Substituted 1,8-naphthyridines, their preparation and their use as
antidotes
    21.
    发明授权
    Substituted 1,8-naphthyridines, their preparation and their use as antidotes 失效
    取代的1,8-萘啶,其制备及其用作解毒剂

    公开(公告)号:US5258356A

    公开(公告)日:1993-11-02

    申请号:US13202

    申请日:1993-02-01

    IPC分类号: A01N25/32 C07D471/04

    CPC分类号: C07D471/04 A01N25/32

    摘要: A combination of a variety of herbicides with safening agents which are substituted 1,8-naphthyridines of the formula ##STR1## where R.sup.1 is mercapto, hydroxyl, halogen, benzylthio, amino or NR.sup.2 R.sup.3, whereR.sup.2 is a group ##STR2## where A is C.sub.1 -C.sub.8 -alkyl, R.sup.3 is hydrogen, XR.sup.4, where X is oxygen or sulfur and R.sup.4 is C.sub.1 -C.sub.12 -alkyl,R.sup.5 and R.sup.7 are each hydrogen, C.sub.1 -C.sub.12 -alkyl, hydroxyl, halogen, mercapto, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, dialkylamino where each alkyl is of 1 to 6 carbon atoms, phenoxy or phenylthio, halo-(C.sub.1 -C.sub.3)-alkyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.3)-alkyl, andR.sup.6 is hydrogen, C.sub.1 -C.sub.12 -alkyl, carboxyl or C.sub.1 -C.sub.4 -alkoxycarbonyl or the plant-tolerated salts thereof.

    摘要翻译: 各种除草剂与安全剂的组合,其为R1为巯基,羟基,卤素,苄硫基,氨基或NR2R3的式VIII取代的1,8-萘啶,其中R2为基团,其中A 是C 1 -C 8 - 烷基,R 3是氢,XR 4,其中X是氧或硫,R 4是C 1 -C 12烷基,R 5和R 7各自是氢,C 1 -C 12烷基,羟基,卤素,巯基,C 1 -C 4 - 烷氧基,C 1 -C 4烷氧基 - (C 1 -C 3) - 烷基,和C 1 -C 4 - 烷氧基 - (C 1 -C 3) - 烷基, R6是氢,C1-C12-烷基,羧基或C1-C4-烷氧基羰基或其植物耐受的盐。

    5-amino-6-pyridazone derivatives, their preparation and herbicidal
mixtures containing these derivatives
    26.
    发明授权
    5-amino-6-pyridazone derivatives, their preparation and herbicidal mixtures containing these derivatives 失效
    5-氨基-6-吡啶酮衍生物,其制备和除草剂混合物含有这些衍生物

    公开(公告)号:US5123952A

    公开(公告)日:1992-06-23

    申请号:US378798

    申请日:1989-07-12

    摘要: 5-Amino-6-pyridazones of the general formulae Ia and Ib ##STR1## where R.sup.1 is C.sub.1 -C.sub.4 -alkyl which may carry up to three halogen atoms, R.sup.2 is C.sub.1 -C.sub.4 -alkyl or C.sub.3 -C.sub.6 -alkenyl, where these groups may carry up to two phenyl radicals, or C.sub.3 -C.sub.6 -alkynyl, A is --CO-- or --SO.sub.2 --, B is C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, where these groups may carry up to three of the following radicals: halogen, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio and/or phenyl; an isocyclic or heterocyclic C.sub.3 -C.sub.7 -cycloalkyl group or an isocyclic or heterocyclic C.sub.3 -C.sub.7 -cycloalkenyl group, where these groups may be fused with one or two cycloalkyl groups of this type or with one or two benzene nuclei, where the total number of ring members is from 3 to 16 and these cyclic radicals may carry up to three of the following groups: halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 - C.sub.6 -alkynyl and/or phenyl; a mononuclear to trinuclear aromatic or heteroaromatic radical which may carry up to three of the following groups: C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -alkylsulfinyl, C.sub.1 -C.sub.4 -alkylsulfonyl, cyano, nitro, carbo-C.sub.1 -C.sub.4 -alkoxy, N,N-di-C.sub.1 -C.sub.4 -alkylcarbamido and/or halogen.These compounds are used as herbicidal active ingredients.

