Herbicidal composition
    11.
    发明授权
    Herbicidal composition 失效
    除草成分

    公开(公告)号:US5312798A

    公开(公告)日:1994-05-17

    申请号:US944084

    申请日:1992-09-11

    CPC分类号: A01N43/78 A01N47/18

    摘要: There is disclosed a herbicidal composition comprising as active ingredients a herbicidally effective amount of (a) an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(C.sub.1 -C.sub.2)alkyl, halo(C.sub.1 -C.sub.2)alkoxy or halo(C.sub.1 -C.sub.2)alkylthio; R.sup.2 is C.sub.1 -c.sub.2 alkyl, chroline, bromine or iodine; R.sup.3 is C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkoxy or C.sub.1 -C.sub.6 alkoxy, all of which are optionally substituted with at least one substituent selected from halogen, C.sub.1 -C.sub.2 alkyl and C.sub.1 -C.sub.2 alkoxy; R.sup.4 is hydrogen or halogen; and (b) at least one of herbicidal triazine compounds, herbicidal uracil compounds, herbicidal urea compounds, herbicidal dinitro aniline compounds, norflurazon, dimethazon, imazaquin and imazethapyr. Also disclosed is a method for controlling undesired weeds by use of the herbicidal composition.

    摘要翻译: 公开了除草组合物,其包含除草有效量的(a)下式的亚氨基噻唑啉化合物:其中R 1是卤素,卤代(C 1 -C 2)烷基,卤代(C 1 -C 2)烷氧基或卤素 (C1-C2)烷硫基; R2是C1-C2烷基,氯原子,溴或碘; R3是C1-C6烷基,C3-C6环烷基,C3-C6环烷氧基或C1-C6烷氧基,它们全部被至少一个选自卤素,C 1 -C 2烷基和C 1 -C 2烷氧基的取代基取代; R4是氢或卤素; 和(b)至少一种除草三嗪化合物,除草尿嘧啶化合物,除草脲化合物,除草二硝基苯胺化合物,诺氟拉津,二甲基噻唑,咪唑啉酮和咪草烟。 还公开了通过使用除草组合物来控制不需要的杂草的方法。

    Iminothiazolines, their production and use as herbicides
    12.
    发明授权
    Iminothiazolines, their production and use as herbicides 失效
    异噻唑啉,其生产和用作除草剂

    公开(公告)号:US5292715A

    公开(公告)日:1994-03-08

    申请号:US936516

    申请日:1992-08-28

    摘要: There is disclosed an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(lower)alkyl, halo(lower)alkoxy or halo(lower)alkylthio; R.sup.2 is methyl, ethyl, chlorine, bromine or iodine; R.sup.3 is lower alkyl, lower cycloalkyl, lower alkoxy, lower cycloalkoxy, lower alkylamino, phenylamino or phenyl, all of which are optionally substituted with at least one substituent selected from halogen, lower alkyl, lower alkoxy, halo(lower)alkyl, lower cycloalkyl and lower cycloalkoxy; and R.sup.4 is hydrogen or halogen. Also disclosed are a process for producing this compound, a herbicidal composition comprising this compound as an active ingredient, and a method for controlling undesired weeds by use of this compound as a herbicide.

    摘要翻译: 公开了下式的亚氨基噻唑啉化合物:(*化学结构*)(I)其中R1是卤素,卤代(低级)烷基,卤代(低级)烷氧基或卤代(低级)烷硫基; R2是甲基,乙基,氯,溴或碘; R3是低级烷基,低级环烷基,低级烷氧基,低级环烷氧基,低级烷基氨基,苯基氨基或苯基,它们全部被至少一个选自卤素,低级烷基,低级烷氧基,卤代(低级)烷基,低级环烷基 和低级环烷氧基; R4是氢或卤素。 还公开了制备该化合物的方法,包含该化合物作为活性成分的除草组合物,以及通过使用该化合物作为除草剂来控制不需要的杂草的方法。

    5-substituted-2,4-diphenylpyrimidine derivatives
    15.
    发明授权
    5-substituted-2,4-diphenylpyrimidine derivatives 失效
    5-取代-2,4-二苯基嘧啶衍生物

    公开(公告)号:US5270467A

    公开(公告)日:1993-12-14

    申请号:US972806

    申请日:1992-11-06

    摘要: A compound is disclosed having the formula: ##STR1## wherein R.sup.1 represents a halo-(C.sub.1 to C.sub.6)-alkoxy group at the ortho or meta position, R.sup.2 and R.sup.3, which may be either the same or different, each represents a hydrogen atom, a halogen atom, a (C.sub.1 to C.sub.2)-alkyl group, a halo-(C.sub.1 to C.sub.2)-alkyl group, a (C.sub.1 to C.sub.2)-alkoxy group, a nitro group, a (C.sub.1 to C.sub.2)-alkylthio group, a halo-(C.sub.1 to C.sub.2)-alkylthio group or a halo-((C.sub.1 to C.sub.2)-alkoxy group, provided that both of R.sup.2 and R.sup.3, if each representing a substituent other than a hydrogen atom, are not at the ortho position for the pyrimidine ring at the same time, and W.sup.1 represents a methanesulfonyl group, or a methylthio group; provided that when W.sup.1 is a methylthio group, R.sup.1, R.sup.2 and R.sup.3 are R.sup.11, R.sup.22 and R.sup.33 wherein R.sup.11 represents a halo-(C.sub.1 to C.sub.6)-alkoxy group at the ortho or meta position, R.sup.22 and R.sup.33, which may be either the same or different, each represents a hydrogen atom, a halogen atom, a (C.sub.1 to C.sub.2)-alkyl group, a halo-(C.sub.1 to C.sub.2)-alkyl group, a (C.sub.1 to C.sub.2)-alkoxy group, or a halo-(C.sub.1 to C.sub.2)-alkoxy group, and both of R.sup.22 and R.sup.33, if each representing a substituent other than a hydrogen atom, are not at the ortho position for the pyrimidine ring at the same time.

