公开(公告)号：US06369460B1

公开(公告)日：2002-04-09

申请号：US09522618

申请日：2000-03-10

申请人： Takeshi Endoh ,  Kouichi Takagi ,  Keizo Ikeda ,  Kazuhiro Aoki

发明人： Takeshi Endoh ,  Kouichi Takagi ,  Keizo Ikeda ,  Kazuhiro Aoki

IPC分类号： H02J100

CPC分类号： B60R16/03 ,  H02J7/0031 ,  H02J2007/0039 ,  H02J2007/004 ,  Y10T307/406

摘要： A power supply monitoring apparatus, for which a plurality of different preset reference current values and corresponding permitted times are provided, includes: a cutoff device; current detection circuits; overcurrent detection circuits; an idle-up command circuit; and a low voltage detection circuit. When an overcurrent detection circuit detects a current value equaling or exceeding at least one of the preset reference current values, and when that condition continues for a time equaling or exceeding a permitted time corresponding to the pertinent reference current value, the circuit transmits a command to the cutoff device to interrupt the current supplied to a power feeding path. Further, when the idle-up command circuit detects an increase in a supplied current, an idle-up command is issued.

摘要翻译： 提供多个不同的预设基准电流值和相应的允许时间的电源监视装置包括：切断装置; 电流检测电路; 过电流检测电路; 空转命令电路; 和低电压检测电路。 当过电流检测电路检测到等于或超过预设参考电流值中的至少一个的电流值时，并且当该条件持续等于或超过对应于相关参考电流值的允许时间的时间时，电路将命令发送到 所述切断装置中断供给到馈电路径的电流。 此外，当怠速命令电路检测到供给电流的增加时，发出怠速命令。

公开(公告)号：US06316967B1

公开(公告)日：2001-11-13

申请号：US09692144

申请日：2000-10-20

申请人： Kouichi Takagi ,  Takeshi Endoh

发明人： Kouichi Takagi ,  Takeshi Endoh

IPC分类号： H03K5153

CPC分类号： G01R19/165

摘要： When a circuit is activated, bases of transistors Q1 and Q2 making up a first current mirror circuit 7 are grounded through switch means 10, whereby a current is forcibly made to flow into the bases of the transistors Q1 and Q2. Thus, the circuit operation can be made reliable at the activation time. A part of load current is shunted with good accuracy via a resistor R1 having a first resistance value of a predetermined magnification of a resistance value of a shunt resistor Rs, the first current mirror circuit 7, and a second current mirror circuit 8, and the output end of the shunted current is grounded via a resistor R2 having a second resistance value, so that an output voltage VOUT proportional to a load current IL can be obtained with good accuracy from the resistor R2 and the load current IL can be found with good accuracy from the output voltage VOUT.

摘要翻译： 当电路被激活时，构成第一电流镜电路7的晶体管Q1和Q2的基极通过开关装置10接地，由此强制地使电流流入晶体管Q1和Q2的基极。 因此，可以在启动时使电路工作可靠。 负载电流的一部分通过具有分流电阻Rs，第一电流镜电路7和第二电流镜电路8的电阻值的预定放大率的第一电阻值的电阻器R1以良好的精度分流，并且 分流电流的输出端经由具有第二电阻值的电阻R2接地，从而可以从电阻R2获得与负载电流IL成正比的输出电压VOUT，并且可以发现负载电流IL良好 从输出电压VOUT的精度。

公开(公告)号：US20180180360A1

公开(公告)日：2018-06-28

申请号：US15844812

申请日：2017-12-18

申请人： Kiyotada Katoh ,  Tomoyasu Hirasawa ,  Norihiko Aze ,  Takeshi Endoh

发明人： Kiyotada Katoh ,  Tomoyasu Hirasawa ,  Norihiko Aze ,  Takeshi Endoh

IPC分类号： F28D15/04 ,  H01L23/427 ,  F28D20/02 ,  F28D15/02

CPC分类号： F28D15/046 ,  F28D15/0283 ,  F28D15/043 ,  F28D20/023 ,  H01L23/427

摘要： A loop heat pipe wick includes porous rubber.