    摘要翻译: 通式Ia和Ib的5-氨基-6-哒嗪酮其中R 1是可以带有三个卤素原子的C 1 -C 4 - 烷基,R 2是C 1 -C 4 - 烷基或C 3 -C 6 - 烯基,其中这些基团可以带有两个苯基或C 3 -C 6 - 炔基,A是-CO-或-SO 2 - ,B是C 1 -C 6 - 烷基,C 2 -C 6 - 烯基或C 2 -C 6 - 炔基 其中这些基团可以带有三个以下基团:卤素,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基和/或苯基; 一个环状或杂环的C 3 -C 7 - 环烷基或者是一个或多个杂环的C 3 -C 7 - 环烯基,其中这些基团可以与一个或两个这样的环烷基或一个或两个苯核稠合, 环成员为3至16,并且这些环状基团可以带有三个以下基团:卤素,C 1 -C 4 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基和/或苯基; 可以携带三个以下基团的单核到三核芳族或杂芳族基团:C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 C 1-4烷基亚磺酰基,C 1 -C 4 - 烷基磺酰基,氰基,硝基,C 1 -C 4 - 烷氧基,N,N-二-C 1 -C 4烷基氨基甲酰基和/或卤素。 这些化合物用作除草活性成分。

    Thiophene-2-carboxylic acid derivatives, their preparation and their use
for controlling undesirable plant growth
    28.
    发明授权
    Thiophene-2-carboxylic acid derivatives, their preparation and their use for controlling undesirable plant growth 失效
    噻吩-2-羧酸衍生物,其制备及其用于控制​​不期望的植物生长的用途

    公开(公告)号:US5034049A

    公开(公告)日:1991-07-23

    申请号:US463163

    申请日:1990-01-09

    CPC分类号: C07D333/38 A01N43/10

    摘要: Thiophene-2-carboxylic acid derivatives of the general formula I ##STR1## where R.sup.1 to R.sup.3 are each hydrogen, halogen, branched or straight-chain C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.8 -alkoxy, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -haloalkoxy, nitro, cyano, unsubstituted phenyl or phenyl which is mono- to trisubstituted by C.sub.1 -C.sub.4 -alkyl, halogen, C.sub.1 -C.sub.5 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.5 -haloalkoxy;X is --OR.sup.4 or --NH--OR.sup.5,R.sup.4 being branched or straight-chain C.sub.3 -C.sub.10 -alkynylalkyl which is unsubstituted or substituted by halogen; andR.sup.5 being branched or straight-chain C.sub.1 -C.sub.5 -alkyl which is unsubstituted or substituted by halogen, or branched or straight-chain C.sub.3 -C.sub.10 -alkynylalkyl which is unsubstituted or substituted by halogen;with the proviso that R.sup.4 is not propargyl when R.sup.2 and R.sup.3 are both hydrogen or when R.sup.2 is halogen or R.sup.3 is chlorine, methyl or methoxy.The compounds I are suitable for combating the growth of unwanted plants.

    摘要翻译: 通式I的噻吩-2-羧酸衍生物其中R 1至R 3各自为氢,卤素,支链或直链C 1 -C 6 - 烷基,C 1 -C 8 - 烷氧基,C 1 -C 6 - 卤代烷基,C 1 C 1-6卤代烷氧基,硝基,氰基,未取代的苯基或被C 1 -C 4 - 烷基,卤素,C 1 -C 5 - 卤代烷基,C 1 -C 4 - 烷氧基或C 1 -C 5 - 卤代烷氧基单 - X为-OR4或-NH-OR5,R4为未取代或被卤素取代的支链或直链C 3 -C 10 - 炔基烷基; 并且R 5是未被取代或被卤素取代的支链或直链C 1 -C 5 - 烷基,或未被取代或被卤素取代的支链或直链C 3 -C 10 - 炔基烷基; 条件是当R 2和R 3均为氢时或R 2为卤素或R 3为氯,甲基或甲氧基时,R 4不是炔丙基。 化合物I适用于对抗不想要的植物的生长。