one another are halogen, C1-C6-alkyl, C1-C6-haloalkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy; with the proviso that when R2 is chlorine in position 4, R1 is not trifluoromethyl in position 3.

Abstract translation: 本发明涉及式I的N-（邻 - 苯基）-1-甲基-3-三氟甲基吡唑-4-甲酰苯胺，其中取代基如下所定义：R 1和R 2彼此独立地为卤素，C 1 -C 6 烷基，C 1 -C 6卤代烷基，氰基，硝基，甲氧基，三氟甲氧基或二氟甲氧基; 条件是当R2在4位是氯时，R1不在3位是三氟甲基。

公开(公告)号：US20080200334A1

公开(公告)日：2008-08-21

申请号：US11791191

申请日：2005-11-23

Applicant: Jordi Tormo I Blasco ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Matthias Niedenbruck ,  Horst Dieter Brix ,  Markus Gewehr ,  Christine Beck

Inventor： Jordi Tormo I Blasco ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Matthias Niedenbruck ,  Horst Dieter Brix ,  Markus Gewehr ,  Christine Beck

IPC: A01N25/26 ,  A01N43/78 ,  A01N43/84 ,  A01N43/32 ,  A01N43/56 ,  A01P3/00

CPC classification number: A01N43/78 ,  A01N47/04 ,  A01N2300/00

Abstract: Method for enhancing the fungicidal effectiveness of a) ethaboxam of the formula I, which comprises applying the active compound I simultaneously, that is separately or together, with at least one active compound II from the group consisting of: b) dithiocarbamates, such as maneb, mancozeb, metam or metiram, sulfenic acid derivatives, such as captan or folpet, strobilurin derivatives, such as kresoxim-methyl or pyraclostrobin, cinnamides and analogs, such as dimethomorph or flumorph, or dithianon, famoxadone, cymoxanil, fluazinam, zoxamide, mefenoxam or chlorothalonil, N-(2-{4-[3-(4-chlorophenyl)prop-2-ynyloxy]-3-methoxyphenyl}ethyl)-2-methanesulfonylamino-3-methylbutyramide, N-(2-{4-[3-(4-chlorophenyl)prop-2-ynyloxy]-3-methoxyphenyl}ethyl)-2-ethanesulfonylamino-3-methylbutyramide or 5-chloro-7-(4-methylpiperidin-1-yl)-6-(2,4,6-trifluorophenyl)-[1,2,4]triazolo[1,5-a]pyrimidine in synergistically effective amounts, by spraying or dusting the seeds, the plants or the soils before or after sowing of the plants or before or after emergence of the plants, no polyoxyalkylene alkyl ether being used as adjuvants, novel synergistic mixtures of ethaboxam and also compositions comprising these mixtures, and the use of ethaboxam for preparing such mixtures.

Abstract translation: 提高a）式I的ethaboxam的方法，其包括将活性化合物I同时与另一种或一起与至少一种活性化合物II一起施用，所述活性化合物II来自以下组中的至少一种活性化合物II：b）二硫代氨基甲酸盐，例如maneb ，代森锰锌，metam或metiram，磺酸衍生物，例如克虏伯或派生物，嗜球果伞形毒素衍生物，例如甲氧基甲基或嘧菌酯，肉桂酸酯和类似物，例如烯酰吗啉或氟吗啉，或二噻尼龙，恶唑酮，胞嘧啶，氟啶胺，唑酰胺， 或百菌清，N-（2- {4- [3-（4-氯苯基）丙-2-炔基氧基] -3-甲氧基苯基}乙基）-2-甲磺酰基氨基-3-甲基丁酰胺，N-（2- {4- [ 3-（4-氯苯基）丙-2-炔基氧基] -3-甲氧基苯基}乙基）-2-乙磺酰基氨基-3-甲基丁酰胺或5-氯-7-（4-甲基哌啶-1-基）-6-（2， 4,6-三氟苯基） - [1,2,4]三唑并[1,5-a]嘧啶，具有协同有效的量，通过在或之前喷洒或除尘种子，植物或土壤 r播种植物或在植物出现之前或之后，不使用聚氧亚烷基烷基醚作为佐剂，含有这些混合物的组合物的ethaboxam的新型协同混合物，以及使用ethaboxam制备这些混合物。

公开(公告)号：US20080171774A1

公开(公告)日：2008-07-17

申请号：US11885990

申请日：2006-03-15

Applicant: Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether ,  Karl Eicken

Inventor： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether ,  Karl Eicken

IPC: C07D213/63 ,  C07D213/56 ,  A61K31/4415 ,  A61K31/455

CPC classification number: C07D213/82

Abstract: The present invention relates to nicotinanilides of the formula I in which: n=0, 1, 2; m=2, 3; X1=F, chlorine; X2=halogen; Y=CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p=0, 1; R1=halogen, methyl, C1-C4-haloalkyl, methoxy, methylthio, methylsulfinyl or methylsulfonyl; R2=hydrogen, methyl or ethyl; W=O, S; processes for preparing these compounds, compositions and seed comprising them and also methods for controlling harmful fungi.