公开(公告)号：US20130172317A1

公开(公告)日：2013-07-04

申请号：US13814346

申请日：2011-08-09

申请人： Hiroyuki Kai ,  Takayuki Kameyama ,  Tohru Horiguchi ,  Kentaro Asahi ,  Takeshi Endoh ,  Yasuhiko Fujii ,  Takuya Shintani ,  Ken'ichiroh Nakamura ,  Sae Jikihara ,  Tsuyoshi Hasegawa ,  Miho Oohara ,  Yukio Tada ,  Toshikatsu Maki ,  Akira Iida

发明人： Hiroyuki Kai ,  Takayuki Kameyama ,  Tohru Horiguchi ,  Kentaro Asahi ,  Takeshi Endoh ,  Yasuhiko Fujii ,  Takuya Shintani ,  Ken'ichiroh Nakamura ,  Sae Jikihara ,  Tsuyoshi Hasegawa ,  Miho Oohara ,  Yukio Tada ,  Toshikatsu Maki ,  Akira Iida

IPC分类号： C07D251/46 ,  C07D417/12 ,  C07D413/12 ,  C07D405/06 ,  C07D401/14 ,  C07D251/52 ,  C07D405/14 ,  C07D401/12 ,  C07D403/12 ,  C07D403/04 ,  C07D413/14

CPC分类号： C07D251/46 ,  C07D251/52 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D403/04 ,  C07D403/06 ,  C07D403/12 ,  C07D405/06 ,  C07D405/12 ,  C07D405/14 ,  C07D409/06 ,  C07D413/06 ,  C07D413/12 ,  C07D413/14 ,  C07D417/06 ,  C07D417/12 ,  C07D417/14

摘要： The present invention provides novel compounds having a P2X3 and/or P2X2/3 receptor antagonistic effect.A pharmaceutical composition having an analgesic effect or an improving effect of urination disorder comprising a compound of the formula (I): wherein Rh and Rj are taken together to form a bond; Ra and Rb and/or Rd and Re are taken together to form oxo or the like; Rc is hydrogen, substituted or unsubstituted alkyl or the like; Rf is —(CR4aR4b)n—R2; R4a and R4b are hydrogen, substituted or unsubstituted alkyl or the like; R2 is substituted or unsubstituted cycloalkyl or the like; n is an integer of 1 to 4; —Rg is —X—R3; —X— is —O—, —S— or the like; R3 is substituted or unsubstituted cycloalkyl or the like, or its pharmaceutically acceptable salt or a solvate thereof.

摘要翻译： 本发明提供具有P2X3和/或P2X2 / 3受体拮抗作用的新化合物。 一种具有止痛作用或排尿障碍改善作用的药物组合物，其包含式（I）化合物：其中Rh和Rj一起形成键; Ra和Rb和/或Rd和Re一起形成氧代等; Rc是氢，取代或未取代的烷基等; Rf是 - （CR4aR4b）n-R2; R4a和R4b是氢，取代或未取代的烷基等; R2是取代或未取代的环烷基等; n为1〜4的整数， -Rg为-X-R3; -X-是-O-，-S-等; R3是取代或未取代的环烷基等，或其药学上可接受的盐或溶剂合物。

公开(公告)号：US20110319414A1

公开(公告)日：2011-12-29

申请号：US13201209

申请日：2010-02-10

申请人： Hiroyuki Kai ,  Takayuki Kameyama ,  Tsuyoshi Hasegawa ,  MIho Oohara ,  Yukio Tada ,  Takeshi Endoh

发明人： Hiroyuki Kai ,  Takayuki Kameyama ,  Tsuyoshi Hasegawa ,  MIho Oohara ,  Yukio Tada ,  Takeshi Endoh

IPC分类号： A61K31/53 ,  C07D251/46 ,  C07D403/06 ,  A61P7/00 ,  C07D413/12 ,  A61K31/5377 ,  A61P29/00 ,  A61P25/00 ,  C07D251/38 ,  C07D251/52

CPC分类号： C07D251/46 ,  C07D251/16 ,  C07D251/44 ,  C07D251/52 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D403/04 ,  C07D403/06 ,  C07D403/12 ,  C07D405/06 ,  C07D405/12 ,  C07D409/06 ,  C07D413/12

摘要： The present invention provides a novel P2X3 and/or P2X2/3 receptor antagonist.A compound represented by the formula (I); wherein Ra, Rb and Rc are, (a) Ra and Rb are taken together ═Z; and Rc is a group represented by R1c; or (b) Rb and Rc are taken together to form a bond; and Ra is a group represented by —Y—R1a; R1a and R1c are each independently hydrogen, substituted or unsubstituted alkyl, etc.; R2 and R3 are each independently substituted or unsubstituted aryl, etc.; R4a and R4b are each independently hydrogen, substituted or unsubstituted alkyl, etc.; X is —N(R5)—, etc.; R5 is hydrogen, substituted or unsubstituted lower alkyl, etc.; —Y— is —O—, etc.; ═Z is ═O, etc.; and n is an integer of 0 to 4.

