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11.Methods for the Preparation of HIV attachment inhibitor piperazine prodrug compound 有权
Title translation: 制备HIV附着抑制剂哌嗪前药化合物的方法公开(公告)号:US09255113B2
公开(公告)日:2016-02-09
申请号:US14516655
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07D471/04 , C07F9/09 , C07F9/6561 , C07C213/08 , C07F1/02 , C07D207/333 , C07D405/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material wherein R7═—H, alkyl, aryl, —SO2R, —C(O)OR, and —C(O)NR2; where R═—H, C1-C6 alkyl, -aryl, and —CH2Aryl.
Abstract translation: 使用其中R 7 = -H,烷基,芳基,-SO 2 R,-C(O)OR和-C(O)NR 2的起始物质来阐述制备该化合物的方法。 其中R = -H,C 1 -C 6烷基, - 芳基和-CH 2芳基。
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公开(公告)号:US20150038710A1
公开(公告)日:2015-02-05
申请号:US14516664
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07F9/09 , C07C213/08
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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公开(公告)号:US20130203992A1
公开(公告)日:2013-08-08
申请号:US13760526
申请日:2013-02-06
Applicant: Bristol-Myers Squibb Company
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07F9/6561 , C07C213/08 , C07D471/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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14.Methods for the preparation of HIV attachment inhibitor piperazine prodrug compound 有权
Title translation: 制备HIV附着抑制剂哌嗪前药化合物的方法公开(公告)号:US09394322B2
公开(公告)日:2016-07-19
申请号:US14516661
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07D405/06 , C07F9/09 , C07F9/6561 , C07D471/04 , C07C213/08 , C07F1/02 , C07D207/333 , C07D405/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
Abstract translation: 使用原料制备化合物的方法
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公开(公告)号:US09249168B2
公开(公告)日:2016-02-02
申请号:US14516669
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07D471/04 , C07F9/09 , C07F9/6561 , C07C213/08 , C07F1/02 , C07D207/333 , C07D405/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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16.Methods for the preparation of HIV attachment inhibitor piperazine prodrug compound 有权
Title translation: 制备HIV附着抑制剂哌嗪前药化合物的方法公开(公告)号:US09243010B2
公开(公告)日:2016-01-26
申请号:US14516641
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07D471/04 , C07F9/09 , C07F9/6561 , C07C213/08 , C07F1/02 , C07D207/333 , C07D405/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A process for the preparation of the compound of Formula I is set forth utilizing the starting compound 1 and the acid chloride compound
Abstract translation: 使用起始化合物1和酰氯化合物来阐述制备式I化合物的方法
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公开(公告)号:US20150038717A1
公开(公告)日:2015-02-05
申请号:US14516655
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07D471/04
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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公开(公告)号:US20150038711A1
公开(公告)日:2015-02-05
申请号:US14516669
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07F9/09
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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公开(公告)号:US20150038709A1
公开(公告)日:2015-02-05
申请号:US14516636
申请日:2014-10-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Martin D. Eastgate , Michael S. Bultman , Ke Chen , Dayne Dustan Fanfair , Richard J. Fox , Thomas E. La Cruz , Boguslaw M. Mudryk , Christina Ann Risatti , James H. Simpson , Maxime C. Soumeillant , Jonathan Clive Tripp , Yi Xiao
IPC: C07F9/6561
CPC classification number: C07D471/04 , C07C213/08 , C07D207/333 , C07D405/04 , C07F1/02 , C07F9/098 , C07F9/650952 , C07F9/6561
Abstract: A method for making the compound is set forth utilizing the starting material
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