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11.
公开(公告)号:US20110306611A1
公开(公告)日:2011-12-15
申请号:US12462405
申请日:2009-08-03
申请人: Michael N. Alekshun , Victor Amoo , Oak K. Kim , Atul K. Verma
发明人: Michael N. Alekshun , Victor Amoo , Oak K. Kim , Atul K. Verma
IPC分类号: A61K31/5377 , C12N1/14 , C12N1/10 , C07H1/00 , A61K31/4184 , C07D235/18 , C07D413/14 , A61K31/422 , C07D261/18 , C07D413/12 , A61K31/454 , C07D211/32 , C07D263/30 , A61K31/427 , C07D277/04 , A61K31/4709 , C07D215/38 , A61K31/497 , A61K31/4196 , C07D249/08 , A61P31/04 , C12N1/20
CPC分类号: A61K31/5377 , A61K31/4184 , A61K31/42 , A61K31/427 , A61K31/4439 , A61K31/4709 , A61K31/496 , C07D235/18 , C07D235/22 , C07D235/24 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , Y02A50/401 , Y02A50/47 , Y02A50/471 , Y02A50/473 , Y02A50/475 , Y02A50/478 , Y02A50/481 , Y02A50/483
摘要: Substituted benzoimidazole compounds useful as anti-infectives that decrease resistance, virulence, or growth of microbes are provided. Methods of making and using substituted benzoimidazole compounds, as well as pharmaceutical preparations thereof, in, e.g., reducing antibiotic resistance and inhibiting biofilms.
摘要翻译: 提供了可用作降低微生物的抗性,毒力或生长的抗感染药物的取代的苯并咪唑化合物。 制备和使用取代的苯并咪唑化合物的方法,以及其药物制剂,例如降低抗生素抗性和抑制生物膜。
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公开(公告)号:US20090170812A1
公开(公告)日:2009-07-02
申请号:US11823103
申请日:2007-06-25
申请人: Michael N. Alekshun , Victoria Bartlett , Lynne Garrity-Ryan , Mark Grier , Oak K. Kim , Atul K. Verma
发明人: Michael N. Alekshun , Victoria Bartlett , Lynne Garrity-Ryan , Mark Grier , Oak K. Kim , Atul K. Verma
IPC分类号: A61K31/675 , C12N1/00 , C07K14/00 , A61K31/4184 , A61K31/437 , A61K31/4196 , A61K31/421 , A61K31/5377 , A61K31/496 , A61K31/4439 , C07D235/04 , C07D471/02 , C07D249/08 , C07D263/30 , C07D413/02 , C07D403/02 , C07D401/02 , C07F9/06 , A01N43/52 , A01N43/40 , A01N43/653 , A01N43/76 , A01N43/84 , A01N43/60 , A01P1/00 , A61P31/00 , A61P13/02
CPC分类号: C07D235/22 , A61K31/4184 , A61K31/4196 , A61K31/422 , A61K31/675 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12 , C07D405/04 , C07D405/12 , C07D413/12 , C07D471/04 , Y02A50/401 , Y02A50/411 , Y02A50/47 , Y02A50/471 , Y02A50/473 , Y02A50/475 , Y02A50/478 , Y02A50/483
摘要: Substituted benzoimidazole compounds useful as anti-infectives that decrease resistance, virulence, or growth of microbes are provided. Methods of making and using substituted benzoimidazole compounds, as well as pharmaceutical preparations thereof, in, e.g., reducing antibiotic resistance and inhibiting biofilms.
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