Abstract translation: 本发明涉及式I的烟酰苯胺，其中：n = 0,1,2; m = 2，3; X 1 = F，氯; X 2 =卤素; Y = CN，NO 2，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 卤代烷基，甲氧基或甲硫基; p = 0,1， R 1 =卤素，甲基，C 1 -C 4 - 卤代烷基，甲氧基，甲硫基，甲基亚磺酰基或甲基磺酰基; R 2 =氢，甲基或乙基; W = O，S; 制备这些化合物的方法，包含它们的组合物和种子以及控制有害真菌的方法。

公开(公告)号：US20080153824A1

公开(公告)日：2008-06-26

申请号：US11793617

申请日：2005-12-16

Applicant: John-Bryan Speakman ,  Reinhard Stierl ,  Siegfried Strathmann ,  Peter Dombo ,  Matthias Niedenbruck ,  Egon Haden ,  Dirk Voeste ,  Ulf Groeger

Inventor： John-Bryan Speakman ,  Reinhard Stierl ,  Siegfried Strathmann ,  Peter Dombo ,  Matthias Niedenbruck ,  Egon Haden ,  Dirk Voeste ,  Ulf Groeger

IPC: A01N37/50 ,  A01N43/653 ,  A01P3/00 ,  A01N43/50 ,  A01N43/56 ,  A01N43/54 ,  A01N43/34 ,  A01N43/36 ,  A01N43/84 ,  A01N47/28 ,  A01N37/00

CPC classification number: A01N37/50 ,  A01N2300/00

Abstract: Method for controlling rust infections in leguminous plants by using orysastrobin, mixtures of orysastrobin and a fungicidally active compound II from the group of the azoles, acylalanines, amine derivatives, anilinopyrimidines, dicarboximides, dithiocarbamates, heterocylic compounds, phenylpyrroles, cinnamides, and analogs, or other fungicides according to the description, and also compositions and seed comprising these mixtures.

Abstract translation: 通过使用orysastrobin来控制豆科植物中的生锈感染的方法，或者来自唑烷类的混合物和来自唑类，酰基丙氨酸，胺衍生物，苯胺基嘧啶，二甲酰亚胺，二硫代氨基甲酸酯，杂环化合物，苯基吡咯，肉桂酸酯和类似物的混合物，或 根据描述的其它杀真菌剂，以及包含这些混合物的组合物和种子。

公开(公告)号：US07388018B2

公开(公告)日：2008-06-17

申请号：US10570893

申请日：2004-09-10

Applicant: Wassilios Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Götz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

Inventor： Wassilios Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Götz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

IPC: A61K31/541 ,  A61K31/496 ,  C07D417/02 ,  C07D403/02

CPC classification number: C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

Abstract: Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2, and R3, R2, R3, are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group —C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

Abstract translation: 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， R 3，R 2，R 3，R 3，R 3，R 3，R 3，R 3，R 3，R 3，R 3， 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 由基团-C（R 6） - NOR 7取代的苯基，其中R 6为烷基，R 7为H 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080103144A1

公开(公告)日：2008-05-01

申请号：US11322211

申请日：2005-12-30

Applicant: Klaus Schelberger ,  Maria Scherer ,  Karl Eicken ,  Manfred Hampel ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

Inventor： Klaus Schelberger ,  Maria Scherer ,  Karl Eicken ,  Manfred Hampel ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC: A01N47/10 ,  A01N43/08 ,  A01N37/34 ,  A01N37/12 ,  A01N37/18 ,  A01N37/44

CPC classification number: A01N43/40 ,  A01N47/34 ,  A01N47/12 ,  A01N43/76 ,  A01N43/08 ,  A01N37/46 ,  A01N37/38 ,  A01N37/36 ,  A01N2300/00

Abstract: Fungicidal mixtures comprise as active componentsa) an amide compound of the formula I A—CO—NR1R2 I in which A, R1 and R2 are as defined in the description, andb) dimethomorph or flumetover, and/orc) a valinamide of the formula III in which R13 is C3-C4-alkyl and R14 is naphthyl or phenyl, where the phenyl radical is substituted in the 4-position by a halogen atom, a C1-C4-alkyl or C1-C4-alkoxy group, and/or d) benalaxyl, ofurace, metalaxyl, furalaxyl or oxydixyl, and/ore) 1-(2-cyano-2-methoxyiminoacetyl)-3-ethylureain a synergistically effective amount.

Abstract translation: 杀真菌混合物包含作为活性组分的a）式I的酰胺化合物<？in-line-formula description =“In-line Formulas”end =“lead”→> A-CO-NR 1 其中A，R 1和R 2各自独立地表示：其中A，R 1，R 2， 2）如说明书中所定义，和b）烯酰吗啉或flumetover，和/或c）式III的缬氨酰胺，其中R 13是C 3

公开(公告)号：US20080076785A1

公开(公告)日：2008-03-27

申请号：US11663982

申请日：2005-09-27

Applicant: Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

Inventor： Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC: A01N43/54 ,  A01P3/00 ,  C07D239/70

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.