    摘要翻译: 公开了具有下式的化合物:其中R1表示邻位或间位的卤代(C1-C6) - 烷氧基,R2和R3可以相同或不同,各自表示 卤素原子,(C1〜C2) - 烷基,卤代(C1〜C2) - 烷基,(C1〜C2) - 烷氧基,硝基,(C1〜C2) (C 1〜C 2) - 烷硫基或卤代((C 1〜C 2) - 烷氧基),条件是如果各自表示除氢原子以外的取代基,则R2和R3均不为 同时在嘧啶环的邻位,W1表示甲磺酰基或甲硫基;条件是当W1是甲硫基时,R1,R2和R3是R11,R22和R33,其中R11表示卤代 - 邻位或间位的(C1-C6) - 烷氧基可以相同或不同,分别表示氢原子,卤原子,(C1-C2) - 烷基, 卤代(C 1〜C 2) - 烷基 (C1〜C2) - 烷氧基或卤代(C1〜C2) - 烷氧基,R22和R33均为氢原子以外的取代基时,不在邻位 嘧啶环同时进行。

    Process for production of fluoroalkane carboxamide derivatives
    17.
    发明授权
    Process for production of fluoroalkane carboxamide derivatives 失效
    氟代烷酰胺衍生物的制备方法

    公开(公告)号:US5484933A

    公开(公告)日:1996-01-16

    申请号:US282562

    申请日:1994-07-29

    IPC分类号: C07D277/46 C07D277/18

    CPC分类号: C07D277/46

    摘要: There is disclosed a process for the production of a fluoroalkanecarboxamide derivative of the formula (I): ##STR1## wherein R.sup.1 is a halogen atom, an alkyl group substituted with at least one halogen atom or an alkoxyl group substituted with at least one halogen atom; R.sup.2 is a hydrogen atom or a halogen atom; and R.sup.3 is a methyl group, an ethyl group, a chlorine atom or a bromine atom; X and Y are the same or different and each of them represents a hydrogen atom, a chlorine atom, a fluorine atom or a trifluoromethyl group, with the proviso that X and Y do not simultaneously represent a hydrogen atom or a chlorine atom, which comprises the steps of:(a) reacting an iminothiazoline compound of the formula (II): ##STR2## wherein R.sup.1, R.sup.2 and R.sup.3 are each as defined above, or a salt thereof with a fluoroolefin of the formula (III):XYC.dbd.CF.sub.2 (III)wherein X and Y are each as defined above, in the presence of a primary or secondary amine; and(b) reacting the resultant reaction mixture with water.

    摘要翻译: 公开了制备式(I)的氟烷烃甲酰胺衍生物的方法:其中R1是卤素原子,被至少一个卤素原子取代的烷基或至少被取代的烷氧基的式 一个卤素原子; R2是氢原子或卤素原子; 且R 3为甲基,乙基,氯原子或溴原子; X和Y相同或不同,它们各自表示氢原子,氯原子,氟原子或三氟甲基,条件是X和Y不同时表示氢原子或氯原子,其包括 步骤:(a)使式(II)的亚氨基噻唑啉化合物:其中R 1,R 2和R 3各自如上所定义,或其盐与式(III)的氟代烯烃反应: XYC = CF 2(III)其中X和Y各自如上所定义,在伯胺或仲胺的存在下; 和(b)使所得反应混合物与水反应。

    Process of producing iminothiazoline derivatives
    19.
    发明授权
    Process of producing iminothiazoline derivatives 失效
    生产亚氨基噻唑啉衍生物的方法

    公开(公告)号:US5360912A

    公开(公告)日:1994-11-01

    申请号:US17259

    申请日:1993-02-12

    IPC分类号: C07D277/40

    CPC分类号: C07D277/40

    摘要: There is disclosed a process for producing an iminothiazoline derivative of the general formula: ##STR1## wherein R.sup.1 is halogen, halo(lower)alkyl, halo(lower)alkoxy or halo(lower)alkylthio; R.sup.2 is hydrogen or halogen; and R.sup.4 is hydrogen or lower alkyl. This compound (I) can be obtained by cyclization of a thiourea derivative of the general formula: ##STR2## wherein R.sup.1, R.sup.2 and R.sup.4 are each the same as defined above, and R.sup.3 is hydrogen or (lower)alkylcarbonyl optionally substituted with at least one substituent selected from the group consisting of halogen, lower alkyl and lower alkoxy.

    摘要翻译: 公开了一种制备下列通式的亚氨基噻唑啉衍生物的方法:其中R 1是卤素,卤代(低级)烷基,卤代(低级)烷氧基或卤代(低级)烷硫基)。 R2是氢或卤素; R4是氢或低级烷基。 该化合物(I)可以通过下列通式的硫脲衍生物的环化得到:其中R 1,R 2和R 4各自与上述相同,且R 3是氢或(低级)烷基羰基任意取代 与至少一个选自卤素,低级烷基和低级烷氧基的取代基取代。