摘要翻译： 本发明提供了一种新型的P2X3和/或P2X2 / 3受体拮抗剂。 由式（I）表示的化合物; 其中Ra，Rb和Rc为（a）Ra和Rb一起为= Z; Rc为由R1c表示的基团; 或（b）Rb和Rc一起形成键; 并且R a是由-Y-R 1a表示的基团; R1a和R1c各自独立地为氢，取代或未取代的烷基等; R2和R3各自独立地是取代或未取代的芳基等; R4a和R4b各自独立地为氢，取代或未取代的烷基等; X是-N（R 5） - 等; R5是氢，取代或未取代的低级烷基等; -Y-是-O-等; ═Z是═O等; n为0〜4的整数。

公开(公告)号：US20100099676A1

公开(公告)日：2010-04-22

申请号：US12447743

申请日：2007-10-31

申请人： Takeshi Endoh ,  Yasuhiko Fujii ,  Eiichi Kojima ,  Genta Tadano ,  Naoko Yamaguchi ,  Yo Adachi ,  Sachie Tagashira ,  Yuki Tachibana ,  Naohiro Onodera

发明人： Takeshi Endoh ,  Yasuhiko Fujii ,  Eiichi Kojima ,  Genta Tadano ,  Naoko Yamaguchi ,  Yo Adachi ,  Sachie Tagashira ,  Yuki Tachibana ,  Naohiro Onodera

IPC分类号： A61K31/5377 ,  C07D417/10 ,  A61K31/497 ,  C07D413/14 ,  C07D401/02 ,  C07D413/02 ,  A61K31/4965 ,  C07D241/04

CPC分类号： C07D209/86 ,  C07D211/96 ,  C07D213/81 ,  C07D215/20 ,  C07D241/04 ,  C07D243/08 ,  C07D263/32 ,  C07D277/28 ,  C07D295/22 ,  C07D295/26 ,  C07D307/81 ,  C07D307/91

摘要： A compound represented by the general formula (I): wherein R1 is wherein R26 and R28 are each independently lower alkyloxy and the like; n1 is an integer of 0 to 3; Z is a optionally substituted C1-C5 alkynylene which may be interrupted with a substituent selected from Substituent group a and the like; A is a group represented by the formula: wherein R6 and R7 are each independently lower alkyl and the like; m and n are each independently 0, 1, or 2; R2 is a hydrogen atom and the like; R3 is optionally substituted lower alkyl and the like; R4 is a hydrogen atom; or R3 and R4 may be taken together with an adjacent carbon atom to from a ring; R5 is hydroxyl and the like, or an optically active isomer, a pharmaceutically acceptable salt or a solvate thereof.

摘要翻译： 由通式（I）表示的化合物：其中R 1是其中R 26和R 28各自独立地为低级烷氧基等; n1为0〜3的整数， Z是可以被选自取代基组a等的取代基中断的任选取代的C 1 -C 5亚炔基; A是由下式表示的基团：其中R6和R7各自独立地为低级烷基等; m和n各自独立地为0,1或2; R2是氢原子等; R3是任选取代的低级烷基等; R4是氢原子; 或者R 3和R 4可以与相邻的碳原子一起与环一起取代; R5是羟基等，或光学活性异构体，其药学上可接受的盐或溶剂化物。

公开(公告)号：US06831177B1

公开(公告)日：2004-12-14

申请号：US09980578

申请日：2001-12-03

申请人： Masaaki Uenaka ,  Kyozo Kawata ,  Masahiko Nagai ,  Takeshi Endoh

发明人： Masaaki Uenaka ,  Kyozo Kawata ,  Masahiko Nagai ,  Takeshi Endoh

IPC分类号： C07D24910

CPC分类号： C07D405/06 ,  Y02P20/55

摘要： Industrial and commercial processes for the preparation of 2-acyl-5-benzylfuran derivatives, 1,2,4-triazole-3-carboxylic acid ester derivatives or propenone derivatives having an anti-HIV activity; and useful crystals of the derivatives. A deblocking: (III-2), (IV-10), (VI-1), wherein R1, R2 and R4 are each independently hydrogen or the like; A is CR6 or N; R6 is hydrogen or the like; Q is a protecting group; and L is a leaving group.