Abstract translation: 本发明涉及通式（I）的7-氨基甲基-1,2,4-三唑并[1,5-a]嘧啶化合物和所述化合物的农业上相容的盐。 在所述式中：R 1和R 2表示氢，烷基，卤代烷基，烷氧基，环烷基，二环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或5-或6-元饱和， 部分不饱和或芳族杂环，含有1至4个含有O，N或S的杂原子，或R 1和R 2与它们所键合的氮原子一起也可以形成五元或六元杂环基或杂芳基 ，其通过N键合并且可以含有来自含有O，N和S的基团的1至3个另外的杂原子作为环成员，并且可以根据描述进行取代; R3和R4代表氢，烷基，卤代烷基，卤代烷氧基，烷氧基或烷氧基烷基; X代表卤素，氰基，含有1,2或3个杂原子的5-或6-元饱和的部分不饱和或芳族杂环，所述杂环含有作为环成员的O，N或S，烷基，烷氧基，烯基或炔基， 由此后4个组可以根据描述被替代; L定义为权利要求书和说明书中引用的; 和m表示0,1,2,3,4或5.本发明还涉及通式（I）的三唑并嘧啶化合物及其农业上相容的盐用于控制植物致病真菌的用途，用于控制植物的方法 致病真菌，含有至少一种通式（I）的化合物和/或所述化合物的农业上相容的盐和至少一种液体或固体载体。

公开(公告)号：US20080058352A1

公开(公告)日：2008-03-06

申请号：US10594268

申请日：2005-03-22

Applicant: Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

Inventor： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

IPC: A01N43/56 ,  A01N43/78 ,  A01N43/90

CPC classification number: A01N43/90 ,  A01N2300/00

Abstract: Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) an anilide of the formula II  in which the variables are as defined below: Ar is phenyl or a five- or six-membered aromatic heterocycle which contains one to four heteroatoms selected from the group consisting of O, N and S, where the cycles are unsubstituted or may be substituted by one to three groups R1: R1 is halogen, alkyl or haloalkyl; R is phenyl, alkyl, haloalkyl, alkoxy, haloalkoxy; Q is hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures, and also compositions comprising these mixtures.

Abstract translation: 作为活性组分的杀真菌混合物包括1）式I的三氮代嘧啶衍生物和2）式II的酰苯胺，其中变量如下所定义：Ar是苯基或五或六元芳族杂环，其含有 一至四个选自O，N和S的杂原子，其中循环是未取代的或可以被一至三个R 1取代：R 1是 卤素，烷基或卤代烷基; R是苯基，烷基，卤代烷基，烷氧基，卤代烷氧基; Q是氢，烷基，卤代烷基，烷氧基，卤代烷氧基; 协同有效量的方法，使用化合物I与化合物II的混合物来控制有害真菌，以及使用化合物I与化合物II制备这种混合物，以及包含这些混合物的组合物。

公开(公告)号：US20080051285A1

公开(公告)日：2008-02-28

申请号：US10590363

申请日：2005-03-14

Applicant: Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

Inventor： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC: A01N43/90 ,  A01C1/06

CPC classification number: A01N43/90 ,  A01N43/76 ,  A01N2300/00

Abstract: Fungicidal mixtures for controlling rice pathogens, which mixtures comprise, as active components,1) the triazolopyrimidine derivative of the formula I and2) vinclozolin of the formula II in a synergistically effective amount, methods for controlling rice pathogens using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures, and also compositions comprising these mixtures.

Abstract translation: 用于控制水稻病原体的杀真菌混合物，其混合物包含作为活性组分的1）式I的三氮代嘧啶衍生物和2）协同有效量的式II的连环唑啉，使用化合物I与 化合物II和化合物II与化合物II用于制备这种混合物的用途，以及包含这些混合物的组合物。

公开(公告)号：US07335661B2

公开(公告)日：2008-02-26

申请号：US10532770

申请日：2003-11-14

Applicant: Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schöfl

Inventor： Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schöfl

IPC: A01N43/90 ,  A01N43/40

CPC classification number: A01N43/90 ,  A01N43/40 ,  A01N2300/00

Abstract: Fungicidal mixtures, comprising A) the triazolopyrimidine of the formula I  and B) amide compounds of the formula II where X1 and X2 are halogen, nitro, cyano, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, haloalkoxy, haloalkylthio, alkylsulfinyl or alkylsulfonyl; x is 1, 2, 3 or 4; and y is 1, 2, 3, 4 or 5; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and II for preparing such mixtures are described.

Abstract translation: 杀真菌混合物，其包含A）式I的三唑并嘧啶和B）式II的酰胺化合物，其中X 1和X 2是卤素，硝基，氰基，烷基， 烯基，炔基，卤代烷基，卤代烯基，卤代炔基，烷氧基，卤代烷氧基，卤代烷硫基，烷基亚磺酰基或烷基磺酰基; x为1,2,3或4; y为1,2,3,4或5; 在协同有效量下，描述了使用化合物I和II的混合物来控制有害真菌的方法，包含这些化合物的组合物以及化合物I和II用于制备这种混合物的用途。