摘要翻译： 用于制备2-酰基-5-苄基呋喃衍生物的工业和商业方法，具有抗HIV活性的1,2,4-三唑-3-羧酸酯衍生物或丙烯酮衍生物; 和衍生物的有用晶体。 解封：（III-2），（IV-10），（VI-1）其中R 1，R 2和R 4各自独立地为氢等; A为CR 6或N; R 6是氢等; Q是保护组; 而L是离职团体。

公开(公告)号：US06762277B2

公开(公告)日：2004-07-13

申请号：US10132468

申请日：2002-04-26

申请人： Hiroto Kudoh ,  Takeshi Endoh

发明人： Hiroto Kudoh ,  Takeshi Endoh

IPC分类号： C08G7300

CPC分类号： C07D263/44

摘要： A method of manufacturing a new N-carboxyamino acid anhydride and polyamino acid using a simple process operation. The method for manufacturing N-carboxyamino acid anhydride comprising reacting &agr;-amino acid with di-tert-butyltricarbonate. The method for manufacturing polyamino acid comprising decarboxylating the N-carboxyamino acid anhydride obtained by reacting &agr;-amino acid with di-tert-butyltricarbonate.

摘要翻译： 使用简单的工艺操作制造新的N-羧基氨基酸酐和聚氨基酸的方法。制备N-羧基氨基酸酐的方法，包括使α-氨基酸与二叔丁基三碳酸酯反应。 制备聚氨基酸的方法包括使α-氨基酸与二叔丁基三碳酸酯反应获得的N-羧基氨基酸酐脱羧。

公开(公告)号：US5768902A

公开(公告)日：1998-06-23

申请号：US766315

申请日：1996-12-13

申请人： Masayuki Nonaka ,  Hiroaki Matsushima ,  Kazuhiro Endoh ,  Kensaku Oguni ,  Kazumoto Urata ,  Kyuhei Ishibane ,  Takeshi Endoh

发明人： Masayuki Nonaka ,  Hiroaki Matsushima ,  Kazuhiro Endoh ,  Kensaku Oguni ,  Kazumoto Urata ,  Kyuhei Ishibane ,  Takeshi Endoh

IPC分类号： F25B9/00 ,  F25B13/00 ,  F25B39/04 ,  F25B43/00

CPC分类号： F25B13/00 ,  F25B9/006 ,  F25B2313/0272 ,  F25B2313/02741 ,  F25B2400/16

摘要： A refrigeration cycle comprises a compressor, an indoor heat exchange, an outdoor heat exchanger, a liquid receiver; and a pressure reducer connected in series to form a closed loop. The liquid receiver and the pressure reducer connected in series are connected between the indoor heat exchanger and said outdoor heat exchanger. A non-azeotropic mixture refrigerant comprising at least two kinds of refrigerant of different boiling temperatures mixed together is charged in and circulated through the refrigeration cycle. The mixing ratio of the azeotropic mixture refrigerant circulated thorough the refrigeration cycle is controlled substantially constant.

摘要翻译： 制冷循环包括压缩机，室内热交换器，室外热交换器，液体接收器; 和串联连接形成闭环的减压器。 串联连接的储液器和减压器连接在室内热交换器和室外热交换器之间。 包含混合在一起的不同沸腾温度的至少两种制冷剂的非共沸混合制冷剂被填充并循环通过制冷循环。 通过制冷循环循环的共沸混合制冷剂的混合比例被控制在大致恒定的范围内。

公开(公告)号：US5469067A

公开(公告)日：1995-11-21

申请号：US163572

申请日：1993-12-08

申请人： Takeshi Endoh ,  Tomoaki Imai ,  Mikio Hagiya

发明人： Takeshi Endoh ,  Tomoaki Imai ,  Mikio Hagiya

IPC分类号： G01R31/02 ,  G01R31/08 ,  G01R31/12

CPC分类号： G01R31/083 ,  G01R31/021 ,  G01R31/024 ,  G01R31/1272

摘要： In an electric apparatus such as an electric power cable system, a high frequency pulse is induced on a conductive member such as a metal sheath, where partial discharge occurs in an insulation. The high frequency pulse is detected by means of a bypass lead wire, a metal foil electrode, a detecting coil, and the like provided on the electric apparatus without interrupting a live operation of the electric apparatus.

摘要翻译： 在诸如电力电缆系统的电气设备中，在绝缘体中发生局部放电的金属护套等导电部件上产生高频脉冲。 通过设置在电气设备上的旁路引线，金属箔电极，检测线圈等检测高频脉冲，而不中断电气设备的实时操作。